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Václav Němec

czech academy of sciences

15H指数
89论文数
717被引数
收录论文 10
发表时间
The Use of Composite 3D Printing in the Design of Optomechanical Components
err2025-11-03
err0
errOAAI
errNemcova, Sarka; Hermanek, Jan; Crha, Pavel; Macuchova, Karolina; Nemec, Vaclav; Poboril, Radek; Tichy, Tomas; Uher, Ondrej; Smrz, Martin; Mocek, Tomas
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Discovery of an Exquisitely Selective WDR5 Chemical Probe Accelerated by a High-Quality DEL-ML Hit由高质量DEL-ML命中加速的精美选择性WDR5化学探针的发现
err2025-08-06
err0
errOAAI
errLasse Hoffmann; Christopher Lenz; Frederic Farges; Serah W. Kimani; Johannes Dopfer; Sabrina Keller; Martin P. Schwalm; Hanna Holzmann; Andreas Krämer; Aiping Dong; Fengling Lu; Irene Chau; Levon Halebelian; Matthias Gstaiger; Susanne Müller; Stefan Knapp; Vaclav Nemec
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Workflow for E3 Ligase Ligand Validation for PROTAC Development
err2025-02-11
err0
errOAAI
errMiletic, Nebojsa; Weckesser, Janik; Mosler, Thorsten; Rathore, Rajeshwari; Hoffmann, Marina E.; Gehrtz, Paul; Schlesiger, Sarah; Hartung, Ingo V.; Berner, Nicola; Wilhelm, Stephanie; Mueller, Juliane; Adhikari, Bikash; Nemec, Vaclav; Sivashanmugam, Saran Aswathaman; Elson, Lewis; Holzmann, Hanna; Schwalm, Martin P.; Hoffmann, Lasse; Azeez, Kamal Rayees Abdul; Mueller, Susanne; Kuster, Bernhard; Wolf, Elmar; Dikic, Ivan; Knapp, Stefan
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Development and Discovery of a Selective Degrader of Casein Kinases 1 δ/ε一种选择性降解CK1 δ/ε的降解剂的研发与发现
err2024-12-27
err0
PREAI
errHaag, Adrian; Nemec, Vaclav; Janovska, Pavlina; Bartosikova, Jana; Adhikari, Bikash; Mueller, Juliane; Schwalm, Martin P.; Cada, Stepan; Ohmayer, Uli; Daub, Henrik; Kim, Yeojin; Born, Florian; Wolf, Elmar; Bryja, Vitezslav
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Discovery of Two Highly Selective Structurally Orthogonal Chemical Probes for Activin Receptor-like Kinases 1 and 2
err2024-07-18
err0
errOAAI
errNemec, Vaclav; Remes, Marek; Benovsky, Petr; Boeck, Michael C.; Srankova, Eliska; Wong, Jong Fu; Cros, Julien; Williams, Eleanor; Tse, Lap Hang; Smil, David; Ensan, Deeba; Isaac, Methvin B.; Al-Awar, Rima; Gomolkova, Regina; Ursachi, Vlad-Constantin; Fafilek, Bohumil; Kahounova, Zuzana; Vichova, Rachel; Vacek, Ondrej; Berger, Benedict-Tilman; Wells, Carrow I.; Corona, Cesear R.; Vasta, James D.; Robers, Matthew B.; Krejci, Pavel; Soucek, Karel; Bullock, Alex N.; Knapp, Stefan; Paruch, Kamil
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A C-Degron Structure-Based Approach for the Development of Ligands Targeting the E3 Ligase TRIM7
err2024-06-27
err1
PREAI
errSosa, Christian J. Munoz; Lenz, Christopher; Hamann, Anton; Farges, Frederic; Dopfer, Johannes; Kraemer, Andreas; Cherkashyna, Veronika; Tarnovskiy, Andrey; Moroz, Yurii S.; Proschak, Ewgenij; Nemec, Vaclav; Mueller, Susanne; Saxena, Krishna; Knapp, Stefan
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Discovery of Potent and Exquisitely Selective Inhibitors of Kinase CK1 with Tunable Isoform Selectivity
err2023-02-02
err5
PREAI
errNemec, Vaclav; Khirsariya, Prashant; Janovska, Pavlina; Moyano, Paula Martin; Maier, Lukas; Prochazkova, Petra; Kebkova, Pavlina; Gybel', Tomas; Berger, Benedict-Tilman; Chaikuad, Apirat; Reinecke, Maria; Kuster, Bernhard; Knapp, Stefan; Bryja, Vitezslav; Paruch, Kamil
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A Chemical Toolbox for Labeling and Degrading Engineered Cas Proteins
errJACS AU
IF8.7
err2021-05-12
err14
errOAAI
errGama-Brambila, Rodrigo A.; Chen, Jie; Dabiri, Yasamin; Tascher, Georg; Nemec, Vaclav; Muench, Christian; Song, Guangqi; Knapp, Stefan; Cheng, Xinlai
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Highly selective inhibitors of protein kinases CLK and HIPK with the furo[3,2-b]pyridine core
err2021-04-01
err21
PREAI
errNemec, Vaclav; Maier, Lukas; Berger, Benedict-Tilman; Chaikuad, Apirat; Drapela, Stanislav; Soucek, Karel; Knapp, Stefan; Paruch, Kamil
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Site-Specific Analysis of Protein Hydration Based on Unnatural Amino Acid Fluorescence
err2015-04-09
err32
PREAI
errAmaro, Mariana; Brezovsky, Jan; Kovacova, Silvia; Sykora, Jan; Bednar, David; Nemec, Vaclav; Liskova, Veronika; Kurumbang, Nagendra Prasad; Beerens, Koen; Chaloupkova, Radka; Paruch, Kamil; Hof, Martin; Damborsky, Jiri
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