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Development of Urea-Bond-Containing Michael Acceptors as Antitrypanosomal Agents Targeting Rhodesain Previti, Santo; Ettari, Roberta; Calcaterra, Elsa; Di Chio, Carla; Ravichandran, Rahul; Zimmer, Collin; Hammerschmidt, Stefan; Wagner, Annika; Bogacz, Marta; Cosconati, Sandro; Schirmeister, Tanja; Zappala, Maria 分享 收藏
Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense Di Chio, Carla; Previti, Santo; Amendola, Giorgio; Ravichandran, Rahul; Wagner, Annika; Cosconati, Sandro; Hellmich, Ute A.; Schirmeister, Tanja; Zappala, Maria; Ettari, Roberta 分享 收藏
Fluorovinylsulfones and -Sulfonates as Potent Covalent Reversible Inhibitors of the Trypanosomal Cysteine Protease Rhodesain: Structure-Activity Relationship, Inhibition Mechanism, Metabolism, and In Vivo Studies Jung, Sascha; Fuchs, Natalie; Johe, Patrick; Wagner, Annika; Diehl, Erika; Yuliani, Tri; Zimmer, Collin; Barthels, Fabian; Zimmermann, Robert A.; Klein, Philipp; Waigel, Waldemar; Meyr, Jessica; Opatz, Till; Tenzer, Stefan; Distler, Ute; Raeder, Hans-Joachim; Kersten, Christian; Engels, Bernd; Hellmich, Ute A.; Klein, Jochen; Schirmeister, Tanja 分享 收藏
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Naphthoquinones as Covalent Reversible Inhibitors of Cysteine Proteases-Studies on Inhibition Mechanism and Kinetics Klein, Philipp; Barthels, Fabian; Johe, Patrick; Wagner, Annika; Tenzer, Stefan; Distler, Ute; Thien Anh Le; Schmid, Paul; Engel, Volker; Engels, Bernd; Hellmich, Ute A.; Opatz, Till; Schirmeister, Tanja 分享 收藏
New Cysteine Protease Inhibitors: Electrophilic (Het)arenes and Unexpected Prodrug Identification for the Trypanosoma Protease Rhodesain Klein, Philipp; Johe, Patrick; Wagner, Annika; Jung, Sascha; Kuehlborn, Jonas; Barthels, Fabian; Tenzer, Stefan; Distler, Ute; Waigel, Waldemar; Engels, Bernd; Hellmich, Ute A.; Opatz, Till; Schirmeister, Tanja 分享 收藏
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Inhibitor-Induced Dimerization of an Essential Oxidoreductase from African Trypanosomes Wagner, Annika; Thien Anh Le; Brennich, Martha; Klein, Philipp; Bader, Nicole; Diehl, Erika; Paszek, Daniel; Weickhmann, A. Katharina; Dirdjaja, Natalie; Krauth-Siegel, R. Luise; Engels, Bernd; Opatz, Till; Schindelin, Hermann; Hellmich, Ute A. 分享 收藏
Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain-2 for the Treatment of Neglected Tropical Diseases (NTDs) Previti, Santo; Ettari, Roberta; Cosconati, Sandro; Arnendola, Giorgio; Chouchene, Khawla; Wagner, Annika; Hellmich, Ute A.; Ulrich, Kathrin; Krauth-Siegel, R. Luise; Wich, Peter R.; Schmid, Ira; Schirmeister, Tanja; Gut, Jiri; Rosenthal, Philip J.; Grasso, Silvana; Zappala, Maria 分享 收藏
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Natural killer cell-mediated lysis of hepatoma cells via specific induction of NKG2D Ligands by the histone deacetylase inhibitor sodium valproate Armeanu, S; Bitzer, M; Lauer, UM; Venturelli, S; Pathil, A; Krusch, M; Kaiser, S; Jobst, K; Smirnow, I; Wagner, A; Steinle, A; Salih, HR 分享 收藏
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