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收藏LRRC8A drives NADPH oxidase-mediated mitochondrial dysfunction and inflammation in allergic rhinitis
Meng, Linghui; Hao, Dingqian; Liu, Yuan; Yu, Peng; Luo, Jinfeng; Li, Chunhao; Jiang, Tianjiao; Yu, Jinzhuang; Zhang, Qian; Liu, Shengyang; Shi, Li
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收藏Pyrido[2, 3-d]pyrimidin-7(8H)-ones as new selective orally bioavailable Threonine Tyrosine Kinase (TTK) inhibitors
Huang, Minhao; Huang, Yongjun; Guo, Jing; Yu, Lei; Chang, Yu; Wang, Xiaolu; Luo, Jinfeng; Huang, Yanhui; Tu, Zhengchao; Lu, Xiaoyun; Xu, Yong; Zhang, Zhimin; Zhang, Zhang; Ding, Ke
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收藏Design and Optimization of 3′-(Imidazo[1,2-α]pyrazin-3-yl)-[1,1′-biphenyl]-3-carboxamides as Selective DDR1 Inhibitors
Mo, Cheng; Zhang, Zhang; Li, Yupeng; Huang, Minhao; Zou, Jian; Luo, Jinfeng; Tu, Zheng-Chao; Xu, Yong; Ren, Xiaomei; Ding, Ke; Lu, Xiaoyun
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收藏2-Amino-2,3-dihydro-1H-indene-5-carboxamide-Based Discoidin Domain Receptor 1 (DDR1) Inhibitors: Design, Synthesis, and in Vivo Antipancreatic Cancer Efficacy
Zhu, Dongsheng; Huang, Huocong; Pinkas, Daniel M.; Luo, Jinfeng; Ganguly, Debolina; Fox, Alice E.; Arner, Emily; Xiang, Qiuping; Tu, Zheng-Chao; Bullock, Alex N.; Brekken, Rolf A.; Ding, Ke; Lu, Xiaoyun
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收藏Design, Synthesis, and Structure-Activity Relationships of 1,2,3-Triazole Benzenesulfonamides as New Selective Leucine-Zipper and Sterile-α Motif Kinase (ZAK) Inhibitors
Yang, Jianzhang; Shibu, Marthandam Asokan; Kong, Lulu; Luo, Jinfeng; BadrealamKhan, Farheen; Huang, Yanhui; Tu, Zheng-Chao; Yun, Cai-Hong; Huang, Chih-Yang; Ding, Ke; Lu, Xiaoyun
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收藏Quinolone antibiotic derivatives as new selective Axl kinase inhibitors
Tan, Li; Zhang, Zhang; Gao, Donglin; Chan, Shingpan; Luo, Jinfeng; Tu, Zheng-Chao; Zhang, Zhi-Min; Ding, Ke; Ren, Xiaomei; Lu, Xiaoyun
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收藏Design, Synthesis, and Biological Evaluation of 3-(Imidazo[1,2-a]pyrazin-3-ylethynyl)-4-isopropyl-N-(3-((4-methylpiperazin-1-yl)methyl)-5-(trifluoromethyl)phenyl)benzamide as a Dual Inhibitor of Discoidin Domain Receptors 1 and 2
Wang, Zhen; Zhang, Yali; Pinkas, Daniel M.; Fox, Alice E.; Luo, Jinfeng; Huang, Huocong; Cui, Shengyang; Xiang, Qiuping; Xu, Tingting; Xun, Qiuju; Zhu, Dongsheng; Tu, Zhengchao; Ren, Xiaomei; Brekken, Rolf A.; Bullock, Alex N.; Liang, Guang; Ding, Ke; Lu, Xiaoyun
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收藏Design, Synthesis, and Structure-Activity Relationship Study of 2-Oxo-3,4-dihydropyrimido[4,5-d]pyrimidines as New Colony Stimulating Factor 1 Receptor (CSF1R) Kinase Inhibitors
Xun, Qiuju; Zhang, Zhang; Luo, Jinfeng; Tong, Linjiang; Huang, Minhao; Wang, Zhen; Zou, Jian; Liu, Yingqiang; Xu, Yong; Xie, Hua; Tu, Zheng-Chao; Lu, Xiaoyun; Ding, Ke
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收藏Design, synthesis, and biological evaluation of novel highly selective polo-like kinase 2 inhibitors based on the tetrahydropteridin chemical scaffold
Zhan, Mei-Miao; Yang, Yang; Luo, Jinfeng; Zhang, Xing-Xing; Xiao, Xuan; Li, Shiyu; Cheng, Kai; Xie, Zhouling; Tu, Zhengchao; Liao, Chenzhong
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收藏EpCAM aptamer-functionalized polydopamine-coated mesoporous silica nanoparticles loaded with DM1 for targeted therapy in colorectal cancerEpCAM适配体功能化聚多巴胺包覆介孔二氧化硅纳米粒子负载DM1在结直肠癌靶向治疗中的应用
Li, Yang; Duo, Yanhong; Bao, Shiyun; He, Lisheng; Ling, Kai; Luo, Jinfeng; Zhang, Yue; Huang, Hao; Zhang, Han; Yu, Xiaofang
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收藏2-Oxo-3, 4-dihydropyrimido[4, 5-d]pyrimidinyl derivatives as new irreversible pan fibroblast growth factor receptor (FGFR) inhibitors
Li, Xueqiang; Guise, Christopher P.; Taghipouran, Rana; Yosaatmadja, Yuliana; Ashoorzadeh, Amir; Paik, Woo-Kyong; Squire, Christopher J.; Jiang, Shuang; Luo, Jinfeng; Xu, Yong; Tu, Zheng-Chao; Lu, Xiaoyun; Ren, Xiaomei; Patterson, Adam V.; Smaill, Jeff B.; Ding, Ke
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收藏Structure Based Design of N-(3-((1H-Pyrazolo[3,4-b]pyridin-5-yl)ethynyl)benzenesulfonamides as Selective Leucine-Zipper and Sterile-α Motif Kinase (ZAK) Inhibitors
Chang, Yu; Lu, Xiaoyun; Shibu, Marthandam Asokan; Dai, Yi-Bo; Luo, Jinfeng; Zhang, Yan; Li, Yingjun; Zhao, Peng; Zhang, Zhang; Xu, Yong; Tu, Zheng-Chao; Zhang, Qing-Wen; Yun, Cai-Hong; Huang, Chih-Yang; Ding, Ke
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收藏2-Aminopyrimidine Derivatives as New Selective Fibroblast Growth Factor Receptor 4 (FGFR4) Inhibitors
Mo, Cheng; Zhang, Zhang; Guise, Christopher P.; Li, Xueqiang; Luo, Jinfeng; Tu, Zhengchao; Xu, Yong; Patterson, Adam V.; Smaill, Jeff B.; Ren, Xiaomei; Lu, Xiaoyun; Ding, Ke
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