Backbone Modification Provides a Long-Acting Inverse Agonist of Pathogenic, Constitutively Active PTH1R VariantsJOURNAL OF THE AMERICAN CHEMICAL SOCIETYIF15.62024-02-281PRE
The mechanism of thia-Michael addition catalyzed by LanC enzymesPROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICAIF9.12023-01-129OAAI
Altered signaling at the PTH receptor via modified agonist contacts with the extracellular domain provides a path to prolonged agonism in vivoPROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICAIF9.12022-11-214OAAI
Spatial bias in cAMP generation determines biological responses to PTH type 1 receptor activationSCIENCE SIGNALINGIF6.62021-10-0541OA
Gq/11-dependent regulation of endosomal cAMP generation by parathyroid hormone class B GPCRPROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICAIF9.12020-03-1735OAAI
Preparation of β2-Homologous Amino Acids Bearing Polar Side Chains via a Collective Synthesis StrategyJOURNAL OF ORGANIC CHEMISTRYIF3.62020-01-1012OAAI
Use of Backbone Modification To Enlarge the Spatiotemporal Diversity of Parathyroid Hormone Receptor-1 Signaling via Biased AgonismJOURNAL OF THE AMERICAN CHEMICAL SOCIETYIF15.62019-09-0928OAAI
Receptor selectivity from minimal backbone modification of a polypeptide agonist多肽激动剂的最小主链修饰的受体选择性PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICAIF9.12018-11-1527OAAI
Synthesis of 2-Thio-Substituted-Benzothiazoles via a Domino Condensation/S-Arylation/Heterocyclization ProcessJOURNAL OF ORGANIC CHEMISTRYIF3.62011-04-2974PRE
Domino Condensation/S-Arylation/Heterocyclization Reactions: Copper-Catalyzed Three-Component Synthesis of 2-N-Substituted BenzothiazolesANGEWANDTE CHEMIE-INTERNATIONAL EDITIONIF16.92010-12-22160PREAI
Facile Benzo-Ring Construction via Palladium-Catalyzed Functionalization of Unactivated sp3 C-H Bonds under Mild Reaction ConditionsORGANIC LETTERSIF52010-06-28147PREAI