未登录Discovery of Novel TLR7 Agonists as Systemic Agent for Combination With aPD1 for Use in Immuno-oncology
Poudel, Yam B.; He, Liqi; Cox, Matthew; Zhang, Qian; Johnson, Walter L.; Cong, Qiang; Cheng, Heng; Chowdari, Naidu S.; Tarby, Christine; Donnell, Andrew F.; Broekema, Matthais; O'Malley, Daniel P.; Zhang, Yong; Subbaiah, Murugaiah A. M.; Kumar, Boda Vijay; Subramani, Lakshumanan; Wang, Bei; Li, Yi-Xin; Sivaprakasam, Prasanna; Critton, David; Mulligan, Dawn; Sandhu, Bhupindar; Xie, Chunshan; Ramakrishnan, Radha; Nagar, Jignesh; Dudhgaonkar, Shailesh; Oderinde, Martins S.; Murtaza, Anwar; Schieven, Gary L.; Mathur, Arvind; Gavai, Ashvinikumar V.; Vite, Gregory; Gangwar, Sanjeev
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收藏DNA-Model-Based Design and Execution of Some Fused Benzodiazepine Hybrid Payloads for Antibody-Drug Conjugate Modality
Sivaprakasam, Prasanna; McDonald, Ivar; Iwuagwu, Christiana; Chowdari, Naidu S.; Peese, Kevin M.; Langley, David R.; Cheng, Heng; Luzung, Michael R.; Schmidt, Michael A.; Zheng, Bin; Tan, Yichen; Cho, Patricia; Rakshit, Souvik; Lakshminarasimhan, Thirumalai; Guturi, Sivakrishna; Kanagavel, Kishorekumar; Kanusu, Umamaheswararao; Niyogi, Ankita G.; Sidhar, Somprabha; Vaidyanathan, Rajappa; Eastgate, Martin D.; Kotapati, Srikanth; Deshpande, Madhura; Pan, Chin; Cardarelli, Pina M.; Xie, Chunshan; Rao, Chetana; Holder, Patrick; Sarma, Ganapathy; Vite, Gregory; Gangwar, Sanjeev
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收藏Design, Synthesis, and Structure-Activity Relationships of Novel Tetrahydroisoquinolino Benzodiazepine Dimer Antitumor Agents and Their Application in Antibody-Drug Conjugates
Chowdari, Naidu S.; Zhang, Yong; McDonald, Ivar; Johnson, Walter; Langley, David R.; Sivaprakasam, Prasanna; Mate, Robert; Huynh, Tram; Kotapati, Srikanth; Deshpande, Madhura; Pan, Chin; Menezes, Daniel; Wang, Yichong; Rao, Chetana; Sarma, Ganapathy; Warrack, Bethanne M.; Rangan, Vangipuram S.; Mei-Chen, Sung; Cardarelli, Pina; Deshpande, Shrikant; Passmore, David; Rampulla, Richard; Mathur, Arvind; Borzilleri, Robert; Rajpal, Arvind; Vite, Gregory; Gangwar, Sanjeev
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收藏Total Synthesis of Meayamycin and O-Acyl Analogues
Gartshore, Christopher; Tadano, Shinji; Chanda, Prem B.; Sarkar, Anindya; Chowdari, Naidu S.; Gangwar, Sanjeev; Zhang, Qian; Vite, Gregory D.; Momirov, Jelena; Boger, Dale L.
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收藏Chemical Modification of Linkers Provides Stable Linker-Payloads for the Generation of Antibody-Drug Conjugates接头的化学修饰为抗体-药物缀合物的产生提供了稳定的接头-有效载荷
Poudel, Yam B.; Chowdari, Naidu S.; Cheng, Heng; Iwuagwu, Christiana I.; King, H. Dalton; Kotapati, Srikanth; Passmore, David; Rampulla, Richard; Mathur, Arvind; Vite, Gregory; Gangwar, Sanjeev
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收藏Universal Affinity Capture Liquid Chromatography-Mass Spectrometry Assay for Evaluation of Biotransformation of Site-Specific Antibody Drug Conjugates in Preclinical Studies
Kotapati, Srikanth; Passmore, David; Yamazoe, Sayumi; Sanku, Rajesh Kishore Kumar; Cong, Qiang; Poudel, Yam B.; Chowdari, Naidu S.; Gangwar, Sanjeev; Rao, Chetana; Rangan, Vangipuram S.; Cardarelli, Pina M.; Deshpande, Shrikant; Strop, Pavel; Dollinger, Gavin; Rajpal, Arvind
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收藏Streamlined Total Synthesis of Uncialamycin and Its Application to the Synthesis of Designed Analogues for Biological Investigations
Nicolaou, K. C.; Wang, Yanping; Lu, Min; Mandal, Debashis; Pattanayak, Manas R.; Yu, Ruocheng; Shah, Akshay A.; Chen, Jason S.; Zhang, Hongjun; Crawford, James J.; Pasunoori, Laxman; Poudel, Yam B.; Chowdari, Naidu S.; Pan, Chin; Nazeer, Ayesha; Gangwar, Sanjeev; Vite, Gregory; Pitsinos, Emmanuel N.
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