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WLB-87848, a Selective σ1 Receptor Agonist, with an Unusually Positioned NH Group as Positive Ionizable Moiety and Showing Neuroprotective Activity Christmann, Ute; Garriga, Lourdes; Llorente, Ana Virginia; Diaz, Jose Luis; Pascual, Rosalia; Bordas, Magda; Dordal, Albert; Porras, Monica; Yeste, Sandra; Reinoso, Raquel F.; Vela, Jose Miguel; Almansa, Carmen 分享 收藏
Efficacy of SIGMAR1-based therapy in the early treatment of confirmed mild symptomatic COVID-19 patients Grau, Santiago; Vela, Jose Miguel; Gurt, Alba; Barcelo-Vidal, Jaime; Ojeda, Fabiola; Lopez, Iago; Gomez-Garcia, Laura; Loza, Maria Isabel; Martin-Garcia, Elena; Maldonado, Rafael; Monfort, Jordi 分享 收藏
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Discovery of WLB-89462, a New Drug-like and Highly Selective s2 Receptor Ligand with Neuroprotective Properties Christmann, Ute; Diaz, Jose Luis; Pascual, Rosalia; Bordas, Magda; Alvarez, Ines; Monroy, Xavier; Porras, Monica; Yeste, Sandra; Reinoso, Raquel F.; Merlos, Manuel; Vela, Jose Miguel; Almansa, Carmen 分享 收藏
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Bispecific sigma-1 receptor antagonism and mu-opioid receptor partial agonism: WLB-73502, an analgesic with improved efficacy and safety profile compared to strong opioids Vidal-Torres, Alba; Fernandez-Pastor, Begona; Garcia, Monica; Ayet, Eva; Cabot, Anna; Burgueno, Javier; Monroy, Xavier; Aubel, Bertrand; Codony, Xavier; Romero, Luz; Pascual, Rosalia; Serafini, Maria Teresa; Encina, Gregorio; Almansa, Carmen; Zamanillo, Daniel; Merlos, Manuel; Vela, Jose Miguel 分享 收藏
TRPA1 modulation by Sigma-1 receptor prevents oxaliplatin-induced painful peripheral neuropathy Marcotti, Aida; Fernandez-Trillo, Jorge; Gonzalez, Alejandro; Vizcaino-Escoto, Marta; Ros-Arlanzon, Pablo; Romero, Luz; Miguel Vela, Jose; Gomis, Ana; Viana, Felix; de la Pena, Elvira 分享 收藏
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Piperazinyl Bicyclic Derivatives as Selective Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels Fernandez, Ariadna; Luis Diaz, Jose; Garcia, Monica; Rodriguez-Escrich, Sergi; Lorente, Adriana; Enrech, Raquel; Dordal, Albert; Portillo-Salido, Enrique; Porras, Monica; Fernandez, Begona; Reinoso, Raquel F.; Vela, Jose Miguel; Almansa, Carmen 分享 收藏
Propionamide Derivatives as Dual μ-Opioid Receptor Agonists and σ1 Receptor Antagonists for the Treatment of Pain Garcia, Monica; Llorente, Virginia; Garriga, Lourdes; Christmann, Ute; Rodriguez-Escrich, Sergi; Virgili, Marina; Fernandez, Begona; Bordas, Magda; Ayet, Eva; Burgueno, Javier; Pujol, Marta; Dordal, Albert; Portillo-Salido, Enrique; Gris, Georgia; Miguel Vela, Jose; Almansa, Carmen 分享 收藏
Tricyclic Triazoles as σ1 Receptor Antagonists for Treating Pain Luis Diaz, Jose; Cuevas, Felix; Oliva, Ana, I; Font, Daniel; Angeles Sarmentero, M.; Alvarez-Bercedo, Paula; Lopez-Valbuena, Jose M.; Pericas, Miquel A.; Enrech, Raquel; Montero, Ana; Yeste, Sandra; Vidal-Torres, Alba; Alvarez, Ines; Perez, Pilar; Miguel Cendan, Cruz; Cobos, Enrique J.; Miguel Vela, Jose; Almansa, Carmen 分享 收藏
Bicyclic Diazepinones as Dual Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels and the Norepinephrine Transporter Luis Diaz, Jose; Cuevas, Felix; Pazos, Gonzalo; Alvarez-Bercedo, Paula; Oliva, Ana, I; Angeles Sarmentero, M.; Font, Daniel; Jimenez-Aquino, Agustin; Moron, Maria; Port, Adriana; Pascual, Rosalia; Dordal, Albert; Portillo-Salido, Enrique; Reinoso, Raquel F.; Miguel Vela, Jose; Almansa, Carmen 分享 收藏
EST64454: a Highly Soluble σ1 Receptor Antagonist Clinical Candidate for Pain Management Luis Diaz, Jose; Garcia, Monica; Torrens, Antoni; Maria Caamano, Ana; Enjo, Juan; Sicre, Cristina; Lorente, Adriana; Port, Adriana; Montero, Ana; Yeste, Sandra; Alvarez, Ines; Martin, Miquel; Maldonado, Rafael; de laPuente, Beatriz; Vidal-Torres, Alba; Miguel Cendan, Cruz; Miguel Vela, Jose; Almansa, Carmen 分享 收藏
Discovery of EST73502, a Dual μ-Opioid Receptor Agonist and σ1 Receptor Antagonist Clinical Candidate for the Treatment of Pain Garcia, Monica; Virgili, Marina; Alonso, Monica; Alegret, Carles; Farran, Joan; Fernandez, Begona; Bordas, Magda; Pascual, Rosalia; Burgueno, Javier; Vidal-Torres, Alba; Fernandez de Henestrosa, Antonio R.; Ayet, Eva; Merlos, Manuel; Miguel Vela, Jose; Plata-Salaman, Carlos R.; Almansa, Carmen 分享 收藏
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Sigma-1 receptors control neuropathic pain and macrophage infiltration into the dorsal root ganglion after peripheral nerve injury Bravo-Caparros, Inmaculada; Carmen Ruiz-Cantero, M.; Perazzoli, Gloria; Cronin, Shane J. F.; Vela, Jose M.; Hamed, Mohamed F.; Penninger, Josef M.; Baeyens, Jose M.; Cobos, Enrique J.; Nieto, Francisco R. 分享 收藏