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收藏Design, synthesis and evaluation of carbamate-bridged amino acid prodrugs of cycloicaritin with improved antitumor activity, aqueous solubility and phase II metabolic stability (vol 276, 116646], 2024)设计、合成及评价具有增强抗肿瘤活性、水溶性和相II代谢稳定性的氨基甲酸酯桥接的环异肌肽氨基酸前药 (vol 276, 116646], 2024)
Wang, Weiping; Fan, Jiaqi; Li, Fengxiao; Gan, Shuo; Zhang, Jiaming; Wang, Yanfang; Li, Yingchao; Li, Wenchao; He, Zhonggui; Ding, Huaiwei; Sun, Yongbing; Zhang, Tianhong; Jiang, Qikun
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收藏Development and optimization of a high-throughput LC-MS/MS method for the simultaneous determination of Exatecan and its Cathepsin B-sensitive prodrug, and ARV-825 in rat plasma: Application to pharmacokinetic study
Xu, Xiaolan; Liu, Yangyang; Yan, Qing; Bai, Chenxia; Ran, Xiaohua; Li, Jing; Zhang, Jiaming; Jiang, Qikun; Zhang, Tianhong
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收藏Inhibition of alanine-serine-cysteine transporter 2-mediated auto-enhanced photodynamic cancer therapy of co-nanoassembly between V-9302 and photosensitizer (vol 629, pg 773, 2023)
Jiang, Qikun; Lu, Sirun; Xu, Xiaolan; Bai, Chenxia; Yan, Qing; Fang, Mengna; Huang, Li; Jin, Chunming; Zhang, Yunran; Sun, Jin; He, Zhonggui; Zhao, Chunyang; Qin, Feng; Wang, Yongjun; Zhang, Tianhong
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收藏Exploring the associations between data-driven insomnia disorder combined with mild anxiety or/and depressive symptoms and the efficacy of Cognitive-Behavioral Therapy for insomnia探究数据驱动的失眠障碍合并轻度焦虑或/和抑郁症状与失眠认知行为疗法疗效之间的关联
Lyu, Dongbin; Qian, Ruiyi; Ge, Fangmei; Wang, Yang; Wang, Hongyan; Zhao, Yating; Han, Hui; Liu, Ruyun; Liu, Yutong; Chen, Yiling; Ji, Caojun; Luo, Xin; Zhang, Tianhong; Leng, Yue; Zhang, Jie; Yuan, Chengmei; Xiao, Zeping
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收藏Design, synthesis and evaluation of carbamate-bridged amino acid prodrugs of cycloicaritin with improved antitumor activity, aqueous solubility and phase II metabolic stability具有改善的抗肿瘤活性,水溶性和II相代谢稳定性的环淫羊藿素氨基甲酸酯桥联氨基酸前药的设计,合成和评价
Wang, Weiping; Fan, Jiaqi; Li, Fengxiao; Gan, Shuo; Zhang, Jiaming; Wang, Yanfang; Li, Yingchao; Li, Wenchao; He, Zhonggui; Ding, Huaiwei; Sun, Yongbing; Zhang, Tianhong; Jiang, Qikun
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收藏Inhibition of alanine-serine-cysteine transporter 2-mediated auto-enhanced photodynamic cancer therapy of co-nanoassembly between V-9302 and photosensitizer
Jiang, Qikun; Lu, Sirun; Xu, Xiaolan; Bai, Chenxia; Yan, Qing; Fang, Mengna; Huang, Li; Jin, Chunming; Zhang, Yunran; Sun, Jin; He, Zhonggui; Zhao, Chunyang; Qin, Feng; Wang, Yongjun; Zhang, Tianhong
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收藏Bioactivatable Pseudotripeptidization of Cyclic Dipeptides To Increase the Affinity toward Oligopeptide Transporter 1 for Enhanced Oral Absorption: An Application to Cyclo(L-Hyp-L-Ser) (JBP485)
Jiang, Qikun; Zhang, Jiangnan; Tong, Peiyue; Gao, Yan; Lv, Yiqin; Wang, Changyuan; Luo, Meiling; Sun, Mengchi; Wang, Jian; Peng, Yao; Cao, Linlin; Wang, Gang; Wang, Yang; Kan, Qiming; Zhang, Tianhong; Wang, Yongjun; Liu, Kexin; Sun, Jin; He, Zhonggui
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收藏Improving the oral bioavailability of tapentadol via a carbamate prodrug approach: synthesis, bioactivation, and pharmacokinetics通过氨基甲酸酯前药方法提高他喷他多的口服生物利用度: 合成,生物活化和药代动力学
Li, Yingchao; Wang, Yongjun; Zhang, Ran; Liu, Cuiru; Wei, Yue; Sun, Jin; He, Zhonggui; Xu, Youjun; Zhang, Tianhong
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收藏Metabolic Pathway of Icotinib In Vitro: The Differential Roles of CYP3A4, CYP3A5, and CYP1A2 on Potential Pharmacokinetic Drug-Drug Interaction
Zhang, TianHong; Zhang, KeRong; Ma, Li; Li, Zheng; Wang, Juan; Zhang, YunXia; Lu, Chuang; Zhu, Mingshe; Zhuang, XiaoMei
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收藏Accumulation of intact sulfur mustard in adipose tissue and toxicokinetics by chemical conversion and isotope-dilution liquid chromatography-tandem mass spectrometry
Xu, Bin; Zong, Cheng; Zhang, Yajiao; Zhang, Tianhong; Wang, Xiaoying; Qi, Meiling; Wu, Jianfeng; Guo, Lei; Wang, Peng; Chen, Jia; Liu, Qin; Xu, Hua; Xie, Jianwei; Zhang, Zhenqing
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收藏Effects of Silymarin, Glycyrrhizin, and Oxymatrine on the Pharmacokinetics of Ribavirin and Its Major Metabolite in Rats
Liao, Sha; Jin, Xueyuan; Li, Jinglai; Zhang, Tianhong; Zhang, Wenpeng; Shi, Weiguo; Fan, Shiyong; Wang, Xiaoying; Wang, Juan; Zhong, Bohua; Zhang, Zhenqing
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