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Emmanuel N. Pitsinos

National Centre of Scientific Research Demokritos

24H指数
83论文数
1.9K被引数
收录论文 25
发表时间
Uncialamycin-based antibody-drug conjugates: Unique enediyne ADCs exhibiting bystander killing effect
err2021-06-21
err29
errOAAI
errNicolaou, K. C.; Rigol, Stephan; Pitsinos, Emmanuel N.; Das, Dipendu; Lu, Yong; Rout, Subhrajit; Schammel, Alexander W.; Holte, Dane; Lin, Baiwei; Gu, Christine; Sarvaiya, Hetal; Trinidad, Jose; Barbour, Nicole; Valdiosera, Amanda M.; Sandoval, Joseph; Lee, Christina; Aujay, Monette; Fernando, Hanan; Dhar, Anukriti; Karsunky, Holger; Taylor, Nicole; Pysz, Marybeth; Gavrilyuk, Julia
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Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody-Drug Conjugates
err2020-07-14
err12
PREAI
errNicolaou, K. C.; Li, Ruofan; Chen, Qifeng; Lu, Zhaoyong; Pitsinos, Emmanuel N.; Schammel, Alexander; Lin, Baiwei; Gu, Christine; Sarvaiya, Hetal; Tchelepi, Robert; Valdiosera, Amanda; Clubb, Justin; Barbour, Nicole; Sisodiya, Vikram; Sandoval, Joseph; Lee, Christina; Aujay, Monette; Gavrilyuk, Julia
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Total Synthesis and Biological Evaluation of Tiancimycins A and B, Yangpumicin A, and Related Anthraquinone-Fused Enediyne Antitumor Antibiotics
err2020-01-24
err40
PREAI
errNicolaou, K. C.; Das, Dipendu; Lu, Yong; Rout, Subhrajit; Pitsinos, Emmanuel N.; Lyssikatos, Joseph; Schammel, Alexander; Sandoval, Joseph; Hammond, Mikhail; Aujay, Monette; Gavrilyuk, Julia
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DNA Binding and Cleavage Modes of Shishijimicin A
err2019-05-03
err21
PREAI
errZhang, Hao; Li, Ruofan; Ba, Sai; Lu, Zhaoyong; Pitsinos, Emmanuel N.; Li, Tianhu; Nicolaou, K. C.
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Streamlined Total Synthesis of Shishijimicin A and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues thereof and Practical Syntheses of PhthNSSMe and Related Sulfenylating Reagents
err2018-09-14
err28
PREAI
errNicolaou, K. C.; Li, Ruofan; Lu, Zhaoyong; Pitsinos, Emmanuel N.; Alemany, Lawrence B.; Aujay, Monette; Lee, Christina; Sandoval, Joseph; Gavrilyuk, Julia
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Total Synthesis and Full Structural Assignment of Namenamicin
err2018-06-22
err15
PREAI
errNicolaou, K. C.; Li, Ruofan; Lu, Zhaoyong; Pitsinos, Emmanuel N.; Alemany, Lawrence B.
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Streamlined Total Synthesis of Uncialamycin and Its Application to the Synthesis of Designed Analogues for Biological Investigations
err2016-06-27
err99
PREAI
errNicolaou, K. C.; Wang, Yanping; Lu, Min; Mandal, Debashis; Pattanayak, Manas R.; Yu, Ruocheng; Shah, Akshay A.; Chen, Jason S.; Zhang, Hongjun; Crawford, James J.; Pasunoori, Laxman; Poudel, Yam B.; Chowdari, Naidu S.; Pan, Chin; Nazeer, Ayesha; Gangwar, Sanjeev; Vite, Gregory; Pitsinos, Emmanuel N.
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A Fast Entry to Furanoditerpenoid-Based Hedgehog Signaling Inhibitors: Identifying Essential Structural Features
err2014-06-04
err20
PREAI
errChatzopoulou, Maria; Antoniou, Antonia; Pitsinos, Emmanuel N.; Bantzi, Marina; Koulocheri, Sofia D.; Haroutounian, Serkos A.; Giannis, Athanassios
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Enantioselective Total Synthesis of (-)-Laurenditerpenol
err2012-08-20
err21
PREAI
errPitsinos, Emmanuel N.; Athinaios, Nikolaos; Vidali, Veroniki P.
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Tumor necrosis factor-α promotes malignant pleural effusion
err2007-10-17
err102
errOAAI
errStathopoulos, Georgios T.; Kollintza, Androniki; Moschos, Charalampos; Psallidas, Loannis; Sherrill, Taylor P.; Pitsinos, Emmanuel N.; Vassiliou, Spyridoula; Karatza, Marilena; Papiris, Spyros A.; Graf, Daniel; Orphanidou, Dora; Light, Richard W.; Roussos, Charis; Blackwell, Timothy S.; Kalomenidis, Ioannis
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Influence of the scyphostatin side chain on the mode of inhibition of neutral sphingomyelinase
err2006-06-30
err18
PREAI
errWascholowski, Veit; Giannis, Athanassios; Pitsinos, Emmanuel N.
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Synthesis and biological evaluation of novel steroid-modified ether phospholipids
err2005-12-01
err1
PREAI
errKarantonis, HC; Pitsinos, EN; Antonopoulou, S; Couladouros, EA; Demopoulos, CA
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A novel 2′-(N-methylpyridinium acetate) prodrug of paclitaxel induces superior antitumor responses in preclinical cancer models
err2002-08-20
err39
PREAI
errWrasidlo, W; Gaedicke, G; Guy, RK; Renaud, J; Pitsinos, E; Nicolaou, KC; Reisfeld, RA; Lode, HN
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TOTAL SYNTHESIS OF CALICHEAMICIN-GAMMA-1(I) .2. DEVELOPMENT OF AN ENANTIOSELECTIVE ROUTE TO (-)-CALICHEAMICINONE
err2002-05-01
err116
PREAI
errSMITH, AL; PITSINOS, EN; HWANG, CK; MIZUNO, Y; SAIMOTO, H; SCARLATO, GR; SUZUKI, T; NICOLAOU, KC
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ENANTIOSELECTIVE TOTAL SYNTHESIS OF (-)-CALICHEAMICINONE
err2002-05-01
err78
PREAI
errSMITH, AL; HWANG, CK; PITSINOS, E; SCARLATO, GR; NICOLAOU, KC
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