未登录
分享
收藏Further Insights Into the Metabolism of LGD-4033 in Human Urine. Part 2. A New Minor Metabolite With Antagonistic Activity on the Androgen Receptor Can Indicate Recent Substance Intake关于LGD-4033在人尿液中的代谢进一步研究。第二部分:一种具有雄激素受体拮抗活性的新微量代谢物可指示近期物质摄入。
Angelis, Yiannis S.; Sakellariou, Panagiotis; Keiler, Annekathrin M.; Thevis, Mario; Thomas, Andreas; Lam, Kevin; Wolber, Gerhard; Vonaparti, Ariadni; Voss, Sven; Petrou, Michael; Pitsinos, Emmanuel N.
分享
收藏Uncialamycin-based antibody-drug conjugates: Unique enediyne ADCs exhibiting bystander killing effect
Nicolaou, K. C.; Rigol, Stephan; Pitsinos, Emmanuel N.; Das, Dipendu; Lu, Yong; Rout, Subhrajit; Schammel, Alexander W.; Holte, Dane; Lin, Baiwei; Gu, Christine; Sarvaiya, Hetal; Trinidad, Jose; Barbour, Nicole; Valdiosera, Amanda M.; Sandoval, Joseph; Lee, Christina; Aujay, Monette; Fernando, Hanan; Dhar, Anukriti; Karsunky, Holger; Taylor, Nicole; Pysz, Marybeth; Gavrilyuk, Julia
分享
收藏Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody-Drug Conjugates
Nicolaou, K. C.; Li, Ruofan; Chen, Qifeng; Lu, Zhaoyong; Pitsinos, Emmanuel N.; Schammel, Alexander; Lin, Baiwei; Gu, Christine; Sarvaiya, Hetal; Tchelepi, Robert; Valdiosera, Amanda; Clubb, Justin; Barbour, Nicole; Sisodiya, Vikram; Sandoval, Joseph; Lee, Christina; Aujay, Monette; Gavrilyuk, Julia
分享
收藏Total Synthesis and Biological Evaluation of Tiancimycins A and B, Yangpumicin A, and Related Anthraquinone-Fused Enediyne Antitumor Antibiotics
Nicolaou, K. C.; Das, Dipendu; Lu, Yong; Rout, Subhrajit; Pitsinos, Emmanuel N.; Lyssikatos, Joseph; Schammel, Alexander; Sandoval, Joseph; Hammond, Mikhail; Aujay, Monette; Gavrilyuk, Julia
分享
收藏
分享
收藏Streamlined Total Synthesis of Shishijimicin A and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues thereof and Practical Syntheses of PhthNSSMe and Related Sulfenylating Reagents
Nicolaou, K. C.; Li, Ruofan; Lu, Zhaoyong; Pitsinos, Emmanuel N.; Alemany, Lawrence B.; Aujay, Monette; Lee, Christina; Sandoval, Joseph; Gavrilyuk, Julia
分享
收藏
分享
收藏Streamlined Total Synthesis of Uncialamycin and Its Application to the Synthesis of Designed Analogues for Biological Investigations
Nicolaou, K. C.; Wang, Yanping; Lu, Min; Mandal, Debashis; Pattanayak, Manas R.; Yu, Ruocheng; Shah, Akshay A.; Chen, Jason S.; Zhang, Hongjun; Crawford, James J.; Pasunoori, Laxman; Poudel, Yam B.; Chowdari, Naidu S.; Pan, Chin; Nazeer, Ayesha; Gangwar, Sanjeev; Vite, Gregory; Pitsinos, Emmanuel N.
分享
收藏
分享
收藏
分享
收藏
分享
收藏Tumor necrosis factor-α promotes malignant pleural effusion
Stathopoulos, Georgios T.; Kollintza, Androniki; Moschos, Charalampos; Psallidas, Loannis; Sherrill, Taylor P.; Pitsinos, Emmanuel N.; Vassiliou, Spyridoula; Karatza, Marilena; Papiris, Spyros A.; Graf, Daniel; Orphanidou, Dora; Light, Richard W.; Roussos, Charis; Blackwell, Timothy S.; Kalomenidis, Ioannis
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏
分享
收藏