未登录 分享 收藏
分享 收藏
分享 收藏
Photoswitchable COX-2-Selective Inhibitors as Light-Regulated Anti-Inflammatory Agents 光开关COX-2选择性抑制剂作为光调控抗炎剂 Morales, Amanda; Cruz, Alejandro; Perez-Sanchez, Alex; D'Avino, Danilo; Galassi, Gaia; Milano, Erica Ginevra; Bernareggi, Irene; Arenos-Bach, Carla; Grazioso, Giovanni; Alibes, Ramon; Hernando, Jordi; Gorostiza, Pau; Rossi, Antonietta; Pistocchi, Anna; Matera, Carlo; Busque, Felix; Gonzalez-Lafont, Angels; Lluch, Jose M. 分享 收藏
分享 收藏
分享 收藏
分享 收藏
Novel non-peptide uracil-derived human gonadotropin-releasing hormone receptor antagonists 新型非肽类尿嘧啶衍生的促性腺激素释放激素受体拮抗剂 Ciceri, Samuele; Fassi, Enrico M. A.; Vezzoli, Valeria; Bonomi, Marco; Colombo, Diego; Ferraboschi, Patrizia; Grazioso, Giovanni; Grisenti, Paride; Villa, Stefania; Castellano, Carlo; Meneghetti, Fiorella 分享 收藏
分享 收藏
Unlocking the Antibiofilm Potential of Natural Compounds by Targeting the NADH:quinone Oxidoreductase WrbA 通过靶向NADH释放天然化合物的抗生物膜潜力: 醌氧化还原酶WrbA Ratti, Alessandro; Fassi, Enrico M. A.; Forlani, Fabio; Zangrossi, Maurizio; Mori, Matteo; Cappitelli, Francesca; Roda, Gabriella; Villa, Stefania; Villa, Federica; Grazioso, Giovanni 分享 收藏
Mechanistic Insights into the Antibiofilm Mode of Action of Ellagic Acid 对鞣花酸的抗生物膜作用模式的机理见解 Ratti, Alessandro; Fassi, Enrico M. A.; Forlani, Fabio; Mori, Matteo; Villa, Federica; Cappitelli, Francesca; Sgrignani, Jacopo; Roda, Gabriella; Cavalli, Andrea; Villa, Stefania; Grazioso, Giovanni 分享 收藏
Computational Design, Synthesis, and Biological Evaluation of Diimidazole Analogues Endowed with Dual PCSK9/HMG-CoAR-Inhibiting Activity 具有双重PCSK9/hmg-coar抑制活性的二咪唑类似物的计算设计,合成和生物学评估 Lammi, Carmen; Fassi, Enrico M. A.; Manenti, Marco; Brambilla, Marta; Conti, Maria; Li, Jianqiang; Roda, Gabriella; Camera, Marina; Silvani, Alessandra; Grazioso, Giovanni 分享 收藏
Elagolix Sodium Salt and Its Synthetic Intermediates: A Spectroscopic, Crystallographic, and Conformational Study Elagolix钠盐及其合成中间体: 光谱,晶体学和构象研究 Ciceri, Samuele; Colombo, Diego; Fassi, Enrico M. A.; Ferraboschi, Patrizia; Grazioso, Giovanni; Grisenti, Paride; Iannone, Marco; Castellano, Carlo; Meneghetti, Fiorella 分享 收藏
分享 收藏
Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors 作为SARS-CoV-2 Mpro抑制剂的 β-酰胺基硼酸的计算设计,合成和生物物理评估 Fassi, Enrico M. A.; Manenti, Marco; Citarella, Andrea; Dei Cas, Michele; Casati, Sara; Micale, Nicola; Schirmeister, Tanja; Roda, Gabriella; Silvani, Alessandra; Grazioso, Giovanni 分享 收藏
分享 收藏
Systematic Development of Peptide Inhibitors Targeting the CXCL12/HMGB1 Interaction 靶向CXCL12/HMGB1相互作用的肽抑制剂的系统开发 Sgrignani, Jacopo; Cecchinato, Valentina; Fassi, Enrico M. A.; D'Agostino, Gianluca; Garofalo, Maura; Danelon, Gabriela; Pedotti, Mattia; Simonelli, Luca; Varani, Luca; Grazioso, Giovanni; Uguccioni, Mariagrazia; Cavalli, Andrea 分享 收藏
Investigation of Chlorella pyrenoidosa Protein as a Source of Novel Angiotensin I-Converting Enzyme (ACE) and Dipeptidyl Peptidase-IV (DPP-IV) Inhibitory Peptides 蛋白核小球藻蛋白作为新型血管紧张素I转换酶 (ACE) 和二肽基肽酶-IV (dpp-iv) 抑制肽来源的研究 Li, Yuchen; Aiello, Gilda; Fassi, Enrico Mario Alessandro; Boschin, Giovanna; Bartolomei, Martina; Bollati, Carlotta; Roda, Gabriella; Arnoldi, Anna; Grazioso, Giovanni; Lammi, Carmen 分享 收藏
分享 收藏
Trans-Epithelial Transport, Metabolism, and Biological Activity Assessment of the Multi-Target Lupin Peptide LILPKHSDAD (P5) and Its Metabolite LPKHSDAD (P5-Met) 多靶点羽扇豆肽LILPKHSDAD (P5) 及其代谢物LPKHSDAD (P5-Met) 的跨上皮转运、代谢和生物活性评估 Lammi, Carmen; Aiello, Gilda; Bollati, Carlotta; Li, Jianqiang; Bartolomei, Martina; Ranaldi, Giulia; Ferruzza, Simonetta; Fassi, Enrico Mario Alessandro; Grazioso, Giovanni; Sambuy, Yula; Arnoldi, Anna 分享 收藏