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Giovanni Grazioso

dipartimento di scienze farmaceutiche

24H指数
104论文数
1.5K被引数
收录论文 55
发表时间
Protein language model-generated enzyme sequences exhibit high stability in molecular dynamics simulations蛋白质语言模型生成的酶序列在分子动力学模拟中表现出高稳定性
err2026-08-31
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errEM Enrico Mario Alessandro Fassi; MN Marco Nicolini; ES Emanuele Saitto; GV Giorgio Valentini; EC Elena Casiraghi; GG Giovanni Grazioso
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A nicotinic-dopaminergic hybrid probe enhances D2-like autoreceptor-mediated inhibition of dopamine release烟碱-多巴胺能杂交探针增强D2样自身受体介导的多巴胺释放抑制
err2026-08-28
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errCarlo Matera; Massimo Grilli; Luca Pucci; Enrico Mario Alessandro Fassi; Sergio Fucile; Mario Marchi; Chiara Fiorentini; Francesco Clementi; Michele Zoli; Clelia Dallanoce; Giovanni Grazioso; Marco De Amici; Cecilia Gotti
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PCSK9 inhibitors: an updated patent review 2024–2025PCSK9抑制剂:2024–2025年专利综述更新
err2026-05-21
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PREAI
errEnrico Mario Alessandro Fassi; Marco Albani; Lorenza D’Adduzio; Erica Ginevra Milano; Carmen Lammi; Giovanni Grazioso
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Photoswitchable COX-2-Selective Inhibitors as Light-Regulated Anti-Inflammatory Agents光开关COX-2选择性抑制剂作为光调控抗炎剂
err2026-04-01
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errMorales, Amanda; Cruz, Alejandro; Perez-Sanchez, Alex; D'Avino, Danilo; Galassi, Gaia; Milano, Erica Ginevra; Bernareggi, Irene; Arenos-Bach, Carla; Grazioso, Giovanni; Alibes, Ramon; Hernando, Jordi; Gorostiza, Pau; Rossi, Antonietta; Pistocchi, Anna; Matera, Carlo; Busque, Felix; Gonzalez-Lafont, Angels; Lluch, Jose M.
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Insights into the catalytic mechanism of formate dehydrogenases from different microbial sources不同微生物来源甲酸脱氢酶催化机制的研究进展
err2026-03-05
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errLaura Legnani; Marco Gargiulo; Elia Lio; Enrico Mario Alessandro Fassi; Giovanni Grazioso; Maria Assunta Chiacchio; Barış Binay; Stefania Brocca; Francesco Secundo
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Computational characterization of peptide binding stability to HLA-C allotypes and its association with HIV-1 infection progression and HIV-1 related neurocognitive impairment肽与HLA-C所有型结合稳定性的计算表征及其与HIV-1感染进展和HIV-1相关神经认知障碍的关联
err2025-12-11
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errMauro Voi; Antonella Sangalli; Erica Ginevra Milano; Carola De Martinis; Elisa Orlandi; Stefano Tamburin; Elisa Mantovani; Angela Federico; Massimiliano Lanzafame; Emanuela Lattuada; Gustavo Adolfo Argañaraz; Bosco Christiano Maciel Da Silva; Alberto Jose Da Silva Duarte; Jorge Casseb; Enrique Roberto Argañaraz; Marina Malena; Marco Albani; Alessandra Ruggiero; Maria Grazia Romanelli; Maria Teresa Valenti; Giovanni Grazioso; Donato Zipeto
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Insights on Zosteric Acid Analogues Activity Against Candida albicans Biofilm Formation关于Zosteric Acid Analogues对Candida albicans生物膜形成的活性见解
err2025-05-20
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PREAI
errCatto, Cristina; Fassi, Enrico M. A.; Grazioso, Giovanni; Gelain, Arianna; Villa, Stefania; Cappitelli, Francesca
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Novel non-peptide uracil-derived human gonadotropin-releasing hormone receptor antagonists新型非肽类尿嘧啶衍生的促性腺激素释放激素受体拮抗剂
err2024-12-01
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PREAI
errCiceri, Samuele; Fassi, Enrico M. A.; Vezzoli, Valeria; Bonomi, Marco; Colombo, Diego; Ferraboschi, Patrizia; Grazioso, Giovanni; Grisenti, Paride; Villa, Stefania; Castellano, Carlo; Meneghetti, Fiorella
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PCSK9 inhibitors: a patent review 2018-2023PCSK9抑制剂: 专利审查2018-2023
err2024-04-11
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PREAI
errFassi, Enrico Mario Alessandro; Citarella, Andrea; Albani, Marco; Milano, Erica Ginevra; Legnani, Laura; Lammi, Carmen; Silvani, Alessandra; Grazioso, Giovanni
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Unlocking the Antibiofilm Potential of Natural Compounds by Targeting the NADH:quinone Oxidoreductase WrbA通过靶向NADH释放天然化合物的抗生物膜潜力: 醌氧化还原酶WrbA
err2023-08-14
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errRatti, Alessandro; Fassi, Enrico M. A.; Forlani, Fabio; Zangrossi, Maurizio; Mori, Matteo; Cappitelli, Francesca; Roda, Gabriella; Villa, Stefania; Villa, Federica; Grazioso, Giovanni
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Mechanistic Insights into the Antibiofilm Mode of Action of Ellagic Acid对鞣花酸的抗生物膜作用模式的机理见解
err2023-06-17
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errRatti, Alessandro; Fassi, Enrico M. A.; Forlani, Fabio; Mori, Matteo; Villa, Federica; Cappitelli, Francesca; Sgrignani, Jacopo; Roda, Gabriella; Cavalli, Andrea; Villa, Stefania; Grazioso, Giovanni
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Computational Design, Synthesis, and Biological Evaluation of Diimidazole Analogues Endowed with Dual PCSK9/HMG-CoAR-Inhibiting Activity具有双重PCSK9/hmg-coar抑制活性的二咪唑类似物的计算设计,合成和生物学评估
err2023-06-01
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errLammi, Carmen; Fassi, Enrico M. A.; Manenti, Marco; Brambilla, Marta; Conti, Maria; Li, Jianqiang; Roda, Gabriella; Camera, Marina; Silvani, Alessandra; Grazioso, Giovanni
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Elagolix Sodium Salt and Its Synthetic Intermediates: A Spectroscopic, Crystallographic, and Conformational StudyElagolix钠盐及其合成中间体: 光谱,晶体学和构象研究
err2023-05-03
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errCiceri, Samuele; Colombo, Diego; Fassi, Enrico M. A.; Ferraboschi, Patrizia; Grazioso, Giovanni; Grisenti, Paride; Iannone, Marco; Castellano, Carlo; Meneghetti, Fiorella
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Development of AMBER Parameters for Molecular Simulations of Selected Boron-Based Covalent Ligands开发用于选定硼基共价配体的分子模拟的琥珀色参数
err2023-03-22
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errChiacchio, Maria Assunta; Legnani, Laura; Fassi, Enrico Mario Alessandro; Roda, Gabriella; Grazioso, Giovanni
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Computational Design, Synthesis, and Biophysical Evaluation of β-Amido Boronic Acids as SARS-CoV-2 Mpro Inhibitors作为SARS-CoV-2 Mpro抑制剂的 β-酰胺基硼酸的计算设计,合成和生物物理评估
err2023-03-03
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errFassi, Enrico M. A.; Manenti, Marco; Citarella, Andrea; Dei Cas, Michele; Casati, Sara; Micale, Nicola; Schirmeister, Tanja; Roda, Gabriella; Silvani, Alessandra; Grazioso, Giovanni
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Computational Design and Biological Evaluation of Analogs of Lupin Peptide P5 Endowed with Dual PCSK9/HMG-CoAR Inhibiting Activity具有双重PCSK9/hmg-coar抑制活性的羽扇豆肽P5类似物的计算设计和生物学评价
err2022-03-18
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errLammi, Carmen; Fassi, Enrico M. A.; Li, Jianqiang; Bartolomei, Martina; Benigno, Giulia; Roda, Gabriella; Arnoldi, Anna; Grazioso, Giovanni
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Systematic Development of Peptide Inhibitors Targeting the CXCL12/HMGB1 Interaction靶向CXCL12/HMGB1相互作用的肽抑制剂的系统开发
err2021-09-13
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errSgrignani, Jacopo; Cecchinato, Valentina; Fassi, Enrico M. A.; D'Agostino, Gianluca; Garofalo, Maura; Danelon, Gabriela; Pedotti, Mattia; Simonelli, Luca; Varani, Luca; Grazioso, Giovanni; Uguccioni, Mariagrazia; Cavalli, Andrea
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Investigation of Chlorella pyrenoidosa Protein as a Source of Novel Angiotensin I-Converting Enzyme (ACE) and Dipeptidyl Peptidase-IV (DPP-IV) Inhibitory Peptides蛋白核小球藻蛋白作为新型血管紧张素I转换酶 (ACE) 和二肽基肽酶-IV (dpp-iv) 抑制肽来源的研究
err2021-05-12
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errLi, Yuchen; Aiello, Gilda; Fassi, Enrico Mario Alessandro; Boschin, Giovanna; Bartolomei, Martina; Bollati, Carlotta; Roda, Gabriella; Arnoldi, Anna; Grazioso, Giovanni; Lammi, Carmen
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Alkene Epoxidations Mediated by Mn-Salen Macrocyclic CatalystsMn-salen大环催化剂介导的烯烃环氧化反应
err2021-04-02
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errPappalardo, Andrea; Ballistreri, Francesco P.; Toscano, Rosa Maria; Chiacchio, Maria Assunta; Legnani, Laura; Grazioso, Giovanni; Veltri, Lucia; Sfrazzetto, Giuseppe Trusso
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Trans-Epithelial Transport, Metabolism, and Biological Activity Assessment of the Multi-Target Lupin Peptide LILPKHSDAD (P5) and Its Metabolite LPKHSDAD (P5-Met)多靶点羽扇豆肽LILPKHSDAD (P5) 及其代谢物LPKHSDAD (P5-Met) 的跨上皮转运、代谢和生物活性评估
err2021-03-05
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errLammi, Carmen; Aiello, Gilda; Bollati, Carlotta; Li, Jianqiang; Bartolomei, Martina; Ranaldi, Giulia; Ferruzza, Simonetta; Fassi, Enrico Mario Alessandro; Grazioso, Giovanni; Sambuy, Yula; Arnoldi, Anna
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