未登录Clinical, Imaging, and Pathological Features of Apocrine Intraductal Carcinoma of Salivary Glands: A Case Report and Literature Review涎腺导管腺癌的临床、影像及病理特征:病例报告及文献综述
Akita, Saki; Kuroki, Masashi; Kato, Hiroki; Suzui, Natsuko; Kawaura, Ryo; Yamada, Tatsuhiko; Shibata, Hirofumi; Okuda, Hiroshi; Iinuma, Ryota; Mori, Kenichi; Ogawa, Takenori
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收藏Discovery of ASP2453, a potent and orally bioavailable covalent inhibitor of KRAS G12C for the treatment of solid tumorsASP2453的发现,一种有效的口服生物可利用的KRAS G12C共价抑制剂,用于治疗实体瘤
Imaizumi, Tomoyoshi; Imanishi, Masashi; Yamaki, Susumu; Shimada, Itsuro; Satake, Yoshiki; Nigawara, Takahiro; Koike, Takanori; Yamanaka, Yosuke; Amano, Yasushi; Mori, Kenichi; Nakayama, Ayako; Nishizono, Yoshihiro; Shimazaki, Masashi; Nagashima, Takeyuki; Kuramoto, Kazuyuki
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收藏Discovery of ASP6918, a KRAS G12C inhibitor: Synthesis and structure-activity relationships of 1-{2,7-diazaspiro[3.5]non-2-yl} prop-2-en-1-one derivatives as covalent inhibitors with good potency and oral activity for the treatment of solid tumors
Imaizumi, Tomoyoshi; Shimada, Itsuro; Satake, Yoshiki; Yamaki, Susumu; Koike, Takanori; Nigawara, Takahiro; Kaneko, Osamu; Amano, Yasushi; Mori, Kenichi; Yamanaka, Yosuke; Nakayama, Ayako; Nishizono, Yoshihiro; Shimazaki, Masashi; Nagashima, Takeyuki; Kuramoto, Kazuyuki
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收藏Discovery and biological evaluation of 1-{2,7-diazaspiro[3.5]nonan-2-yl} prop-2-en-1-one derivatives as covalent inhibitors of KRAS G12C with favorable metabolic stability and anti-tumor activity
Imaizumi, Tomoyoshi; Akaiwa, Michinori; Abe, Tomoaki; Nigawara, Takahiro; Koike, Takanori; Satake, Yoshiki; Watanabe, Kazushi; Kaneko, Osamu; Amano, Yasushi; Mori, Kenichi; Yamanaka, Yosuke; Nagashima, Takeyuki; Shimazaki, Masashi; Kuramoto, Kazuyuki
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收藏The role of prostaglandin and E series prostaglandin receptor type 4 receptors in the development of bladder overactivity in a rat model of chemically induced prostatic inflammation
Mizoguchi, Shinsuke; Wolf-Johnson, Amanda S.; Ni, Jianshu; Mori, Kenichi; Suzuki, Takahisa; Takaoka, Eiichiro; Mimata, Hiromitsu; DeFranco, Donald B.; Wang, Zhou; Birder, Lori A.; Yoshimura, Naoki
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收藏Gilteritinib, a FLT3/AXL inhibitor, shows antileukemic activity in mouse models of FLT3 mutated acute myeloid leukemia
Mori, Masamichi; Kaneko, Naoki; Ueno, Yoko; Yamada, Masaki; Tanaka, Ruriko; Saito, Rika; Shimada, Itsuro; Mori, Kenichi; Kuromitsu, Sadao
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收藏The Selective Anaplastic Lymphoma Receptor Tyrosine Kinase Inhibitor ASP3026 Induces Tumor Regression and Prolongs Survival in Non-Small Cell Lung Cancer Model Mice
Mori, Masamichi; Ueno, Yoko; Konagai, Satoshi; Fushiki, Hiroshi; Shimada, Itsuro; Kondoh, Yutaka; Saito, Rika; Mori, Kenichi; Shindou, Nobuaki; Soga, Takatoshi; Sakagami, Hideki; Furutani, Takashi; Doihara, Hitoshi; Kudoh, Masafumi; Kuromitsu, Sadao
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收藏Discovery of N-[2-Hydroxy-6-(4-methoxybenzamido)phenyl]-4-(4-methyl-1,4-diazepan-1-yl)benzamide (Darexaban, YM150) as a Potent and Orally Available Factor Xa Inhibitor
Hirayama, Fukushi; Koshio, Hiroyuki; Ishihara, Tsukasa; Hachiya, Shunichiro; Sugasawa, Keizo; Koga, Yuji; Seki, Norio; Shiraki, Ryouta; Shigenaga, Takeshi; Iwatsuki, Yoshiyuki; Moritani, Yumiko; Mori, Kenichi; Kadokura, Takeshi; Kawasaki, Tomihisa; Matsumoto, Yuzo; Sakamoto, Shuichi; Tsukamoto, Shin-ichi
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