未登录In vivo efficacy of anti-B7-H3 antibody-drug conjugate (ADC) ifinatamab deruxtecan (I-DXd; DS-7300): An update from the Pediatric Preclinical In Vivo Testing (PIVOT) Program
Gorlick, Richard; Gill, Jonathan; Zhang, Wendong; Mosse, Yael; Maris, John; Groff, David; Smith, Malcolm; Teicher, Beverly; Neuhauser, Steve; Stearns, Tim; Philip, Vivek; Jocoy, Emily; Chuang, Jeff; Bult, Carol J.; Hasegawa, Jun; Qian, Xiaozhong; Houghton, Peter; Kurmasheva, Raushan
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收藏Ifinatamab deruxtecan (I-DXd), a novel B7-H3-targeting antibody-drug conjugate, demonstrates efficient payload delivery into tumor through target-dependent internalization
Katsumata, Len; Deguchi, Tsuneo; Hasegawa, Jun; Yamato, Michiko; Nishiya, Yumi; Watanabe, Akiko; Honda, Tomoyo; Minami, Megumi; Kasanuki, Naomi; Maejima, Takanori; Muramatsu, Sumie; Herrmann, Monika; Schulte, Nina; Polier, Gernot; Wang, Xuya; Yoshida, Takanori; Izumi, Nanae; Qian, Xiaozhong; Agatsuma, Toshinori; Nakamaru, Kenji
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收藏Identification and Therapeutic Targeting of GPR20, Selectively Expressed in Gastrointestinal Stromal Tumors, with DS-6157a, a First-in-Class Antibody-Drug Conjugate
Iida, Kenji; Ahmed, Amr H. Abdelhamid; Nagatsuma, Akiko Kawano; Shibutani, Tomoko; Yasuda, Satoru; Kitamura, Michiko; Hattori, Chiharu; Abe, Manabu; Hasegawa, Jun; Iguchi, Takuma; Karibe, Tsuyoshi; Nakada, Takashi; Inaki, Koichiro; Kamei, Reiko; Abe, Yuki; Nomura, Taisei; Andersen, Jessica L.; Santagata, Sandro; Hemming, Matthew L.; George, Suzanne; Doi, Toshihiko; Ochiai, Atsushi; Demetri, George D.; Agatsuma, Toshinori
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收藏Therapeutic targeting of GPR20, selectively expressed in gastrointestinal stromal tumor (GIST), with DS-6157a, an antibody-drug conjugate (ADC)
Iida, Kenji; Abdelhamid, Amr H.; Nagatsuma, Akiko Kawano; Shibutani, Tomoko; Yasuda, Satoru; Kitamura, Michiko; Hattori, Chiharu; Abe, Manabu; Hasegawa, Jun; Iguchi, Takuma; Karibe, Tsuyoshi; Nakada, Takashi; Inaki, Koichiro; Kamei, Reiko; Abe, Yuki; Andersen, Jessica L.; Santagata, Sandro; Hemming, Matthew L.; George, Suzanne; Doi, Toshihiko; Ochiai, Atsushi; Demetri, George D.; Agatsuma, Toshinori
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收藏Pharmacokinetic and Pharmacodynamic Profiles of Glyco-Modified Atrial Natriuretic Peptide Derivatives Synthesized Using Chemo-enzymatic Synthesis Approaches
Iwamoto, Mitsuhiro; Yamaguchi, Takahiro; Sekiguchi, Yukiko; Oishi, Shohei; Shiiki, Takeshi; Soma, Masako; Nakamura, Kensuke; Yoshida, Makoto; Chaya, Hiroyuki; Mori, Yutaka; Miyauchi, Ryuki; Hasegawa, Jun; Nagayama, Takahiro; Honda, Takeshi
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收藏Novel anti-EPHA2 antibody, DS-8895a for cancer treatment
Hasegawa, Jun; Sue, Mayumi; Yamato, Michiko; Ichikawa, Junya; Ishida, Saori; Shibutani, Tomoko; Kitamura, Michiko; Wada, Teiji; Agatsuma, Toshinori
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收藏Molecular Imaging and Quantitation of EphA2 Expression in Xenograft Models with 89Zr-DS-8895a
Burvenich, Ingrid J. G.; Parakh, Sagun; Gan, Hui K.; Lee, Fook-Thean; Guo, Nancy; Rigopoulos, Angela; Lee, Sze-Ting; Gong, Sylvia; O'Keefe, Graeme J.; Tochon-Danguy, Henri; Kotsuma, Masakatsu; Hasegawa, Jun; Senaldi, Giorgio; Scott, Andrew M.
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收藏Phosphorylation of p62 Activates the Keap1-Nrf2 Pathway during Selective Autophagyp62磷酸化激活选择性自噬过程中的Keap1-Nrf2途径
Ichimura, Yoshinobu; Waguri, Satoshi; Sou, Yu-shin; Kageyama, Shun; Hasegawa, Jun; Ishimura, Ryosuke; Saito, Tetsuya; Yang, Yinjie; Kouno, Tsuguka; Fukutomi, Toshiaki; Hoshii, Takayuki; Hirao, Atsushi; Takagi, Kenji; Mizushima, Tsunehiro; Motohashi, Hozumi; Lee, Myung-Shik; Yoshimori, Tamotsu; Tanaka, Keiji; Yamamoto, Masayuki; Komatsu, Masaaki
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收藏Crystal Structure of the Ubiquitin-associated (UBA) Domain of p62 and Its Interaction with Ubiquitin
Isogai, Shin; Morimoto, Daichi; Arita, Kyohei; Unzai, Satoru; Tenno, Takeshi; Hasegawa, Jun; Sou, Yu-shin; Komatsu, Masaaki; Tanaka, Keiji; Shirakawa, Masahiro; Tochio, Hidehito
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