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PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models (vol 67, pg 1262, 2024) PROTACs靶向BRM(SMARCA2)可在体内实现对BRG1(SMARCA4)的选择性降解,并在BRG1突变异种移植肿瘤模型中表现出活性(vol 67, pg 1262, 2024) Berlin, Michael; Cantley, Jennifer; Bookbinder, Mark; Bortolon, Elizabeth; Broccatelli, Fabio; Cadelina, Greg; Chan, Emily W.; Chen, Huifen; Chen, Xin; Cheng, Yunxing; Cheung, Tommy K.; Crew, Andrew P.; Davenport, Kim; Dinicola, Dean; Dong, Hanqing; Gordon, Debbie; Hamman, Brian D.; Harbin, Alicia; Haskell, Roy; He, Mingtao; Hole, Alison J.; Januario, Thomas; Kerry, Philip S.; Koenig, Stefan G.; Li, Limei; Merchant, Mark; Perez-Dorado, Inmaculada; Pizzano, Jennifer; Quinn, Connor; Rose, Christopher M.; Rousseau, Emma; Snyder, Lawrence B.; Soto, Leofal; Staben, Leanna R.; Sun, Hongming; Tian, Qingping; Wang, Gan; Wang, Jing; Wang, Weifeng; Ye, Crystal S.; Ye, Xiaofen; Zhang, Penghong; Zhou, Yuhui; Yauch, Robert; Dragovich, Peter S. 分享 收藏
Development of a Broadly Applicable Enzymatic Ligation Process for the Production of Single Guide RNAs 开发一种广泛适用的酶促连接过程用于单链引导RNA的生产 Bigatti, Martina; Moser, Andre; Dierssen, Bas; Frrokaj, Shtjefen; Covato, Elena; Pfleger, Christophe; Lill, Joerg; Leiser, Yael; Zuber, Joel; Staempfli, Andreas; Sladojevich, Filippo; Koenig, Stefan G. 分享 收藏
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Process Mass Intensity (PMI): A Holistic Analysis of Current Peptide Manufacturing Processes Informs Sustainability in Peptide Synthesis 过程质量强度 (PMI): 对当前肽制造过程的整体分析为肽合成的可持续性提供了信息 Kekessie, Ivy; Wegner, Katarzyna; Martinez, Isamir; Kopach, Michael E.; White, Timothy D.; Tom, Janine K.; Kenworthy, Martin N.; Gallou, Fabrice; Lopez, John; Koenig, Stefan G.; Payne, Philippa R.; Eissler, Stefan; Arumugam, Balasubramanian; Li, Changfeng; Mukherjee, Subha; Isidro-Llobet, Albert; Ludemann-Hombourger, Olivier; Richardson, Paul; Kittelmann, Jorg; Pedersen, Daniel Sejer; van den Bos, Leendert J. 分享 收藏
PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models Berlin, Michael; Cantley, Jennifer; Bookbinder, Mark; Bortolon, Elizabeth; Broccatelli, Fabio; Cadelina, Greg; Chan, Emily W.; Chen, Huifen; Chen, Xin; Cheng, Yunxing; Cheung, Tommy K.; Davenport, Kim; DiNicola, Dean; Gordon, Debbie; Hamman, Brian D.; Harbin, Alicia; Haskell, Roy; He, Mingtao; Hole, Alison J.; Januario, Thomas; Kerry, Philip S.; Koenig, Stefan G.; Li, Limei; Merchant, Mark; Perez-Dorado, Inmaculada; Pizzano, Jennifer; Quinn, Connor; Rose, Christopher M.; Rousseau, Emma; Soto, Leofal; Staben, Leanna R.; Sun, Hongming; Tian, Qingping; Wang, Jing; Wang, Weifeng; Ye, Crystal S.; Ye, Xiaofen; Zhang, Penghong; Zhou, Yuhui; Yauch, Robert; Dragovich, Peter S. 分享 收藏
Characterization of antisense oligonucleotide and guide ribonucleic acid diastereomers by hydrophilic interaction liquid chromatography coupled to mass spectrometry Goyon, Alexandre; Blevins, Molly S.; Napolitano, Jose G.; Nguyen, Daniel; Goel, Meenakshi; Scott, Brandon; Wang, Jenny; Koenig, Stefan G.; Chen, Tao; Zhang, Kelly 分享 收藏
Practical Synthesis of Reactive Immuno-PET Linker-Chelator (1R,2R)-RESCA-TFP Wong, Nicholas; Zhao, Eileen; Bao, Jiangyin; Koenig, Stefan G.; Molinaro, Carmela; Timmerman, Jacob C.; Zhang, Haiming; Sowell, C. Gregory; Gosselin, Francis 分享 收藏
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The η-sweet-spot (ηmax) in liquid-assisted mechanochemistry: polymorph control and the role of a liquid additive as either a catalyst or an inhibitor in resonant acoustic mixing (RAM) Gonnet, Lori; Borchers, Tristan H.; Lennox, Cameron B.; Vainauskas, Jogirdas; Teoh, Yong; Titi, Hatem M.; Barrett, Christopher J.; Koenig, Stefan G.; Nagapudi, Karthik; Friscic, Tomislav 分享 收藏
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