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Stefan G. Koenig

roche holding

30H指数
105论文数
3.1K被引数
收录论文 46
发表时间
Establishing Parameters for Resonant Acoustic Mixing (RAM) Chemistry using Buchwald-Hartwig Amination as a Model建立用于共振声波混合(RAM)化学的参数:以Buchwald-Hartwig胺化反应为模型
err2026-02-25
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errOAAI
errLori Gonnet; Cameron B. Lennox; Tristan H Borchers; Mohammad Askari; Alexander Wahrhaftig-Lewis; Stefan G Koenig; Karthik Nagapudi; Tomislav Friščić
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PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models (vol 67, pg 1262, 2024)PROTACs靶向BRM(SMARCA2)可在体内实现对BRG1(SMARCA4)的选择性降解,并在BRG1突变异种移植肿瘤模型中表现出活性(vol 67, pg 1262, 2024)
err2025-05-21
err0
PREAI
errBerlin, Michael; Cantley, Jennifer; Bookbinder, Mark; Bortolon, Elizabeth; Broccatelli, Fabio; Cadelina, Greg; Chan, Emily W.; Chen, Huifen; Chen, Xin; Cheng, Yunxing; Cheung, Tommy K.; Crew, Andrew P.; Davenport, Kim; Dinicola, Dean; Dong, Hanqing; Gordon, Debbie; Hamman, Brian D.; Harbin, Alicia; Haskell, Roy; He, Mingtao; Hole, Alison J.; Januario, Thomas; Kerry, Philip S.; Koenig, Stefan G.; Li, Limei; Merchant, Mark; Perez-Dorado, Inmaculada; Pizzano, Jennifer; Quinn, Connor; Rose, Christopher M.; Rousseau, Emma; Snyder, Lawrence B.; Soto, Leofal; Staben, Leanna R.; Sun, Hongming; Tian, Qingping; Wang, Gan; Wang, Jing; Wang, Weifeng; Ye, Crystal S.; Ye, Xiaofen; Zhang, Penghong; Zhou, Yuhui; Yauch, Robert; Dragovich, Peter S.
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Development of a Broadly Applicable Enzymatic Ligation Process for the Production of Single Guide RNAs开发一种广泛适用的酶促连接过程用于单链引导RNA的生产
err2025-05-05
err0
PREAI
errBigatti, Martina; Moser, Andre; Dierssen, Bas; Frrokaj, Shtjefen; Covato, Elena; Pfleger, Christophe; Lill, Joerg; Leiser, Yael; Zuber, Joel; Staempfli, Andreas; Sladojevich, Filippo; Koenig, Stefan G.
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Redox-Neutral, Iron-Mediated Directed C-H Activation: General Principles and Mechanistic Insights
err2024-10-25
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PREAI
errZhang, Tianyi; Whitehurst, William G.; Pecoraro, Matthew V.; Kim, Junho; Koenig, Stefan G.; Chirik, Paul J.
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Process Mass Intensity (PMI): A Holistic Analysis of Current Peptide Manufacturing Processes Informs Sustainability in Peptide Synthesis过程质量强度 (PMI): 对当前肽制造过程的整体分析为肽合成的可持续性提供了信息
err2024-03-20
err28
errOAAI
errKekessie, Ivy; Wegner, Katarzyna; Martinez, Isamir; Kopach, Michael E.; White, Timothy D.; Tom, Janine K.; Kenworthy, Martin N.; Gallou, Fabrice; Lopez, John; Koenig, Stefan G.; Payne, Philippa R.; Eissler, Stefan; Arumugam, Balasubramanian; Li, Changfeng; Mukherjee, Subha; Isidro-Llobet, Albert; Ludemann-Hombourger, Olivier; Richardson, Paul; Kittelmann, Jorg; Pedersen, Daniel Sejer; van den Bos, Leendert J.
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PROTACs Targeting BRM (SMARCA2) Afford Selective In Vivo Degradation over BRG1 (SMARCA4) and Are Active in BRG1 Mutant Xenograft Tumor Models
err2024-01-05
err7
PREAI
errBerlin, Michael; Cantley, Jennifer; Bookbinder, Mark; Bortolon, Elizabeth; Broccatelli, Fabio; Cadelina, Greg; Chan, Emily W.; Chen, Huifen; Chen, Xin; Cheng, Yunxing; Cheung, Tommy K.; Davenport, Kim; DiNicola, Dean; Gordon, Debbie; Hamman, Brian D.; Harbin, Alicia; Haskell, Roy; He, Mingtao; Hole, Alison J.; Januario, Thomas; Kerry, Philip S.; Koenig, Stefan G.; Li, Limei; Merchant, Mark; Perez-Dorado, Inmaculada; Pizzano, Jennifer; Quinn, Connor; Rose, Christopher M.; Rousseau, Emma; Soto, Leofal; Staben, Leanna R.; Sun, Hongming; Tian, Qingping; Wang, Jing; Wang, Weifeng; Ye, Crystal S.; Ye, Xiaofen; Zhang, Penghong; Zhou, Yuhui; Yauch, Robert; Dragovich, Peter S.
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Characterization of antisense oligonucleotide and guide ribonucleic acid diastereomers by hydrophilic interaction liquid chromatography coupled to mass spectrometry
err2023-10-01
err23
PREAI
errGoyon, Alexandre; Blevins, Molly S.; Napolitano, Jose G.; Nguyen, Daniel; Goel, Meenakshi; Scott, Brandon; Wang, Jenny; Koenig, Stefan G.; Chen, Tao; Zhang, Kelly
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Practical Synthesis of Reactive Immuno-PET Linker-Chelator (1R,2R)-RESCA-TFP
err2023-06-28
err2
PREAI
errWong, Nicholas; Zhao, Eileen; Bao, Jiangyin; Koenig, Stefan G.; Molinaro, Carmela; Timmerman, Jacob C.; Zhang, Haiming; Sowell, C. Gregory; Gosselin, Francis
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Resonant acoustic mixing (RAM) for efficient mechanoredox catalysis without grinding or impact media
err2023-01-01
err26
errOAAI
errEffaty, Farshid; Gonnet, Lori; Koenig, Stefan G.; Nagapudi, Karthik; Ottenwaelder, Xavier; Friscic, Tomislav
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Direct mechanocatalysis by resonant acoustic mixing (RAM)
err2023-01-01
err16
errOAAI
errLennox, Cameron B.; Borchers, Tristan H.; Gonnet, Lori; Barrett, Christopher J.; Koenig, Stefan G.; Nagapudi, Karthik; Friscic, Tomislav
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The η-sweet-spot (ηmax) in liquid-assisted mechanochemistry: polymorph control and the role of a liquid additive as either a catalyst or an inhibitor in resonant acoustic mixing (RAM)
err2023-01-01
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PREAI
errGonnet, Lori; Borchers, Tristan H.; Lennox, Cameron B.; Vainauskas, Jogirdas; Teoh, Yong; Titi, Hatem M.; Barrett, Christopher J.; Koenig, Stefan G.; Nagapudi, Karthik; Friscic, Tomislav
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C-H Activation by Isolable Cationic Bis(phosphine) Cobalt(III) Metallacycles
err2022-10-04
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errOAAI
errWhitehurst, William G.; Kim, Junho; Koenig, Stefan G.; Chirik, Paul J.
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Development of Dual Practical Manufacturing Routes to Cognate Pyrrolobenzodiazepine-Based Linker-Drugs开发基于吡咯并苯并二氮杂的同源接头药物的双重实际制造路线
err2022-08-08
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PREAI
errKoenig, Stefan G.; Angelaud, Remy; Crittenden, Christopher M.; Kurita, Kenji; Russell, David J.; Marcoux, Jean-Francois; Matt, Thomas; Gosselin, Francis
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Challenges in the structure determination of a dimeric impurity found during development of GDC-0326
err2022-05-01
err1
PREAI
errSegraves, Nathaniel L.; Koenig, Stefan G.; Stults, Jeffrey; Ma, Shengli; DiPasquale, Antonio G.; Robinson, Sarah J.; Russell, David J.
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Metal-Catalyzed Organic Reactions by Resonant Acoustic Mixing**
err2022-02-09
err31
PREAI
errGonnet, Lori; Lennox, Cameron B.; Do, Jean-Louis; Malvestiti, Ivani; Koenig, Stefan G.; Nagapudi, Karthik; Friscic, Tomislav
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Sustainable Chemistry and Engineering in Pharma
err2021-10-11
err7
errOAAI
errMartin-Matute, Belen; Meier, Michael A. R.; Metro, Thomas-Xavier; Koenig, Stefan G.; Sneddon, Helen F.; Sudarsanam, Putla; Watts, Paul
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An Efficient Second-Generation Manufacturing Process for the pan-RAF Inhibitor Belvarafenib
err2021-09-11
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PREAI
errZell, Daniel; Dalziel, Michael E.; Carrera, Diane E.; Stumpf, Andreas; Bachmann, Stephan; Mercado-Marin, Eduardo; Koenig, Stefan G.; Zhang, Haiming; Gosselin, Francis
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