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收藏Multi-Modal Design, Synthesis, and Biological Evaluation of Novel Fusidic Acid Derivatives多模态设计、合成及新型 fusidic acid 衍生物的生物评价
Wang, Luqi; Geng, Zhiyuan; Liu, Yuhang; Cao, Linhui; Liu, Yao; Zhang, Hourui; Bi, Yi; Lu, Jing
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收藏Rational Design of the First Dual Agonist at Trace Amine-Associated Receptor 1 and 5-HT2C Receptors Based on Binding Pocket Similarity for the Treatment of Schizophrenia and Alzheimer's Disease-Related Psychosis基于结合口袋相似性的首例双靶点激动剂(Trace Amine-Associated Receptor 1和5-HT2C Receptors)的理性设计,用于治疗精神分裂症和阿尔茨海默病相关精神病
Lu, Jing; Yu, Pengfei; Wang, Yunjie; Dai, Yusen; Wang, Wenyan; Liu, Chunjiao; Dong, Lin; Lei, Hui; Yang, Yifei; Wang, Lin; Zou, Fangxia; Deng, Xuan; Wang, Bingsi; Wei, Shujuan; Ma, Mingxu; Wang, Hongbo; Ye, Liang; Zhang, Jianzhao; Tian, Jingwei
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收藏Phylogeny-Informed Discovery of New Glycopeptide Antibiotics Produced by a Minimal Biosynthetic Gene Cluster
Li, Xingkun; Wang, Mengru; Yin, Lixin; Cao, Jiawei; Wang, Rui; Guo, Wei; Lu, Jing; Zhao, Zhilong; Deng, Zixin; Hou, Anwei; Xu, Min
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收藏Discovery of the thieno[2,3-d]pyrimidine-2,4-dione derivative 21a: A potent and orally bioavailable gonadotropin-releasing hormone receptor antagonist
Zou, Fangxia; Wang, Yao; Yu, Dawei; Liu, Chunjiao; Lu, Jing; Zhao, Min; Ma, Mingxu; Wang, Wenyan; Jiang, Wanglin; Gao, Yonglin; Zhang, Rui; Zhang, Jianzhao; Ye, Liang; Tian, Jingwei
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收藏Natural product 1,2,3,4,6-penta-O-galloyl-β-D-glucopyranose is a reversible inhibitor of glyceraldehyde 3-phosphate dehydrogenase
Li, Wen; Liao, Li-ping; Song, Ning; Liu, Yan-jun; Ding, Yi-luan; Zhang, Yuan-yuan; Zhou, Xiao-ru; Sun, Zhong-ya; Xiao, Sen-hao; Wang, Hong-bo; Lu, Jing; Zhang, Nai-xia; Jiang, Hua-liang; Chen, Kai-xian; Liu, Chuan-peng; Zheng, Jie; Zhao, Ke-hao; Luo, Cheng
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收藏Benzothiazole Amides as TRPC3/6 Inhibitors for Gastric Cancer Treatment
Wei, Yingjie; Zhang, Mengxian; Lyu, Zhenbin; Yang, Guolin; Tian, Tian; Ding, Mingmin; Zeng, Xiaodong; Xu, Fuchun; Wang, Pengyu; Li, Fangfang; Liu, Yixuan; Cao, Zhengyu; Lu, Jing; Hong, Xuechuan; Wang, Hongbo
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收藏Discovery of a novel 53BP1 inhibitor through AlphaScreen-based high-throughput screening通过基于AlphaScreen的高通量筛选发现新型53BP1抑制剂
Sun, Yanli; Lu, Haibo; Fang, Xueyu; Xiao, Senhao; Yang, Feng; Chen, Yantao; Wang, Hongbo; Li, Xiaopeng; Lu, Jing; Lin, Hua; Luo, Cheng; Zhao, Kehao; Chen, Shijie
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收藏Design, synthesis, and discovery of ocotillol-type amide derivatives as orally available modulators of P-glycoprotein-mediated multidrug resistance
Ren, Qianwen; Yang, Gangqiang; Guo, Mengqi; Guo, Jingwen; Li, Yang; Lu, Jing; Yang, Qing; Tang, Hanhan; Li, Yi; Fang, Xiaojuan; Sun, Yixiao; Qi, Jia Grace; Tian, Jingwei; Wang, Hongbo
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收藏H6, a novel hederagenin derivative, reverses multidrug resistance in vitro and in vivo
Yang, Yanting; Guan, Daokun; Lei, Lei; Lu, Jing; Liu, Jia Qi; Yang, Gangqiang; Yan, Chunhong; Zhai, Rong; Tian, Jingwei; Bi, Yi; Fu, Fenghua; Wang, Hongbo
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