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收藏Design, synthesis, and antiviral activity of fragmented-lapatinib aminoquinazoline analogs towards SARS-CoV-2 inhibition
Adediji, Ayomide; Sroithongmoon, Akeanan; Suroengrit, Aphinya; Wilasluck, Patcharin; Deetanya, Peerapon; Sanachai, Kamonpan; Karnchanapandh, Kun; Boonyasuppayakorn, Siwaporn; Wangkanont, Kittikhun; Rungrotmongkol, Thanyada; Khotavivattana, Tanatorn
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收藏Unveiling the antiviral inhibitory activity of ebselen and ebsulfur derivatives on SARS-CoV-2 using machine learning-based QSAR, LB-PaCS-MD, and experimental assay
Sinsulpsiri, Silpsiri; Nishii, Yuji; Xu-Xu, Qing-Feng; Miura, Masahiro; Wilasluck, Patcharin; Salamteh, Kanokwan; Deetanya, Peerapon; Wangkanont, Kittikhun; Suroengrit, Aphinya; Boonyasuppayakorn, Siwaporn; Duan, Lian; Harada, Ryuhei; Hengphasatporn, Kowit; Shigeta, Yasuteru; Shi, Liyi; Maitarad, Phornphimon; Rungrotmongkol, Thanyada
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收藏Design, Synthesis, and Biological Evaluation of Darunavir Analogs as HIV-1 Protease Inhibitors
Rehman, Muhammad Asad Ur; Chuntakaruk, Hathaichanok; Amphan, Soraat; Suroengrit, Aphinya; Hengphasatporn, Kowit; Shigeta, Yasuteru; Rungrotmongkol, Thanyada; Krusong, Kuakarun; Boonyasuppayakorn, Siwaporn; Aonbangkhen, Chanat; Khotavivattana, Tanatorn
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收藏Alpha and gamma mangostins inhibit wild-type B SARS-CoV-2 more effectively than the SARS-CoV-2 variants and the major target is unlikely the 3C-like protease
Suroengrit, Aphinya; Cao, Van; Wilasluck, Patcharin; Deetanya, Peerapon; Wangkanont, Kittikhun; Hengphasatporn, Kowit; Harada, Ryuhei; Chamni, Supakarn; Leelahavanichkul, Asada; Shigeta, Yasuteru; Rungrotmongkol, Thanyada; Hannongbua, Supot; Chavasiri, Warinthorn; Wacharapluesadee, Supaporn; Prompetchara, Eakachai; Boonyasuppayakorn, Siwaporn
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收藏The 8-bromobaicalein alleviated chikungunya-induced musculoskeletal inflammation and reduced the viral load in healthy adult mice
Cao, Van; Loeanurit, Naphat; Hengphasatporn, Kowit; Hairani, Rita; Wacharachaisurapol, Noppadol; Prompila, Nantaporn; Wittayalertpanya, Supeecha; Shigeta, Yasuteru; Khotavivattana, Tanatorn; Chavasiri, Warinthorn; Boonyasuppayakorn, Siwaporn
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收藏Identification of Promising Sulfonamide Chalcones as Inhibitors of SARS-CoV-2 3CLpro through Structure-Based Virtual Screening and Experimental Approaches
Pojtanadithee, Piyatida; Hengphasatporn, Kowit; Suroengrit, Aphinya; Boonyasuppayakorn, Siwaporn; Wilasluck, Patcharin; Deetanya, Peerapon; Wangkanont, Kittikhun; Sukanadi, I. Putu; Chavasiri, Warinthorn; Wolschann, Peter; Langer, Thierry; Shigeta, Yasuteru; Maitarad, Phornphimon; Sanachai, Kamonpan; Rungrotmongkol, Thanyada
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收藏The 8-bromobaicalein inhibited the replication of dengue, and Zika viruses and targeted the dengue polymerase (Mar, 10.1038/s41598-023-32049-x, 2023)
Boonyasuppayakorn, Siwaporn; Saelee, Thanaphon; Huynh, Thao Nguyen Thanh; Hairani, Rita; Hengphasatporn, Kowit; Loeanurit, Naphat; Cao, Van; Vibulakhaophan, Vipanee; Siripitakpong, Panattida; Kaur, Parveen; Chu, Justin Jang Hann; Tunghirun, Chairat; Choksupmanee, Opas; Chimnaronk, Sarin; Shigeta, Yasuteru; Rungrotmongkol, Thanyada; Chavasiri, Warinthorn
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收藏The 8-bromobaicalein inhibited the replication of dengue, and Zika viruses and targeted the dengue polymerase
Boonyasuppayakorn, Siwaporn; Saelee, Thanaphon; Huynh, Thao Nguyen Thanh; Hairani, Rita; Hengphasatporn, Kowit; Loeanurit, Naphat; Cao, Van; Vibulakhaophan, Vipanee; Siripitakpong, Panattida; Kaur, Parveen; Chu, Justin Jang Hann; Tunghirun, Chairat; Choksupmanee, Opas; Chimnaronk, Sarin; Shigeta, Yasuteru; Rungrotmongkol, Thanyada; Chavasiri, Warinthorn
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收藏Lichen-Derived Diffractaic Acid Inhibited Dengue Virus Replication in a Cell-Based System
Loeanurit, Naphat; Tuong, Truong Lam; Nguyen, Van-Kieu; Vibulakhaophan, Vipanee; Hengphasatporn, Kowit; Shigeta, Yasuteru; Ho, Si Xian; Chu, Justin Jang Hann; Rungrotmongkol, Thanyada; Chavasiri, Warinthorn; Boonyasuppayakorn, Siwaporn
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收藏Design, synthesis, in vitro, in silico, and SAR studies of flavone analogs towards anti-dengue activity
Patigo, Apinya; Hengphasatporn, Kowit; Cao, Van; Paunrat, Wattamon; Vijara, Natthanan; Chokmahasarn, Thamonwan; Maitarad, Phornphimon; Rungrotmongkol, Thanyada; Shigeta, Yasuteru; Boonyasuppayakorn, Siwaporn; Khotavivattana, Tanatorn
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收藏Promising SARS-CoV-2 main protease inhibitor ligand-binding modes evaluated using LB-PaCS-MD/FMO
Hengphasatporn, Kowit; Harada, Ryuhei; Wilasluck, Patcharin; Deetanya, Peerapon; Sukandar, Edwin R.; Chavasiri, Warinthorn; Suroengrit, Aphinya; Boonyasuppayakorn, Siwaporn; Rungrotmongkol, Thanyada; Wangkanont, Kittikhun; Shigeta, Yasuteru
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收藏Semi-Synthesis of N-Aryl Amide Analogs of Piperine from Piper nigrum and Evaluation of Their Antitrypanosomal, Antimalarial, and Anti-SARS-CoV-2 Main Protease Activities
Wansri, Rattanaporn; Lin, Aye Chan Khine; Pengon, Jutharat; Kamchonwongpaisan, Sumalee; Srimongkolpithak, Nitipol; Rattanajak, Roonglawan; Wilasluck, Patcharin; Deetanya, Peerapon; Wangkanont, Kittikhun; Hengphasatporn, Kowit; Shigeta, Yasuteru; Liangsakul, Jatupol; Suroengrit, Aphinya; Boonyasuppayakorn, Siwaporn; Chuanasa, Taksina; De-Eknamkul, Wanchai; Hannongbua, Supot; Rungrotmongkol, Thanyada; Chamni, Supakarn
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