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New Pyridobenothiazolone Derivatives Display Nanomolar Pan-Serotype Anti-Dengue Virus Activity Felicetti, Tommaso; Gwee, Chin Piaw; Chan, Kitti Wing Ki; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Watanabe, Satoru; Mazlan, Muhammad Danial Bin Mohd; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Sbardella, Gianluca; Vasudevan, Subhash G.; Manfroni, Giuseppe 分享 收藏
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The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit to Lead 欧洲药物化学和化学生物学联合会 (EFMC) 最佳实践倡议: 领先 Quancard, Jean; Bach, Anders; Borsari, Chiara; Craft, Russell; Gnamm, Christian; Gueret, Stephanie M.; Hartung, Ingo V.; Koolman, Hannes F.; Laufer, Stefan; Lepri, Susan; Messinger, Josef; Ritter, Kurt; Sbardella, Gianluca; Lopez, Andrea Unzue; Willwacher, Marina K.; Cox, Brian; Young, Robert J. 分享 收藏
Prodrug Approach to Exploit (S)-Alanine Amide as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors. Milite, Ciro; Sarno, Giuliana; Pacilio, Ida; Cianciulli, Agostino; Viviano, Monica; Iannelli, Giulia; Gazzillo, Erica; Feoli, Alessandra; Cipriano, Alessandra; Giovanna Chini, Maria; Castellano, Sabrina; Bifulco, Giuseppe; Sbardella., Gianluca 分享 收藏
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Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor Feoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L.; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G.; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca 分享 收藏
First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8 赖氨酸乙酰转移酶KAT8的一流选择性抑制剂 Fiorentino, Francesco; Sementilli, Sara; Menna, Martina; Turrisi, Federica; Tomassi, Stefano; Pellegrini, Francesca Romana; Iuzzolino, Angela; D'Acunzo, Francesca; Feoli, Alessandra; Wapenaar, Hannah; Taraglio, Sophie; Fraschetti, Caterina; Del Bufalo, Donatella; Sbardella, Gianluca; Dekker, Frank J.; Paiardini, Alessandro; Trisciuoglio, Daniela; Mai, Antonello; Rotili, Dante 分享 收藏
The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit Generation Quancard, Jean; Vulpetti, Anna; Bach, Anders; Cox, Brian; Gueret, Stephanie M.; Hartung, Ingo V.; Koolman, Hannes F.; Laufer, Stefan; Messinger, Josef; Sbardella, Gianluca; Craft, Russell 分享 收藏
Discovery of Benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca 分享 收藏
Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models Menna, Martina; Fiorentino, Francesco; Marrocco, Biagina; Lucidi, Alessia; Tomassi, Stefano; Cilli, Domenica; Romanenghi, Mauro; Cassandri, Matteo; Pomella, Silvia; Pezzella, Michele; Del Bufalo, Donatella; Ansari, Mohammad Salik Zeya; Tomasevic, Nevena; Mladenovic, Milan; Viviano, Monica; Sbardella, Gianluca; Rota, Rossella; Trisciuoglio, Daniela; Minucci, Saverio; Mattevi, Andrea; Rotili, Dante; Mai, Antonello 分享 收藏
Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction- Reconstruction and Fragment-Growing Approach Iannelli, Giulia; Milite, Ciro; Marechal, Nils; Cura, Vincent; Bonnefond, Luc; Troffer-Charlier, Nathalie; Feoli, Alessandra; Rescigno, Donatella; Wang, Yalong; Cipriano, Alessandra; Viviano, Monica; Bedford, Mark T.; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca 分享 收藏
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The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Phenotypic Drug Discovery Quancard, Jean; Bach, Anders; Cox, Brian; Craft, Russell; Finsinger, Dirk; Gueret, Stephanie M.; Hartung, Ingo V.; Laufer, Stefan; Messinger, Josef; Sbardella, Gianluca; Koolman, Hannes F. 分享 收藏