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Gianluca Sbardella

university of salerno

42H指数
183论文数
4.7K被引数
收录论文 78
发表时间
2-Phenylquinolines Exhibit Anti-Severe Acute Respiratory Syndrome Coronavirus-2 Activity Through the Nonstructural Protein 13 Helicase Inhibition2-苯基喹啉通过非结构蛋白13解旋酶抑制表现出抗严重急性呼吸综合征冠状病毒2活性
err2026-04-10
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errOAAI
errGiada Cernicchi; Maria Giulia Nizi; Roberta Emmolo; Leentje Persoons; Manon Laporte; Dirk Jochmans; Isabella Romeo; Giacomo Pepe; Ciro Milite; Pietro Campiglia; Jacopo Spezzini; Alma Martelli; Simone Brogi; Francesca Esposito; Tommaso Felicetti; Serena Massari; Giuseppe Manfroni; Stefano Sabatini; Gianluca Sbardella; Stefano Alcaro; Johan Neyts; Angela Corona; Enzo Tramontano; Steven De Jonghe; Oriana Tabarrini
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Dynamic epigenetic regulation of BCLAF1 splicing in acute myeloid leukemia急性髓系白血病中BCLAF1剪接的动态表观遗传调控
err2026-03-24
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errOAAI
errGiulia Sgueglia; Crescenzo Massaro; Annamaria Muro; Ida Lettiero; Erika D’Agostino; Gregorio Favale; Nicla Simonelli; Nunzio Del Gaudio; Vincenzo Carafa; Tommaso De Marchi; Dante Rotili; Sergio Valente; Antonello Mai; Gianluca Sbardella; Mariacarla De Simone; Lucia Altucci; Carmela Dell’Aversana
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Sulfonyl Anthranilic Acid Analogues Display Pan-Serotype Anti-Dengue Activity by Downregulating the Expression of Ribosomal Proteins Encoded by 5′-Terminal Oligopyrimidine Motif-Containing mRNA磺酰基邻氨基苯甲酸类似物通过下调含有5′-端寡聚嘧啶基序的mRNA编码的核糖体蛋白的表达,显示出泛血清型抗登革病毒活性。
err2026-03-10
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errChin Piaw Gwee; Tommaso Felicetti; Kitti Wing Ki Chan; Min Jie Alvin Tan; Muhammad Danial Bin Mohd Mazlan; Ciro Milite; Giacomo Pepe; Chiara Sarnari; Xiao Dan Ng; Wint Wint Phoo; Jasmine Hwee Yee Tan; Marcus G. Mah; Satoru Watanabe; Jing Xiu Huang; Serena Massari; Oriana Tabarrini; Stefano Sabatini; Pietro Campiglia; Gianluca Sbardella; Gavin J. D. Smith; Sylvie Alonso; Alfred Xuyang Sun; Radoslaw M. Sobota; Subhash G. Vasudevan; Giuseppe Manfroni
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Ferroptosis and Autophagy-Dependent Cell Death in Oncology Medicinal Chemistry: Call for Papers
err2026-01-08
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PREAI
errGiustiniano, Mariateresa; Neamati, Nouri; Sbardella, Gianluca; Bolognesi, Maria Laura
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Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses开发具有抗呼吸道病毒保护作用的Type II F508del-CFTR纠正剂
err2025-08-28
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errFrancesca Barbieri; Maria Grazia Martina; Emanuela Pesce; Elena Bianchi; Noemi Cabella; Emmanuele Crespan; Sara Rossi; Sandra Gemma; Giuseppe Campiani; Ciro Milite; Giacomo Pepe; Pietro Campiglia; Gianluca Sbardella; Giovanni Maga; Valeria Cagno; Nicoletta Pedemonte; Marco Radi
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New Pyridobenothiazolone Derivatives Display Nanomolar Pan-Serotype Anti-Dengue Virus Activity
err2025-04-01
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PREAI
errFelicetti, Tommaso; Gwee, Chin Piaw; Chan, Kitti Wing Ki; Pepe, Giacomo; Milite, Ciro; Campiglia, Pietro; Watanabe, Satoru; Mazlan, Muhammad Danial Bin Mohd; Sabatini, Stefano; Massari, Serena; Tabarrini, Oriana; Sbardella, Gianluca; Vasudevan, Subhash G.; Manfroni, Giuseppe
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The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit to Lead欧洲药物化学和化学生物学联合会 (EFMC) 最佳实践倡议: 领先
err2025-02-16
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PREAI
errQuancard, Jean; Bach, Anders; Borsari, Chiara; Craft, Russell; Gnamm, Christian; Gueret, Stephanie M.; Hartung, Ingo V.; Koolman, Hannes F.; Laufer, Stefan; Lepri, Susan; Messinger, Josef; Ritter, Kurt; Sbardella, Gianluca; Lopez, Andrea Unzue; Willwacher, Marina K.; Cox, Brian; Young, Robert J.
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Prodrug Approach to Exploit (S)-Alanine Amide as Arginine Mimic Moiety in the Development of Protein Arginine Methyltransferase 4 Inhibitors.
err2024-06-25
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errMilite, Ciro; Sarno, Giuliana; Pacilio, Ida; Cianciulli, Agostino; Viviano, Monica; Iannelli, Giulia; Gazzillo, Erica; Feoli, Alessandra; Cipriano, Alessandra; Giovanna Chini, Maria; Castellano, Sabrina; Bifulco, Giuseppe; Sbardella., Gianluca
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Successes and challenges in the development of BD1-selective BET inhibitors: a patent review
err2024-03-11
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PREAI
errViviano, Monica; Cipriano, Alessandra; Fabbrizi, Emanuele; Feoli, Alessandra; Castellano, Sabrina; Sbardella, Gianluca; Mai, Antonello; Milite, Ciro; Rotili, Dante
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NADPH Oxidases: From Molecular Mechanisms to Current Inhibitors
err2023-08-31
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errCipriano, Alessandra; Viviano, Monica; Feoli, Alessandra; Milite, Ciro; Sarno, Giuliana; Castellano, Sabrina; Sbardella, Gianluca
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Identification of a Protein Arginine Methyltransferase 7 (PRMT7)/Protein Arginine Methyltransferase 9 (PRMT9) Inhibitor
err2023-08-10
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errFeoli, Alessandra; Iannelli, Giulia; Cipriano, Alessandra; Milite, Ciro; Shen, Lei; Wang, Zhihao; Hadjikyriacou, Andrea; Lowe, Troy L.; Safaeipour, Cyrus; Viviano, Monica; Sarno, Giuliana; Morretta, Elva; Monti, Maria Chiara; Yang, Yanzhong; Clarke, Steven G.; Cosconati, Sandro; Castellano, Sabrina; Sbardella, Gianluca
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First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8赖氨酸乙酰转移酶KAT8的一流选择性抑制剂
err2023-05-08
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errFiorentino, Francesco; Sementilli, Sara; Menna, Martina; Turrisi, Federica; Tomassi, Stefano; Pellegrini, Francesca Romana; Iuzzolino, Angela; D'Acunzo, Francesca; Feoli, Alessandra; Wapenaar, Hannah; Taraglio, Sophie; Fraschetti, Caterina; Del Bufalo, Donatella; Sbardella, Gianluca; Dekker, Frank J.; Paiardini, Alessandro; Trisciuoglio, Daniela; Mai, Antonello; Rotili, Dante
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The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Hit Generation
err2023-03-09
err8
PREAI
errQuancard, Jean; Vulpetti, Anna; Bach, Anders; Cox, Brian; Gueret, Stephanie M.; Hartung, Ingo V.; Koolman, Hannes F.; Laufer, Stefan; Messinger, Josef; Sbardella, Gianluca; Craft, Russell
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Discovery of Benzo[d]imidazole-6-sulfonamides as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain
err2022-09-15
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errCipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca
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Novel non-covalent LSD1 inhibitors endowed with anticancer effects in leukemia and solid tumor cellular models
err2022-07-01
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errMenna, Martina; Fiorentino, Francesco; Marrocco, Biagina; Lucidi, Alessia; Tomassi, Stefano; Cilli, Domenica; Romanenghi, Mauro; Cassandri, Matteo; Pomella, Silvia; Pezzella, Michele; Del Bufalo, Donatella; Ansari, Mohammad Salik Zeya; Tomasevic, Nevena; Mladenovic, Milan; Viviano, Monica; Sbardella, Gianluca; Rota, Rossella; Trisciuoglio, Daniela; Minucci, Saverio; Mattevi, Andrea; Rotili, Dante; Mai, Antonello
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Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction- Reconstruction and Fragment-Growing Approach
err2022-04-28
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errIannelli, Giulia; Milite, Ciro; Marechal, Nils; Cura, Vincent; Bonnefond, Luc; Troffer-Charlier, Nathalie; Feoli, Alessandra; Rescigno, Donatella; Wang, Yalong; Cipriano, Alessandra; Viviano, Monica; Bedford, Mark T.; Cavarelli, Jean; Castellano, Sabrina; Sbardella, Gianluca
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Lysine methyltransferase inhibitors: where we are now
err2022-01-01
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errFeoli, Alessandra; Viviano, Monica; Cipriano, Alessandra; Milite, Ciro; Castellano, Sabrina; Sbardella, Gianluca
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The European Federation for Medicinal Chemistry and Chemical Biology (EFMC) Best Practice Initiative: Phenotypic Drug Discovery
err2021-04-07
err10
PREAI
errQuancard, Jean; Bach, Anders; Cox, Brian; Craft, Russell; Finsinger, Dirk; Gueret, Stephanie M.; Hartung, Ingo V.; Laufer, Stefan; Messinger, Josef; Sbardella, Gianluca; Koolman, Hannes F.
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