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Marc A. Giulianotti

sierra space corp.

33H指数
147论文数
4.8K被引数
收录论文 58
发表时间
Biomanufacturing in low Earth orbit: A paradigm shift低地球轨道生物制造:一种范式转变
err2025-06-19
err0
errOAAI
errDavide Marotta; Noor Ward; Steven R. Bauer; Joshua Hunsberger; Jana Stoudemire; Kenneth Savin; Marc Giulianotti; Catriona H.M. Jamieson; Donna Roberts; Michael Roberts
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N-Branched Tricyclic Guanidines as Novel Melanocortin-3 Receptor Agonists and Melanocortin-4 Receptor AntagonistsN-支链三环胍类化合物作为新型促黑激素-3受体激动剂和促黑激素-4受体拮抗剂
err2025-01-20
err0
PREAI
errWeirath, Nicholas A.; Zajac, Jonathan W. P.; Donow, Haley M.; Lavoi, Travis M.; Pinilla, Clemencia; Santos, Radleigh G.; Prajapati, Ritu; Speth, Robert; Ericson, Mark D.; Sarupria, Sapna; Giulianotti, Marcello A.
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Lab on a chip (LOC) platform for drug screening against the intracellular forms of Trypanosoma cruzi
err2024-08-01
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PREAI
errCadena, Maria Fernanda; Rosero-Yanez, Gustavo; Isa-Jara, Ramiro; Belaunzaran, Maria Laura; Giulianotti, Marc A.; Pinilla, Clemencia; Soto, Catalina D. Alba; Perez, Maximiliano; Lerner, Betiana; Gimenez, Guadalupe
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Structure-Activity Relationship of Pyrrolidine Pentamine Derivatives as Inhibitors of the Aminoglycoside 6′-N-Acetyltransferase Type Ib
err2024-07-19
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errOAAI
errSklenicka, Jan; Tran, Tung; Ramirez, Maria S.; Donow, Haley M.; Magana, Angel J.; Lavoi, Travis; Mamun, Yasir; Jimenez, Veronica; Chapagain, Prem; Santos, Radleigh; Pinilla, Clemencia; Giulianotti, Marc A.; Tolmasky, Marcelo E.
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Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High Throughput 'Unbiased' Screening Campaign (vol 64, pg 5577, 2021)
err2023-05-08
err0
errOAAI
errDoering, Skye R.; Freeman, Katie; Debevec, Ginamarie; Geer, Phaedra; Santos, Radleigh G.; Lavoi, Travis M.; Giulianotti, Marc A.; Pinilla, Clemencia; Appel, Jon R.; Houghten, Richard A.; Ericson, Mark D.; Haskell-Luevano, Carrie
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Restoring susceptibility to aminoglycosides: identifying small molecule inhibitors of enzymatic inactivation
err2023-01-01
err6
PREAI
errMagana, Angel J.; Sklenicka, Jan; Pinilla, Clemencia; Giulianotti, Marc; Chapagain, Prem; Santos, Radleigh; Ramirez, Maria Soledad; Tolmasky, Marcelo E.
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Identification of SARS-CoV-2 Spike Palmitoylation Inhibitors That Results in Release of Attenuated Virus with Reduced Infectivity
err2022-03-04
err31
errOAAI
errRamadan, Ahmed A.; Mayilsamy, Karthick; McGill, Andrew R.; Ghosh, Anandita; Giulianotti, Marc A.; Donow, Haley M.; Mohapatra, Shyam S.; Mohapatra, Subhra; Chandran, Bala; Deschenes, Robert J.; Roy, Arunava
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Biomanufacturing in low Earth orbit for regenerative medicine
err2022-01-01
err31
errOAAI
errSharma, Arun; Clemens, Rachel A.; Garcia, Orquidea; Taylor, D. Lansing; Wagner, Nicole L.; Shepard, Kelly A.; Gupta, Anjali; Malany, Siobhan; Grodzinsky, Alan J.; Kearns-Jonker, Mary; Mair, Devin B.; Kim, Deok-Ho; Roberts, Michael S.; Loring, Jeanne F.; Hu, Jianying; Warren, Lara E.; Eenmaa, Sven; Bozada, Joe; Paljug, Eric; Roth, Mark; Taylor, Donald P.; Rodrigue, Gary; Cantini, Patrick; Smith, Amelia W.; Giulianotti, Marc A.; Wagner, William R.
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Identification and characterization of an atypical Gas-biased β2AR agonist that fails to evoke airway smooth muscle cell tachyphylaxis
err2021-12-02
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errOAAI
errKim, Donghwa; Tokmakova, Alina; Lujan, Lauren K.; Strzelinski, Hannah R.; Kim, Nicholas; Beidokhti, Maliheh Najari; Giulianotti, Marc A.; Mafi, Amirhossein; Woo, Jung-A A.; An, Steven S.; Goddard, William A., III; Liggett, Stephen B.
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Functional Mixture-Based Positional Scan Identifies a Library of Antagonist Tetrapeptide Sequences (LAtTeS) with Nanomolar Potency for the Melanocortin-4 Receptor and Equipotent with the Endogenous AGRP(86-132) Antagonist
err2021-09-30
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errOAAI
errEricson, Mark D.; Doering, Skye R.; Larson, Courtney M.; Freeman, Katie T.; LaVoi, Travis M.; Donow, Haley M.; Santos, Radleigh G.; Cho, Rachel H.; Koerperich, Zoe M.; Giulianotti, Marc A.; Pinilla, Clemencia; Houghten, Richard A.; Haskell-Luevano, Carrie
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Inhibition of Aminoglycoside 6′-N-acetyltransferase Type Ib (AAC(6′)-Ib): Structure-Activity Relationship of Substituted Pyrrolidine Pentamine Derivatives as Inhibitors
err2021-09-14
err4
errOAAI
errRocha, Kenneth; Magallon, Jesus; Reeves, Craig; Phan, Kimberly; Vu, Peter; Oakley-Havens, Crista L.; Kwan, Stella; Ramirez, Maria Soledad; LaVoi, Travis; Donow, Haley; Chapagain, Prem; Santos, Radleigh; Pinilla, Clemencia; Giulianotti, Marc A.; Tolmasky, Marcelo E.
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Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High-Throughput Unbiased Screening Campaign
err2021-04-22
err6
errOAAI
errDoering, Skye R.; Freeman, Katie; Debevec, Ginamarie; Geer, Phaedra; Santos, Radleigh G.; Lavoi, Travis M.; Giulianotti, Marc A.; Pinilla, Clemencia; Appel, Jon R.; Houghten, Richard A.; Ericson, Mark D.; Haskell-Luevano, Carrie
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The value of antimicrobial peptides in the age of resistance抗菌肽在耐药时代的价值
err2020-09-01
err693
PREAI
errMagana, Maria; Pushpanathan, Muthuirulan; Santos, Ana L.; Leanse, Leon; Fernandez, Michael; Ioannidis, Anastasios; Giulianotti, Marc A.; Apidianakis, Yiorgos; Bradfute, Steven; Ferguson, Andrew L.; Cherkasov, Artem; Seleem, Mohamed N.; Pinilla, Clemencia; de la Fuente-Nunez, Cesar; Lazaridis, Themis; Dai, Tianhong; Houghten, Richard A.; Hancock, Robert E. W.; Tegos, George P.
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A Novel Class of Common Docking Domain Inhibitors That Prevent ERK2 Activation and Substrate Phosphorylation
err2019-05-06
err23
errOAAI
errSammons, Rachel M.; Perry, Nicole A.; Li, Yangmei; Cho, Eun Jeong; Piserchio, Andrea; Zamora-Olivares, Diana P.; Ghose, Ranajeet; Kaoud, Tamer S.; Debevec, Ginamarie; Bartholomeusz, Chandra; Gurevich, Vsevolod V.; Iverson, Tina M.; Giulianotti, Marc; Houghten, Richard A.; Dalby, Kevin N.
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Discovery of Polypharmacological Melanocortin-3 and-4 Receptor Probes and Identification of a 100-Fold Selective nM MC3R Agonist versus a μM MC4R Partial Agonist
err2019-02-11
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errOAAI
errFleming, Katlyn A.; Freeman, Katie T.; Powers, Mike D.; Santos, Radleigh G.; Debevec, Ginamarie; Giulianotti, Marc A.; Houghten, Richard A.; Doering, Skye R.; Pinilla, Clemencia; Haskell-Luevano, Carrie
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Scaffold Ranking and Positional Scanning Identify Novel Neurite Outgrowth Promoters with Nanomolar Potency
err2018-09-24
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errOAAI
errAl-Ali, Hassan; Debevec, Ginamarie; Santos, Radleigh G.; Houghten, Richard A.; Davis, Jennifer C.; Nefzi, Adel; Lemmon, Vance P.; Bixby, John L.; Giulianotti, Marc A.
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Identification of a Novel Polyamine Scaffold With Potent Efflux Pump Inhibition Activity Toward Multi-Drug Resistant Bacterial Pathogens
err2018-06-14
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errOAAI
errFleeman, Renee M.; Debevec, Ginamarie; Antonen, Kirsten; Adams, Jessie L.; Santos, Radleigh G.; Welmaker, Gregory S.; Houghten, Richard A.; Giulianotti, Marc A.; Shaw, Lindsey N.
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Differential regulation of alcohol taking and seeking by antagonism at α4β2 and α3β4 nAChRs
err2018-03-23
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errOAAI
errCippitelli, Andrea; Brunori, Gloria; Schoch, Jennifer; Armishaw, Christopher J.; Wu, Jinhua; Zaveri, Nurulain T.; Giulianotti, Marc A.; Welmaker, Gregory S.; Toll, Lawrence
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