未登录.png)
分享.png)
收藏分享 收藏 Guanidine Derivative ADS1017, a Potent Histamine H3 Receptor Antagonist with Promising Analgesic Activity and Satisfactory Safety Profile
Karcz, Tadeusz; Szczepanska, Katarzyna; Mogilski, Szczepan; Moroz, Aleksandra; Olejarz-Maciej, Agnieszka; Humphrys, Laura J.; Pockes, Steffen; Siwek, Agata; Dubiel, Krzysztof; Staszewski, Marek; Calmels, Thierry; Waczynski, Krzysztof; Kiec-Kononowicz, Katarzyna 分享 收藏 分享 收藏 Discovery of New Highly Potent Histamine H3 Receptor Antagonists, Calcium Channel Blockers, and Acetylcholinesterase InhibitorsMalek, Rim; Salat, Kinga; Totoson, Perle; Karcz, Tadeusz; Refouvelet, Bernard; Skrzypczak-Wiercioch, Anna; Maj, Maciej; Simakov, Alexey; Martin, Helene; Siwek, Agata; Szalaj, Natalia; Godyn, Justyna; Panek, Dawid; Wieckowska, Anna; Jozwiak, Krzysztof; Demougeot, Celine; Kiec-Kononowicz, Katarzyna; Chabchoub, Fakher; Iriepa, Isabel; Marco-Contelles, Jose; Ismaili, Lhassane 分享 收藏 The Effect of KSK-94, a Dual Histamine H3 and Sigma-2 Receptor Ligand, on Adipose Tissue in a Rat Model of Developing ObesityKotanska, Magdalena; Zadrozna, Monika; Kubacka, Monika; Mika, Kamil; Szczepanska, Katarzyna; Nowak, Barbara; Alesci, Alessio; Miller, Anthea; Lauriano, Eugenia Rita; Kiec-Kononowicz, Katarzyna 分享 收藏 分享 收藏 Potent, Selective Agonists for the Cannabinoid-like Orphan G Protein-Coupled Receptor GPR18: A Promising Drug Target for Cancer and ImmunityMahardhika, Andhika B.; Zaluski, Michal; Schoeder, Clara T.; Boshta, Nader M.; Schabikowski, Jakub; Perri, Filomena; Lazewska, Dorota; Neumann, Alexander; Kremers, Sarah; Oneto, Angelo; Ressemann, Anastasiia; Latacz, Gniewomir; Namasivayam, Vigneshwaran; Kiec-Kononowicz, Katarzyna; Mueller, Christa E. 分享 收藏 分享 收藏 分享 收藏 Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic PainSzczepanska, Katarzyna; Karcz, Tadeusz; Dichiara, Maria; Mogilski, Szczepan; Kalinowska-Tluscik, Justyna; Pilarski, Boguslaw; Leniak, Arkadiusz; Pietrus, Wojciech; Podlewska, Sabina; Popiolek-Barczyk, Katarzyna; Humphrys, Laura J.; Ruiz-Cantero, M. Carmen; Reiner-Link, David; Leitzbach, Luisa; Lazewska, Dorota; Pockes, Steffen; Gorka, Michal; Zmyslowski, Adam; Calmels, Thierry; Cobos, Enrique J.; Marrazzo, Agostino; Stark, Holger; Bojarski, Andrzej J.; Amata, Emanuele; Kiec-Kononowicz, Katarzyna 分享 收藏 Trisubstituted 1,3,5-Triazines as Histamine H4 Receptor Antagonists with Promising Activity In VivoOlejarz-Maciej, Agnieszka; Mogilski, Szczepan; Karcz, Tadeusz; Werner, Tobias; Kaminska, Katarzyna; Kupczyk, Jaroslaw; Honkisz-Orzechowska, Ewelina; Latacz, Gniewomir; Stark, Holger; Kiec-Kononowicz, Katarzyna; Lazewska, Dorota 分享 收藏 Multitargeting Histamine H3 Receptor Ligands among Acetyl- and Propionyl-Phenoxyalkyl DerivativesLazewska, Dorota; Kaleta, Maria; Zareba, Paula; Godyn, Justyna; Dubiel, Mariam; Honkisz-Orzechowska, Ewelina; Doroz-Plonka, Agata; Wieckowska, Anna; Stark, Holger; Kiec-Kononowicz, Katarzyna 分享 收藏 Benzophenone Derivatives with Histamine H3 Receptor Affinity and Cholinesterase Inhibitory Potency as Multitarget-Directed Ligands for Possible Therapy of Alzheimer's DiseaseGodyn, Justyna; Zareba, Paula; Stary, Dorota; Kaleta, Maria; Kuder, Kamil J.; Latacz, Gniewomir; Mogilski, Szczepan; Reiner-Link, David; Frank, Annika; Doroz-Plonka, Agata; Olejarz-Maciej, Agnieszka; Sudol-Talaj, Sylwia; Nolte, Tobias; Handzlik, Jadwiga; Stark, Holger; Wieckowska, Anna; Malawska, Barbara; Kiec-Kononowicz, Katarzyna; Lazewska, Dorota; Bajda, Marek 分享 收藏 Dual Targeting Ligands-Histamine H3 Receptor Ligands with Monoamine Oxidase B Inhibitory Activity-In Vitro and In Vivo EvaluationLasewska, Dorota; Siwek, Agata; Olejarz-Maciej, Agnieszka; Doroz-Plonka, Agata; Wiktorowska-Owczarek, Anna; Jozwiak-Bebenista, Marta; Reiner-Link, David; Frank, Annika; Sromek-Trzaskowska, Wioletta; Honkisz-Orzechowska, Ewelina; Krolicka, Ewelina; Stark, Holger; Wieczorek, Marek; Wagner, Waldemar; Kiec-Kononowicz, Katarzyna; Stasiak, Anna 分享 收藏 分享 收藏 Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H3 and Sigma-1 Receptor Antagonists with Promising Antinociceptive PropertiesSzczepanska, Katarzyna; Podlewska, Sabina; Dichiara, Maria; Gentile, Davide; Patamia, Vincenzo; Rosier, Niklas; Moennich, Denise; Ruiz Cantero, Ma Carmen; Karcz, Tadeusz; Lazewska, Dorota; Siwek, Agata; Pockes, Steffen; Cobos, Enrique J.; Marrazzo, Agostino; Stark, Holger; Rescifina, Antonio; Bojarski, Andrzej J.; Amata, Emanuele; Kiec-Kononowicz, Katarzyna 分享 收藏 分享 收藏 Histamine H3 Receptor Ligands-KSK-59 and KSK-73-Reduce Body Weight Gain in a Rat Model of Excessive EatingMika, Kamil; Szafarz, Malgorzata; Bednarski, Marek; Latacz, Gniewomir; Sudol, Sylwia; Handzlik, Jadwiga; Pociecha, Krzysztof; Knutelska, Joanna; Nicosia, Noemi; Szczepanska, Katarzyna; Kuder, Kamil J.; Kiec-Kononowicz, Katarzyna; Kotanska, Magdalena 分享 收藏 Metabolic benefits of novel histamine H3 receptor ligands in the model of excessive eating: The importance of intrinsic activity and pharmacokinetic propertiesMika, Kamil; Szafarz, Malgorzata; Bednarski, Marek; Kuder, Kamil; Szczepanska, Katarzyna; Pociecha, Krzysztof; Pomierny, Bartosz; Kiec-Kononwicz, Katarzyna; Sapa, Jacek; Kotanska, Magdalena 分享 收藏 
.png){kind=icon}
.png){kind=icon}
.png){kind=icon}
.png){kind=icon}
