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Simon J. Cook

University of Dundee

60H指数
243论文数
1.3W被引数
收录论文 102
发表时间
RAF inhibitors activate the integrated stress response by direct activation of GCN2RAF抑制剂通过直接激活GCN2来激活整合应激反应
err2025-11-17
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errRebecca Gilley; Andrew M. Kidger; Graham Neill; Eve Morrison; Paul Severson; Dominic P. Byrne; Niall S. Kenneth; Gideon Bollag; Chao Zhang; Taiana Maia de Oliveira; Patrick A. Eyers; Richard Bayliss; Glenn R. Masson; Simon J. Cook
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Hypoxia drives HIF2-dependent reversible macrophage cell cycle entry
err2024-07-01
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errMeng, Bo; Zhao, Na; Mlcochova, Petra; Ferreira, Isabella A. T. M.; Ortmann, Brian M.; Davis, Tanja; Wit, Niek; Rehwinkel, Jan; Cook, Simon; Maxwell, Patrick H.; Nathan, James A.; Gupta, Ravindra K.
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EU-LIFE charter of independent life science research institutes欧盟-独立生命科学研究机构的生命宪章
err2024-03-21
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errSuperti-Furga, Giulio; Agostinho, Marta; Bury, Jo; Cook, Simon; Durinx, Christine; Ender, Anita; van Luenen, Henri; Lund, Anders H.; Medema, Rene H.; Miaczynska, Marta; Nickel, Dorthe; Pelicci, Pier Giuseppe; Puisieux, Alain; Ripatti, Samuli; Sander, Maike; Schubeler, Dirk; Serrano, Luis; Sommer, Thomas; Sonne-Hansen, Katrine; Tomancak, Pavel; Vives, Joan; Vontas, John; Bettencourt-Dias, Monica
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Reporter cell lines to screen for inhibitors or regulators of the KRAS-RAF-MEK1/2-ERK1/2 pathway
err2024-03-07
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errWeatherdon, Laura; Stuart, Kate; Cassidy, Megan; de la Gandara, Alberto Moreno; Okkenhaug, Hanneke; Muellener, Markus; Mckenzie, Grahame; Cook, Simon J.; Gilley, Rebecca
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ERK1/2 inhibitors act as monovalent degraders inducing ubiquitylation and proteasome-dependent turnover of ERK2, but not ERK1
err2023-05-04
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errBalmanno, Kathryn; Kidger, Andrew M.; Byrne, Dominic P.; Sale, Matthew J.; Nassman, Nejma; Eyers, Patrick A.; Cook, Simon J.
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Escape from G1 arrest during acute MEK inhibition drives the acquisition of drug resistance
err2022-10-17
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errChannathodiyil, Prasanna; May, Kieron; Segonds-Pichon, Anne; Smith, Paul D.; Cook, Simon J.; Houseley, Jonathan
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Parallel Optimization of Potency and Pharmacokinetics Leading to the Discovery of a Pyrrole Carboxamide ERK5 Kinase Domain Inhibitor
err2022-04-25
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errMiller, Duncan C.; Reuillon, Tristan; Molyneux, Lauren; Blackburn, Timothy; Cook, Simon J.; Edwards, Noel; Endicott, Jane A.; Golding, Bernard T.; Griffin, Roger J.; Hardcastle, Ian; Harnor, Suzannah J.; Heptinstall, Amy; Lochhead, Pamela; Martin, Mathew P.; Martin, Nick C.; Myers, Stephanie; Newell, David R.; Noble, Richard A.; Phillips, Nicole; Rigoreau, Laurent; Thomas, Huw; Tucker, Julie A.; Wang, Lan-Zhen; Waring, Michael J.; Wong, Ai-Ching; Wedge, Stephen R.; Noble, Martin E. M.; Cano, Celine
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Environmental Sustainability and Supply Resilience of Cobalt
err2022-03-30
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errEarl, Cathryn; Shah, Izhar Hussain; Cook, Simon; Cheeseman, Christopher Robert
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IKKα plays a major role in canonical NF-KB signalling in colorectal cells
err2022-02-04
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errPrescott, Jack A.; Balmanno, Kathryn; Mitchell, Jennifer P.; Okkenhaug, Hanneke; Cook, Simon J.
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Inhibitory feedback control of NF-KB signalling in health and disease
err2021-07-16
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errPrescott, Jack A.; Mitchell, Jennifer P.; Cook, Simon J.
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CDK1, the Other 'Master Regulator' of Autophagy
err2021-02-01
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errOdle, Richard, I; Florey, Oliver; Ktistakis, Nicholas T.; Cook, Simon J.
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Paradoxical activation of the protein kinase-transcription factor ERK5 by ERK5 kinase inhibitors
err2020-03-13
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errLochhead, Pamela A.; Tucker, Julie A.; Tatum, Natalie J.; Wang, Jinhua; Oxley, David; Kidger, Andrew M.; Johnson, Victoria P.; Cassidy, Megan A.; Gray, Nathanael S.; Noble, Martin E. M.; Cook, Simon J.
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Macroautophagy is repressed during mitosis - seeing is believing
errAUTOPHAGY
IF14.3
err2020-02-20
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errOdle, Richard I.; Cook, Simon J.
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Dual-Mechanism ERK1/2 Inhibitors Exploit a Distinct Binding Mode to Block Phosphorylation and Nuclear Accumulation of ERK1/2
err2020-02-06
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errKidger, Andrew M.; Munck, Joanne M.; Saini, Harpreet K.; Balmanno, Kathryn; Minihane, Emma; Courtin, Aurelie; Graham, Brent; O'Reilly, Marc; Odle, Richard; Cook, Simon J.
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An mTORC1-to-CDK1 Switch Maintains Autophagy Suppression during Mitosis有丝分裂过程中mTORC1-to-CDK1开关维持自噬抑制
err2020-01-01
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errOdle, Richard I.; Walker, Simon A.; Oxley, David; Kidger, Andrew M.; Balmanno, Kathryn; Gilley, Rebecca; Okkenhaug, Hanneke; Florey, Oliver; Ktistakis, Nicholas T.; Cook, Simon J.
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Targeting melanoma's MCL1 bias unleashes the apoptotic potential of BRAF and ERK1/2 pathway inhibitors
err2019-11-14
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errSale, Matthew J.; Minihane, Emma; Monks, Noel R.; Gilley, Rebecca; Richards, Frances M.; Schifferli, Kevin P.; Andersen, Courtney L.; Davies, Emma J.; Vicente, Mario Aladren; Ozono, Eiko; Markovets, Aleksandra; Dry, Jonathan R.; Drew, Lisa; Flemington, Vikki; Proia, Theresa; Jodrell, Duncan I.; Smith, Paul D.; Cook, Simon J.
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