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Michael J. Stocks

University of Nottingham

28H指数
126论文数
2.3K被引数
收录论文 51
发表时间
Discovery of uracil-based antagonists and fluorescent ligands of the P2Y2 receptor尿嘧啶基拮抗剂和P2Y2受体荧光配体的发现
err2026-08-01
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PREAI
errPuthanveedu, Mahesh; Dale, Natasha; Knight, Rebecca; Comeo, Eleonora; Kindon, Nicholas D.; Kellam, Barrie; Kilpatrick, Laura E.; Hill, Stephen J.; Stocks, Michael J.
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Discovery of a Potent Lysine-Specific Histone Demethylase-1 (LSD-1) Inhibitor for Cancer Treatment via Machine Learning, Molecular Modeling, and In Vitro Validation通过机器学习、分子建模和体外验证发现一种用于癌症治疗的强效赖氨酸特异性组蛋白去甲基化酶-1(LSD-1)抑制剂
err2025-10-28
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PREAI
errShuya Wang; Lihui Duo; Zhangyi Ma; Zixuan Zhang; Dr. Biyu Hu; Dr. Hainam Do; Binjie Hu; Prof. Michael J. Stocks; Prof. Jianfeng Ren; Dr. Bruno N. Falcone; Prof. Jonathan D. Hirst; Prof. Guang Yang; Prof. Bencan Tang
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Sebetralstat (KVD900): A Potent and Selective Small Molecule Plasma Kallikrein Inhibitor Featuring a Novel P1 Group as a Potential Oral On-Demand Treatment for Hereditary Angioedema ( vol 6565 , pg 13629 , 2022)
err2025-10-01
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PREAI
errDavie, Rebecca L.; Edwards, Hannah J.; Evans, D. Michael; Hodgson, Simon T.; Stocks, Michael J.; Smith, Alun J.; Rushbrooke, Louise J.; Pethen, Stephen J.; Roe, Michael B.; Clark, David E.; Mcewan, Paul A.; Hampton, Sally L.
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Discovery of Highly Potent BET Inhibitors based on a Tractable Tricyclic Scaffold
err2025-03-01
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errOAAI
errZaidi, Jaffer M.; Comeo, Eleonora; Baxter, Andrew; Preston, Alex G. S.; Chan, Weng C.; Stocks, Michael J.
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Rapeseed oleosomes facilitate intestinal lymphatic delivery and oral bioavailability of cannabidiol油菜籽油质体促进肠淋巴递送和大麻二酚的口服生物利用度
err2025-01-01
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errOAAI
errJi, Liuhang; Feng, Wanshan; Chen, Haojie; Chu, Yenju; Wong, Abigail; Zhu, Yufei; Sinatra, Graziamarina; Bramante, Filippo; Carriere, Frederic; Stocks, Michael J.; di Bari, Vincenzo; Gray, David A.; Gershkovich, Pavel
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Delivery of imiquimod to intestinal lymph nodes following oral administration
err2024-12-01
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errOAAI
errChen, Haojie; Ji, Liuhang; Wong, Abigail; Chu, Yenju; Feng, Wanshan; Zhu, Yufei; Wang, Junting; Comeo, Eleonora; Kim, Dong-Hyun; Stocks, Michael J.; Gershkovich, Pavel
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Theoretical Study on the Biosynthesis of the Mandapamates: Mechanistic Insights Using Density Functional Theory
err2024-09-09
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errOAAI
errWang, Di; Pattenden, Gerald; Fow, Kam Loon; Stocks, Michael J.; Hirst, Jonathan D.; Tang, Bencan
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Design, Synthesis, and Evaluation of a New Chemotype Fluorescent Ligand for the P2Y2 Receptor
err2024-06-12
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errOAAI
errKnight, Rebecca; Kilpatrick, Laura E.; Hill, Stephen J.; Stocks, Michael J.
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Discovery of α-Amidobenzylboronates as Highly Potent Covalent Inhibitors of Plasma Kallikrein
err2024-03-28
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errOAAI
errAllison, Matthew; Davie, Rebecca L.; Mogg, Adrian J.; Hampton, Sally L.; Emsley, Jonas; Stocks, Michael J.
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CXCL17 is an allosteric inhibitor of CXCR4 through a mechanism of action involving glycosaminoglycans
err2024-03-19
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errOAAI
errWhite, Carl W.; Platt, Simon; Kilpatrick, Laura E.; Dale, Natasha; Abhayawardana, Rekhati S.; Dekkers, Sebastian; Kindon, Nicholas D.; Kellam, Barrie; Stocks, Michael J.; Pfleger, Kevin D. G.; Hill, Stephen J.
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Design, Synthesis, and Evaluation of New 1H-Benzo[d]imidazole Based PqsR Inhibitors as Adjuvant Therapy for Pseudomonas aeruginosa Infections
err2024-01-03
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errOAAI
errSoukarieh, Fadi; Mashabi, Alaa; Richardson, William; Oton, Eduard Vico; Romero, Manuel; Dubern, Jean-Frederic; Robertson, Shaun N.; Lucanto, Simone; Markham-Lee, Zoe; Sou, Tomas; Kukavica-Ibrulj, Irena; Levesque, Roger C.; Bergstrom, Christel A. S.; Halliday, Nigel; Kellam, Barrie; Emsley, Jonas; Heeb, Stephan; Williams, Paul; Stocks, Michael J.; Camara, Miguel
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Small Molecule Fluorescent Ligands for the Atypical Chemokine Receptor 3 (ACKR3)
err2023-12-08
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errOAAI
errDekkers, Sebastian; Comez, Dehan; Karsai, Noemi; Arimont-Segura, Marta; Canals, Meritxell; Caspar, Birgit; de Graaf, Chris; Kilpatrick, Laura E.; Leurs, Rob; Kellam, Barrie; Hill, Stephen J.; Briddon, Stephen J.; Stocks, Michael J.
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Distribution of lamivudine into lymph node HIV reservoir
err2023-12-01
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errOAAI
errWong, Abigail; Chu, Yenju; Chen, Haojie; Feng, Wanshan; Ji, Liuhang; Qin, Chaolong; Stocks, Michael J.; Marlow, Maria; Gershkovich, Pavel
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Small-Molecule Fluorescent Ligands for the CXCR4 Chemokine Receptor
err2023-03-21
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errOAAI
errDekkers, Sebastian; Caspar, Birgit; Goulding, Joelle; Kindon, Nicholas D.; Kilpatrick, Laura E.; Stoddart, Leigh A.; Briddon, Stephen J.; Kellam, Barrie; Hill, Stephen J.; Stocks, Michael J.
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Sebetralstat (KVD900): A Potent and Selective Small Molecule Plasma Kallikrein Inhibitor Featuring a Novel P1 Group as a Potential Oral On-Demand Treatment for Hereditary Angioedema
err2022-10-17
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errOAAI
errDavie, Rebecca L.; Edwards, Hannah J.; Evans, D. Michael; Hodgson, Simon T.; Stocks, Michael J.; Smith, Alun J.; Rushbrooke, Louise J.; Pethen, Stephen J.; Roe, Michael B.; Clark, David E.; McEwan, Paul A.; Hampton, Sally L.
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Vegetable oils composition affects the intestinal lymphatic transport and systemic bioavailability of co-administered lipophilic drug cannabidiol
err2022-08-01
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errOAAI
errFeng, Wanshan; Qin, Chaolong; Abdelrazig, Salah; Bai, Ziyu; Raji, Mekha; Darwish, Randa; Chu, YenJu; Ji, Liuhang; Gray, David A.; Stocks, Michael J.; Constantinescu, Cris S.; Barrett, David A.; Fischer, Peter M.; Gershkovich, Pavel
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Design, Synthesis, and Evaluation of Lung-Retentive Prodrugs for Extending the Lung Tissue Retention of Inhaled Drugs
err2022-07-07
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errAyre, Jack; Redmond, Joanna M.; Vitulli, Giovanni; Tomlinson, Laura; Weaver, Richard; Comeo, Eleonora; Bosquillon, Cynthia; Stocks, Michael J.
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