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Yong Chen

tianjin medical center for medical device evaluation and inspection

18H指数
94论文数
955被引数
收录论文 44
发表时间
Supramolecular Degraders: An Emerging Paradigm in Targeted Protein Degradation超分子降解剂:靶向蛋白质降解中的新兴范式
err2026-09-14
err0
errOAAI
errKongjun Liu; Xue Yuan; Yan Zhou; Rui Yuan; Shaocheng Xie; Yong Chen; Peiyi Wang; Jianmei Gao; Qihai Gong
err分享
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Rational Design and Optimization of Highly Selective CSF1R Inhibitors for the Treatment of Acute Liver Injury急性肝损伤治疗中高选择性CSF1R抑制剂的理性设计与优化
err2026-04-23
err0
PREAI
errXue Yuan; Kongjun Liu; Yurong Zou; Yuhan Wei; Qianhuan Liu; Guoli Zheng; Miao Ru; Yuandong Zhang; Baojian Xiong; Jianmei Gao; Yong Chen; Qihai Gong
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CMD-OPT model enables the discovery of a potent and selective RIPK2 inhibitor as preclinical candidate for the treatment of acute liver injuryCMD-OPT模型能够发现一种强效且选择性的RIPK2抑制剂,作为治疗急性肝损伤的预临床试验候选药物。
err2025-05-13
err0
errOAAI
errYong Chen; Xue Yuan; Wei Yan; Yurong Zou; Haoche Wei; Yuhan Wei; Minghai Tang; Yulian Chen; Ziyan Ma; Tao Yang; Kongjun Liu; Baojian Xiong; Xiuying Hu; Jianhong Yang; Lijuan Chen
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Latent profile and determinants of self-management behaviors among older adult patients with chronic diseases: a cross-sectional study老年慢性病患者自我管理行为的潜在特征和决定因素: 一项横断面研究
err2025-02-05
err0
errOAAI
errShao, Yu Jiao; Duan, Xiao Cui; Xu, Xue Jun; Guo, Hong Yan; Zhang, Ze Yu; Zhao, Shuang; Wang, Fu Zhi; Chen, Yong Xia; Chen, Qin; Zhang, Shi Qing; Yang, Xiu Mu
err分享
err收藏
Water-soluble and predictable-release triptolide prodrugs block bleomycin-induced pulmonary fibrosis in mice
err2024-12-01
err0
PREAI
errChen, Yuhan; Liang, Meiyu; Li, Wen; Yang, Zhiming; Yan, Xingting; Wu, Liuying; Yu, Qin; Chen, Yubai; Chen, Yong; Xu, Yan; Song, Wei; Peng, Zhihong
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Discovery of Potent, Specific, and Orally Available NLRP3 Inflammasome Inhibitors Based on Pyridazine Scaffolds for the Treatment of Septic Shock and Peritonitis
err2024-08-22
err2
PREAI
errFu, Zhiyuan; Duan, Yangqin; Pei, Heying; Zou, Yurong; Tang, Minghai; Chen, Yong; Yang, Tao; Ma, Ziyan; Yan, Wei; Su, Kaiyue; Cai, Xiaoying; Guo, Tao; Teng, Yaxin; Jia, Tao; Chen, Lijuan
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Design, Synthesis, and Biological Evaluation of 5-Amino-4-fluoro-1H-benzo[d]imidazole-6-carboxamide Derivatives as Novel and Potential MEK/RAF Complex Inhibitors Based on the Clamp Strategy
err2024-08-21
err0
PREAI
errWang, Peng; Yuan, Yongting; Yang, Tao; Zou, Yurong; Tang, Minghai; Ma, Ziyan; Bo, Weichen; Qin, Songhui; Chen, Yong; Guo, Tao; Guo, Zhongning; Yang, Jianhong; Xiang, Mingli; Chen, Lijuan
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Discovery, Optimization, and Evaluation of Potent and Selective DNA-PK Inhibitors in Combination with Chemotherapy or Radiotherapy for the Treatment of Malignancies
err2023-12-20
err3
PREAI
errLiu, Kongjun; Yuan, Xue; Yang, Tao; Deng, Dexin; Chen, Yong; Tang, Minghai; Zhang, Chufeng; Zou, Yurong; Zhang, Shunjie; Li, Dan; Shi, Mingsong; Guo, Yong; Zhou, Yanting; Zhao, Min; Yang, Zhuang; Chen, Lijuan
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Discovery of Potent and Selective Phosphatidylinositol 3-Phosphate 5-Kinase (PIKfyve) Inhibitors as Methuosis Inducers
err2023-12-20
err4
PREAI
errChen, Yong; Liu, Shuai; Wei, Yuhan; Wei, Haoche; Yuan, Xue; Xiong, Baojian; Tang, Minghai; Yang, Tao; Yang, Zhuang; Ye, Haoyu; Yang, Jianhong; Chen, Lijuan
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Discovery and Evaluation of 3-Quinoxalin Urea Derivatives as Potent, Selective, and Orally Available ATM Inhibitors Combined with Chemotherapy for the Treatment of Cancer via Goal-Oriented Molecule Generation and Virtual Screening
err2023-07-13
err9
PREAI
errDeng, Dexin; Yang, Yingxue; Zou, Yurong; Liu, Kongjun; Zhang, Chufeng; Tang, Minghai; Yang, Tao; Chen, Yong; Yuan, Xue; Guo, Yong; Zhang, Shunjie; Si, Wenting; Peng, Bin; Xu, Qing; He, Wen; Xu, Dingguo; Xiang, Mingli; Chen, Lijuan
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Rational design and appraisal of selective Cdc2-Like kinase 1 (Clk1) inhibitors as novel autophagy inducers for the treatment of acute liver injury (ALI)
err2023-03-01
err0
PREAI
errYang, Tao; Yang, Yingxue; Chen, Yong; Tang, Minghai; Shi, Mingsong; Tian, Yang; Yuan, Xue; Yang, Zhuang; Chen, Lijuan
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MagicGAN: Multiagent Attacks Generate Interferential Category via GAN
err2022-12-01
err2
PREAI
errChen, Yong; Wang, Xu; Hu, Peng; Peng, Dezhong
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Design, synthesis, and pharmacological evaluation of 2-(1-(1,3,4-thiadiazol-2-yl)piperidin-4-yl)ethan-1-ol analogs as novel glutaminase 1 inhibitors
err2022-12-01
err5
PREAI
errYang, Tao; Tian, Yang; Yang, Yingxue; Tang, Minghai; Shi, Mingsong; Chen, Yong; Yang, Zhuang; Chen, Lijuan
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Discovery, Optimization, and Evaluation of Potent and Selective PI3Kδ-γ Dual Inhibitors for the Treatment of B-cell Malignancies
err2022-07-13
err2
PREAI
errLiu, Kongjun; Zheng, Wei; Chen, Yong; Tang, Minghai; Li, Dan; Deng, Dexin; Yang, Tao; Zhang, Chufeng; Liu, Jiang; Yuan, Xue; Shi, Mingsong; Li, Xiandeng; Guo, Yong; Zhou, Yanting; Zhao, Min; Chen, Lijuan
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Discovery of Potent and Selective Receptor-Interacting Serine/ Threonine Protein Kinase 2 (RIPK2) Inhibitors for the Treatment of Inflammatory Bowel Diseases (IBDs)
err2022-06-16
err13
PREAI
errYuan, Xue; Chen, Yong; Tang, Minghai; Wei, Yuhan; Shi, Mingsong; Yang, Yingxue; Zhou, Yanting; Yang, Tao; Liu, Jiang; Liu, Kongjun; Deng, Dexin; Zhang, Chufeng; Chen, Lijuan
err分享
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