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收藏Lead optimization of 2-hydroxymethyl imidazoles as non-hydroxamate LpxC inhibitors: Discovery of TP0586532
Ushiyama, Fumihito; Takashima, Hajime; Matsuda, Yohei; Ogata, Yuya; Sasamoto, Naoki; Kurimoto-Tsuruta, Risa; Ueki, Kaori; Tanaka-Yamamoto, Nozomi; Endo, Mayumi; Mima, Masashi; Fujita, Kiyoko; Takata, Iichiro; Tsuji, Satoshi; Yamashita, Haruhiro; Okumura, Hirotoshi; Otake, Katsumasa; Sugiyama, Hiroyuki
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收藏Fragment-Based Discovery of Novel Non-Hydroxamate LpxC Inhibitors with Antibacterial Activity
Yamada, Yousuke; Takashima, Hajime; Walmsley, David Lee; Ushiyama, Fumihito; Matsuda, Yohei; Kanazawa, Harumi; Yamaguchi-Sasaki, Toru; Tanaka-Yamamoto, Nozomi; Yamagishi, Junya; Kurimoto-Tsuruta, Risa; Ogata, Yuya; Ohtake, Norikazu; Angove, Hayley; Baker, Lisa; Harris, Richard; Macias, Alba; Robertson, Alan; Surgenor, Allan; Watanabe, Hayato; Nakano, Koichiro; Mima, Masashi; Iwamoto, Kunihiko; Okada, Atsushi; Takata, Iichiro; Hitaka, Kosuke; Tanaka, Akihiro; Fujita, Kiyoko; Sugiyama, Hiroyuki; Hubbard, Roderick E.
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收藏Ursolic acid, an antagonist for transforming growth factor (TGF)-β1
Murakami, S; Takashima, H; Sato-Watanabe, M; Chonan, S; Yamamoto, K; Saitoh, M; Saito, S; Yoshimura, H; Sugawara, K; Yang, JS; Gao, NN; Zhang, XG
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收藏Development of MOE (molecular orbital calculation engine)
Nagashima, U; Obara, S; Murakami, K; Yoshii, T; Shirakawa, S; Amisaki, T; Kitamura, K; Takashima, H; Kitao, O; Tanabe, K
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