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ADT-1004: a first-in-class, oral pan-RAS inhibitor with robust antitumor activity in preclinical models of pancreatic ductal adenocarcinoma ADT-1004: 在胰腺导管腺癌的临床前模型中具有强大抗肿瘤活性的一流口服pan-ras抑制剂 Bandi, Dhana Sekhar Reddy; Nagaraju, Ganji Purnachandra; Sarvesh, Sujith; Carstens, Julienne L.; Foote, Jeremy B.; Graff, Emily C.; Fang, Yu-Hua D.; Keeton, Adam B.; Chen, Xi; Valiyaveettil, Jacob; Berry, Kristy L.; Bae, Sejong; Akce, Mehmet; Gorman, Greg; Yoon, Karina J.; Manne, Upender; Boyd, Michael R.; Buchsbaum, Donald J.; Azmi, Asfar S.; Maxuitenko, Yulia Y.; Piazza, Gary A. 分享 收藏
Combined Use of Ziftomenib and Selinexor Is Effective in NPM1 Mutant Acute Myeloid Leukemia Ziftomenib与Selinexor的联合使用对NPM1突变急性髓系白血病有效 Dhiman, Sandhya; Uddin, Md. Hafiz; Dhillon, Vikram; Aguilar, Jeff Justin; Aboukameel, Amro; Khan, Husain; Bannoura, Sahar; Yang, Jay; Dyson, Gregory; Buck, Steven; Azmi, Asfar; Polin, Lisa; Burrows, Francis; Kessler, Linda; Maciejewski, Jaroslaw; Balasubramanian, Suresh Kumar 分享 收藏
RCC1 regulation of subcellular protein localization via Ran GTPase drives pancreatic ductal adenocarcinoma growth Bannoura, Sahar F.; Aboukameel, Amro; Khan, Husain Yar; Uddin, Md Hafiz; Jang, Hyejeong; Beal, Eliza W.; Thangasamy, Amalraj; Shi, Yang; Kim, Seongho; Wagner, Kay-Uwe; Beydoun, Rafic; El-Rayes, Bassel F.; Philip, Philip A.; Mohammad, Ramzi M.; Saif, Muhammad Wasif; Al-Hallak, Mohammed Najeeb; Pasche, Boris C.; Azmi, Asfar S. 分享 收藏
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Nuclear exporter protein exportin 1 (XPO1) as a novel therapeutic target in pancreatic neuroendocrine tumors Azmi, A. S.; Uddin, M. H.; Bannoura, S. F.; Khan, H. M.; Diab, M.; Kim, S.; Beal, E.; Tobon, M.; Chen, H.; Beydoun, R.; Dyson, G.; Mohammad, R. M.; Philip, P. A.; Al-Hallak, M. N.; El-Rayes, B. F.; Pasche, B. 分享 收藏
A phase I study of CPI-613 (devimistat) in combination with chemoradiation in patients with pancreatic ductal adenocarcinoma Kamgar, Mandana; Khan, Husain Yar; Aboukameel, Amro; Bannoura, Sahar F.; Chung, Brian Y.; Szabo, Aniko; Li, Yiwei; Al Hallak, Mohammed Najeeb; Philip, Philip A.; George, Ben; Christians, Kathleen K.; Evans, Douglas B.; Tsai, Susan; Erickson, Beth; Goldberg, John M.; Azmi, Asfar S.; Hall, William A. 分享 收藏
Next generation nuclear export blocker KPT8602 synergizes with KRASG12D inhibitor MRTX1133 resulting in improved antitumor effects against pancreatic ductal adenocarcinoma Khan, Husain Yar; Aboukameel, Amro; Uddin, Md Hafiz; Bannoura, Sahar F.; Keffri, Khaled; Jasti, Medha; Virga, Rachael; Motorwala, Sarah; Choucair, Khalil; Hadid, Tarik; Al-Hallak, Mohammad Najeeb; Beal, Eliza; Tobon, Miguel; Beydoun, Rafic; Dyson, Greg; Kim, Steve; Nagasaka, Misako; Philip, A. Philip; El-Rayes, Basel; Chen, Herbert; Shields, Anthony; Mohammad, Ramzi; Pasche, Boris; Azmi, Asfar 分享 收藏
NT219, a dual inhibitor of IRS1/2 and STAT3, suppresses cancer stem cell mediated resistance to KRASG12C and KRASG12D inhibitors in solid tumors Reuveni, Hadas; Al-Hallak, Mohammed Najeeb; Motorwala, Sarah; Beal, Eliza; Kim, Steve; Beydoun, Rafic; Dyson, Gergory; El-Rayes, Bassel; Chen, Herbert; Philip, A. Philip; Shields, Anthony F.; Pasche, Boris; Sigalov, Katy; Ben-David, Hava; Miron, Daphna; Azmi, Asfar S. 分享 收藏
Regulator of chromosome condensation 1 (RCC1) as a novel therapeutic target in pancreatic ductal adenocarcinoma Bannoura, Sahar F.; Khan, Husain Y.; Aboukameel, Amro; Uddin, Md Hafiz; Nimri, Rund; Beal, Eliza; Kim, Seongho; Al Hallak, Mohammed Najeeb; El-Rayes, Bassel; Philip, Philip A.; Pasche, Boris; Mohammad, Ramzi; Azmi, Asfar S. 分享 收藏
Nuclear export inhibitor cooperates with PARP inhibitor to suppress the growth of metastatic castration resistant prostate cancer in vivo Uddin, Md Hafiz; Aboukameel, Amro; Khan, Husain Y.; Bannoura, Sahar F.; Cackowski, Frank; Beydoun, Rafic; Dyson, Gregory; Kim, Seongho; Boerner, Julie; Shidham, Vinod; Mohammad, Ramzi M.; Pasche, Boris C.; Azmi, Asfar S.; Heath, Elisabeth I. 分享 收藏
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KRASG12D inhibitor MRTX1133 synergizes with the next generation nuclear transport protein inhibitor eltanexor resulting in enhanced antitumor activity against pancreatic ductal adenocarcinoma KRASG12D抑制剂MRTX1133与下一代核转运蛋白抑制剂eltanexor协同作用,增强对胰腺导管腺癌的抗肿瘤活性 Khan, Husain Y.; Aboukameel, Amro; Uddin, Md Hafiz; Al-Hallak, Mohammad Najeeb; Beal, Eliza W.; Azar, Ibrahim; Baloglu, Erkan; Beydoun, Rafic; Sukari, Ammar; Nagasaka, Misako; Mohamed, Amr; Kaseb, Ahmed; Philip, A. Philip; El-Rayes, Basel; Chen, Herbert; Shields, Anthony; Azmi, Asfar 分享 收藏
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Molecular analysis of XPO1 inhibitor and gemcitabine-nab-paclitaxel combination in KPC pancreatic cancer mouse model XPO1抑制剂和吉西他滨-nab-紫杉醇联合应用在KPC胰腺癌小鼠模型中的分子分析 Uddin, Md. Hafiz; Al-Hallak, Mohammad Najeeb; Khan, Husain Yar; Aboukameel, Amro; Li, Yiwei; Bannoura, Sahar F.; Dyson, Gregory; Kim, Seongho; Mzannar, Yosef; Azar, Ibrahim; Odisho, Tanya; Mohamed, Amr; Landesman, Yosef; Kim, Steve; Beydoun, Rafic; Mohammad, Ramzi M.; Philip, Philip A.; Shields, Anthony F.; Azmi, Asfar S. 分享 收藏