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收藏Analysis of genotypic distribution and rare variants of patients with α/β-thalassemia screened in one hospital in Beijing, China
Zhang, Han; Wang, Ziran; Yang, Zhuo; Chen, Xinfei; Xu, Hongrui; Zeng, Xianhui; Yu, Qi; Kong, Lingjun; Zhang, Rui; Yi, Jie; Wu, Jie; Gan, Yong; Chen, Yu; Ye, Ali; Wang, Ziyi; Zhang, Dong; Han, Xiao; Du, Juan; Dou, Yaling
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收藏Discovery of a Potent and Selective GSPT1 Molecular Glue Degrader for the Treatment of Castration-Resistant Prostate Cancer发现一种用于治疗去势抵抗性前列腺癌的高效且特异性的GSPT1分子胶降解剂
Shen, Hui; Xu, Hongrui; Jin, Weiqin; Wu, Tianbang; Hu, Jiankang; Zhang, Cheng; Zhong, Zhixin; Li, Junhua; Mao, Rui; Zhang, Sheng; Zhang, Xiao; Wu, Xishan; Smaill, Jeff B.; Xu, Jinxin; Zhang, Yan
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收藏Fluorescent microsphere-based strip for sensitive and quantitative detection of 3-quinuclidinyl benzilate and clidinium bromide in biological samples基于荧光微球的试纸条,用于生物样品中对3-奎宁环基苯甲酸酯和氯化氯二甲哌的敏感定量检测
Guo, Jing; Liu, Yulong; Xue, Jinjuan; Jiang, Jinqiao; Fan, Jiyong; Xu, Hongrui; Yu, Tao; Xu, Na; Xu, Zhanlin; Wu, Jianfeng; Xie, Jianwei
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收藏Efficient Chemical Synthesis of Multi-Monoubiquitylated and Diubiquitylated Histones by the α-Halogen Ketone-Mediated Strategy
Peng, Shuai; Liu, Xin; Lu, Chengpiao; Wang, Haibo; Liu, Xiaotong; Gong, Qingyue; Tao, Huizhong; Xu, Hongrui; Tian, Changlin; Xu, Guoqiang; Li, Jia-Bin
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收藏Discovery of a Promising CBP/p300 Degrader XYD129 for the Treatment of Acute Myeloid Leukemia
Wu, Tianbang; Hu, Jiankang; Zhao, Xiaofan; Zhang, Cheng; Dong, Ruibo; Hu, Qingqing; Xu, Hongrui; Shen, Hui; Zhang, Xiaohan; Zhang, Yan; Lin, Bin; Wu, Xishan; Xiang, Qiuping; Xu, Yong
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收藏Discovery of Highly Potent and Efficient CBP/p300 Degraders with Strong In Vivo Antitumor Activity
Hu, Jiankang; Xu, Hongrui; Wu, Tianbang; Zhang, Cheng; Shen, Hui; Dong, Ruibo; Hu, Qingqing; Xiang, Qiuping; Chai, Shuang; Luo, Guolong; Chen, Xiaoshan; Huang, Yumin; Zhao, Xiaofan; Peng, Chao; Wu, Xishan; Lin, Bin; Zhang, Yan; Xu, Yong
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收藏Discovery of Novel Phenoxyaryl Pyridones as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with High Selectivity for the Second Bromodomain (BD2) to Potentially Treat Acute Myeloid Leukemia
Jiang, Wenhua; Hou, Qiangqiang; Xu, Hongrui; Yang, Kexin; Wang, Xiaohui; Zhang, Kuojun; Zeng, Yi; Li, Wenqiang; Wang, Bingrui; Luo, Guangmei; Zhao, Xiaofan; Shen, Hui; Xu, Yong; Wu, Xiaoxing
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收藏Discovery of (R)-4-(8-methoxy-2-methyl-1-(1-phenylethy)-1H-imidazo [4,5-c]quinnolin-7-yl)-3,5-dimethylisoxazole as a potent and selective BET inhibitor for treatment of acute myeloid leukemia (AML) guided by FEP calculation
Yu, Su; Zhang, Yan; Yang, Jie; Xu, Hongrui; Lan, Suke; Zhao, Binyan; Luo, Meng; Ma, Xinyu; Zhang, Hongjia; Wang, Shirui; Shen, Hui; Xu, Yong; Li, Rui
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收藏Discovery, optimization and evaluation of 1-(indolin-1-yl)ethan-1-ones as novel selective TRIM24/BRPF1 bromodomain inhibitors
Xiang, Qiuping; Luo, Guolong; Zhang, Cheng; Hu, Qingqing; Wang, Chao; Wu, Tianbang; Xu, Hongrui; Hu, Jiankang; Zhuang, Xiaoxi; Zhang, Maofeng; Wu, Shuang; Xu, Jinxin; Zhang, Yan; Liu, Jinsong; Xu, Yong
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收藏Structure-Based Discovery and Optimization of Furo[3,2-c]pyridin-4(5H)-one Derivatives as Potent and Second Bromodomain (BD2)-Selective Bromo and Extra Terminal Domain (BET) Inhibitors
Li, Junhua; Zhang, Cheng; Xu, Hongrui; Wang, Chao; Dong, Ruibo; Shen, Hui; Zhuang, Xiaoxi; Chen, Xiaoshan; Li, Qiu; Lu, Jibu; Zhang, Maofeng; Wu, Xishan; Loomes, Kerry M.; Zhou, Yulai; Zhang, Yan; Liu, Jinsong; Xu, Yong
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