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A small molecule exerts selective antiviral activity by targeting the human cytomegalovirus nuclear egress complex Chen, Han; Lye, Ming F.; Gorgulla, Christoph; Ficarro, Scott B.; Cuny, Gregory D.; Scott, David A.; Wu, Fan; Rothlauf, Paul W.; Wang, Xiaoou; Fernandez, Rosio; Pesola, Jean M.; Draga, Sorin; Marto, Jarrod A.; Hogle, James M.; Arthanari, Haribabu; Coen, Donald M. 分享 收藏
An Immunconjugate Vaccine Alters Distribution and Reduces the Antinociceptive, Behavioral and Physiological Effects of Fentanyl in Male and Female Rats Haile, Colin N.; Baker, Miah D.; Sanchez, Sergio A.; Arteaga, Carlos A. Lopez; Duddupudi, Anantha L.; Cuny, Gregory D.; Norton, Elizabeth B.; Kosten, Thomas R.; Kosten, Therese A. 分享 收藏
A D-Phenylalanine-Benzoxazole Derivative Reveals the Role of the Essential Enzyme Rv3603c in the Pantothenate Biosynthetic Pathway of Mycobacterium tuberculosis Pepi, Michael J.; Chacko, Shibin; Marqus, Gary M.; Singh, Vinayak; Wang, Zhe; Planck, Kyle; Cullinane, Ryan T.; Meka, Penchala N.; Gollapalli, Deviprasad R.; Ioerger, Thomas R.; Rhee, Kyu Y.; Cuny, Gregory D.; Boshoff, Helena I. M.; Hedstrom, Lizbeth 分享 收藏
Expanding Benzoxazole-Based Inosine 5′-Monophosphate Dehydrogenase (IMPDH) Inhibitor Structure-Activity As Potential Antituberculosis Agents (vol 61, pg 4739, 2018) Chacko, Shibin; Boshoff, Helena I. M.; Singh, Vinayak; Ferraris, Davide M.; Gollapalli, Deviprasad R.; Zhang, Minjia; Lawson, Ana P.; Pepi, Michael J.; Joachimiak, Andrzej; Rizzi, Menico; Mizrahi, Valerie; Cuny, Gregory D.; Hedstrom, Lizbeth 分享 收藏
The Enzymatic Activity of Inosine 5′-Monophosphate Dehydrogenase May Not Be a Vulnerable Target for Staphylococcus aureus Infections Modi, Gyan; Marqus, Gary M.; Vippila, Mohana Rao; Gollapalli, Deviprasad R.; Kim, Youngchang; Manna, Adhar C.; Chacko, Shibin; Maltseva, Natalia; Wang, Xingyou; Cullinane, Ryan T.; Zhang, Yubo; Kotler, Judy L. M.; Kuzmic, Petr; Zhang, Minjia; Lawson, Ann P.; Joachimiak, Andrzej; Cheung, Ambrose; Snider, Barry B.; Rothstein, David M.; Cuny, Gregory D.; Hedstrom, Lizbeth 分享 收藏
Development of Rofecoxib-Based Fluorescent Probes and Investigations on Their Solvatochromism, AIE Activity, Mechanochromism, and COX-2-Targeted Bioimaging Xie, Lijun; Li, Renfu; Zheng, Biyun; Xie, Zuoxu; Fang, Xuefen; Wang, Yanqi; Cuny, Gregory D.; Li, Zhenli; Lin, Bin; Chen, Xueyuan; Hu, Ming 分享 收藏
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Antioxidant and food additive BHA prevents TNF cytotoxicity by acting as a direct RIPK1 inhibitor Delanghe, Tom; Huyghe, Jon; Lee, Seungheon; Priem, Dario; Van Coillie, Samya; Gilbert, Barbara; Choi, Sze Men; Vandenabeele, Peter; Degterev, Alexei; Cuny, Gregory D.; Dondelinger, Yves; Bertrand, Mathieu J. M. 分享 收藏
Fentanyl conjugate vaccine by injected or mucosal delivery with dmLT or LTA1 adjuvants implicates IgA in protection from drug challenge Stone, Addison E.; Scheuermann, Sarah E.; Haile, Colin N.; Cuny, Gregory D.; Velasquez, Marcela Lopez; Linhuber, Joshua P.; Duddupudi, Anantha L.; Vigliaturo, Jennifer R.; Pravetoni, Marco; Kosten, Therese A.; Kosten, Thomas R.; Norton, Elizabeth B. 分享 收藏
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Receptor-interacting protein kinase 2 (RIPK2) and nucleotide-binding oligomerization domain (NOD) cell signaling inhibitors based on a 3,5-diphenyl-2-aminopyridine scaffold 基于3,5-二苯基-2-氨基吡啶支架的受体相互作用蛋白激酶2 (RIPK2) 和核苷酸结合寡聚化结构域 (NOD) 细胞信号抑制剂 Suebsuwong, Chalada; Dai, Bing; Pinkas, Daniel M.; Duddupudi, Anantha Lakshmi; Li, Li; Bufton, Joshua C.; Schlicher, Lisa; Gyrd-Hansen, Mads; Hu, Ming; Bullock, Alex N.; Degterev, Alexei; Cuny, Gregory D. 分享 收藏
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Canvass: A Crowd-Sourced, Natural-Product Screening Library for Exploring Biological Space Kearney, Sara E.; Zahoranszky-Kohalmi, Gergely; Brimacombe, Kyle R.; Henderson, Mark J.; Lynch, Caitlin; Zhao, Tongan; Wan, Kanny K.; Itkin, Zina; Dillon, Christopher; Shen, Min; Cheff, Dorian M.; Lee, Tobie D.; Bougie, Danielle; Cheng, Ken; Coussens, Nathan P.; Dorjsuren, Dorjbal; Eastman, Richard T.; Huang, Ruili; Iannotti, Michael J.; Karavadhi, Surendra; Klumpp-Thomas, Carleen; Roth, Jacob S.; Sakamuru, Srilatha; Sun, Wei; Titus, Steven A.; Yasgar, Adam; Zhang, Ya-Qin; Zhao, Jinghua; Andrade, Rodrigo B.; Brown, M. Kevin; Burns, Noah Z.; Cha, Jin K.; Mevers, Emily E.; Clardy, Jon; Clement, Jason A.; Crooks, Peter A.; Cuny, Gregory D.; Ganor, Jake; Moreno, Jesus; Morrill, Lucas A.; Picazo, Elias; Susick, Robert B.; Garg, Neil K.; Goess, Brian C.; Grossman, Robert B.; Hughes, Chambers C.; Johnston, Jeffrey N.; Joullie, Madeleine M.; Kinghorn, A. Douglas; Kingston, David G. I.; Krische, Michael J.; Kwon, Ohyun; Maimone, Thomas J.; Majumdar, Susruta; Maloney, Katherine N.; Mohamed, Enas; Murphy, Brian T.; Nagorny, Pavel; Olson, David E.; Overman, Larry E.; Brown, Lauren E.; Snyder, John K.; Porco, John A., Jr.; Rivas, Fatima; Ross, Samir A.; Sarpong, Richmond; Sharma, Indrajeet; Shaw, Jared T.; Xu, Zhengren; Shen, Ben; Shi, Wei; Stephenson, Corey R. J.; Verano, Alyssa L.; Tan, Derek S.; Tang, Yi; Taylor, Richard E.; Thomson, Regan J.; Vosburg, David A.; Wu, Jimmy; Wuest, William M.; Zakarian, Armen; Zhang, Yufeng; Ren, Tianjing; Zuo, Zhong; Inglese, James; Michael, Sam; Simeonov, Anton; Zheng, Wei; Shinn, Paul; Jadhav, Ajit; Boxer, Matthew B.; Hall, Matthew D.; Xia, Menghang; Guha, Rajarshi; Rohde, Jason M. 分享 收藏