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摘要
Keyword:EXTRA-TERMINAL DOMAIN
BROMODOMAIN
INHIBITORS
DISCOVERY
IDENTIFICATION
AFFINITY
LIGANDS
DESIGN

引用论文
Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors
Seal, Jonathan T.; Atkinson, Stephen J.; Bamborough, Paul; Bassil, Anna; Chung, Chun-Wa; Foley, James; Gordon, Laurie; Grandi, Paola; Gray, James R. J.; Harrison, Lee A.; Kruger, Ryan G.; Matteo, Jeanne J.; McCabe, Michael T.; Messenger, Cassie; Mitchell, Darren; Phillipou, Alex; Preston, Alex; Prinjha, Rab K.; Rianjongdee, Francesco; Rioja, Inmaculada; Taylor, Simon; Wall, Ian D.; Watson, Robert J.; Woolven, James M.; Wyce, Anastasia; Zhang, Xi-Ping; Demont, Emmanuel H.
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收藏Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain
Brand, Michael; Clayton, James; Moroglu, Mustafa; Schiedel, Matthias; Picaud, Sarah; Bluck, Joseph P.; Skwarska, Anna; Bolland, Hannah; Chan, Anthony K. N.; Laurin, Corentine M. C.; Scorah, Amy R.; See, Larissa; Rooney, Timothy P. C.; Andrews, Katrina H.; Fedorov, Oleg; Perell, Gabriella; Kalra, Prakriti; Vinh, Kayla B.; Cortopassi, Wilian A.; Heitel, Pascal; Christensen, Kirsten E.; Cooper, Richard, I; Paton, Robert S.; Pomerantz, William C. K.; Biggin, Philip C.; Hammond, Ester M.; Filippakopoulos, Panagis; Conway, Stuart J.
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收藏Discovery of High-Affinity Inhibitors of the BPTF Bromodomain
Lu, Tian; Lu, Haibo; Duan, Zhe; Wang, Jun; Han, Jie; Xiao, Senhao; Chen, HuanHuan; Jiang, Hao; Chen, Yu; Yang, Feng; Chen, Dongying; Lin, Jin; Li, Bo; Jiang, Hualiang; Chen, Kaixian; Lu, Wenchao; Lin, Hua; Luo, Cheng
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收藏Structure-Activity Relationship and In Silico Evaluation of cis- and trans-PCPA-Derived Inhibitors of LSD1 and LSD2
Niwa, Hideaki; Watanabe, Chiduru; Sato, Shin; Harada, Toshiyuki; Watanabe, Hisami; Tabusa, Ryo; Fukasawa, Shunsuke; Shiobara, Ayane; Hashimoto, Tomoko; Ohno, Osamu; Nakamura, Kana; Tsuganezawa, Keiko; Tanaka, Akiko; Shirouzu, Mikako; Honma, Teruki; Matsuno, Kenji; Umehara, Takashi
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