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ACS Medicinal Chemistry Letters 封面图
ACS Medicinal Chemistry Letters
IF:
4
论文数:
4.4K
被引数:
10.0K

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Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors
err2021-07-13
err17
PREAI
errSeal, Jonathan T.; Atkinson, Stephen J.; Bamborough, Paul; Bassil, Anna; Chung, Chun-Wa; Foley, James; Gordon, Laurie; Grandi, Paola; Gray, James R. J.; Harrison, Lee A.; Kruger, Ryan G.; Matteo, Jeanne J.; McCabe, Michael T.; Messenger, Cassie; Mitchell, Darren; Phillipou, Alex; Preston, Alex; Prinjha, Rab K.; Rianjongdee, Francesco; Rioja, Inmaculada; Taylor, Simon; Wall, Ian D.; Watson, Robert J.; Woolven, James M.; Wyce, Anastasia; Zhang, Xi-Ping; Demont, Emmanuel H.
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Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain
err2021-07-13
err19
errOAAI
errBrand, Michael; Clayton, James; Moroglu, Mustafa; Schiedel, Matthias; Picaud, Sarah; Bluck, Joseph P.; Skwarska, Anna; Bolland, Hannah; Chan, Anthony K. N.; Laurin, Corentine M. C.; Scorah, Amy R.; See, Larissa; Rooney, Timothy P. C.; Andrews, Katrina H.; Fedorov, Oleg; Perell, Gabriella; Kalra, Prakriti; Vinh, Kayla B.; Cortopassi, Wilian A.; Heitel, Pascal; Christensen, Kirsten E.; Cooper, Richard, I; Paton, Robert S.; Pomerantz, William C. K.; Biggin, Philip C.; Hammond, Ester M.; Filippakopoulos, Panagis; Conway, Stuart J.
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Discovery of High-Affinity Inhibitors of the BPTF Bromodomain
err2021-08-10
err16
PREAI
errLu, Tian; Lu, Haibo; Duan, Zhe; Wang, Jun; Han, Jie; Xiao, Senhao; Chen, HuanHuan; Jiang, Hao; Chen, Yu; Yang, Feng; Chen, Dongying; Lin, Jin; Li, Bo; Jiang, Hualiang; Chen, Kaixian; Lu, Wenchao; Lin, Hua; Luo, Cheng
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Multivalent Peptide Ligands To Probe the Chromocenter Microenvironment in Living Cells
err2022-04-21
err14
errOAAI
errGuidotti, Nora; Eoerdogh, Adam; Mivelaz, Maxime; Rivera-Fuentes, Pablo; Fierz, Beat
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Structure-Activity Relationship and In Silico Evaluation of cis- and trans-PCPA-Derived Inhibitors of LSD1 and LSD2
err2022-08-18
err11
errOAAI
errNiwa, Hideaki; Watanabe, Chiduru; Sato, Shin; Harada, Toshiyuki; Watanabe, Hisami; Tabusa, Ryo; Fukasawa, Shunsuke; Shiobara, Ayane; Hashimoto, Tomoko; Ohno, Osamu; Nakamura, Kana; Tsuganezawa, Keiko; Tanaka, Akiko; Shirouzu, Mikako; Honma, Teruki; Matsuno, Kenji; Umehara, Takashi
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