Virtual Special Issue: Epigenetics 2022

doi:10.1021/acsinfecdis.2c00434

2022-09-08

PRE

DOI：10.1021/acsinfecdis.2c00434

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Without question, epigenetics is one of the fastest growing, and most impactful, fields in chemical biology, neuroscience, medicinal chemistry, and drug discovery today. Recognizing the importance of this area, in 2020 we invited submissions for a virtual special issue on this topic hosted by Pharmacology & Translational Science, and the Journal of Medicinal Chemistry. We are now delighted to present the Epigenetics 2022 virtual special issue. Below, content from each of the journals involved in this collection of papers is highlighted.

Keyword:

EXTRA-TERMINAL DOMAIN

BROMODOMAIN

INHIBITORS

DISCOVERY

IDENTIFICATION

AFFINITY

LIGANDS

DESIGN

期刊

ACS Infectious Diseases

IF:

3.8

论文数:

2.5K

被引数:

6.9K

机构

暂无机构信息

引用论文

Fragment-based Scaffold Hopping: Identification of Potent, Selective, and Highly Soluble Bromo and Extra Terminal Domain (BET) Second Bromodomain (BD2) Inhibitors

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2021-07-13

PREAI

Seal, Jonathan T.; Atkinson, Stephen J.; Bamborough, Paul; Bassil, Anna; Chung, Chun-Wa; Foley, James; Gordon, Laurie; Grandi, Paola; Gray, James R. J.; Harrison, Lee A.; Kruger, Ryan G.; Matteo, Jeanne J.; McCabe, Michael T.; Messenger, Cassie; Mitchell, Darren; Phillipou, Alex; Preston, Alex; Prinjha, Rab K.; Rianjongdee, Francesco; Rioja, Inmaculada; Taylor, Simon; Wall, Ian D.; Watson, Robert J.; Woolven, James M.; Wyce, Anastasia; Zhang, Xi-Ping; Demont, Emmanuel H.

Chemical Biology Approaches to Identify and Profile Interactors of Chromatin Modifications

ACS CHEMICAL BIOLOGY

IF3.8

2022-03-03

OAAI

Nickel, Garrison A.; Diehl, Katharine L.

Non trivial behaviour of the photoluminescence transition intensities in a modulation doped GaAs/GaAlAs single quantum well in tilted magnetic field

Solid State Communications

IF0

1998-05-01

PREAI

B. Couzinet; M. Dyakonov; A. Raymond; I. Elmezouar; M. Kamal-Saadi; B. Etienne

Controlling Intramolecular Interactions in the Design of Selective, High-Affinity Ligands for the CREBBP Bromodomain

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2021-07-13

OAAI

Brand, Michael; Clayton, James; Moroglu, Mustafa; Schiedel, Matthias; Picaud, Sarah; Bluck, Joseph P.; Skwarska, Anna; Bolland, Hannah; Chan, Anthony K. N.; Laurin, Corentine M. C.; Scorah, Amy R.; See, Larissa; Rooney, Timothy P. C.; Andrews, Katrina H.; Fedorov, Oleg; Perell, Gabriella; Kalra, Prakriti; Vinh, Kayla B.; Cortopassi, Wilian A.; Heitel, Pascal; Christensen, Kirsten E.; Cooper, Richard, I; Paton, Robert S.; Pomerantz, William C. K.; Biggin, Philip C.; Hammond, Ester M.; Filippakopoulos, Panagis; Conway, Stuart J.

Discovery of High-Affinity Inhibitors of the BPTF Bromodomain

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2021-08-10

PREAI

Lu, Tian; Lu, Haibo; Duan, Zhe; Wang, Jun; Han, Jie; Xiao, Senhao; Chen, HuanHuan; Jiang, Hao; Chen, Yu; Yang, Feng; Chen, Dongying; Lin, Jin; Li, Bo; Jiang, Hualiang; Chen, Kaixian; Lu, Wenchao; Lin, Hua; Luo, Cheng

YEATS Domains as Novel Epigenetic Readers: Structures, Functions, and Inhibitor Development

ACS CHEMICAL BIOLOGY

IF3.8

2022-01-18

PREAI

Li, Xin; Liu, Sha; Li, Xiang; Li, Xiang David

Multivalent Peptide Ligands To Probe the Chromocenter Microenvironment in Living Cells

ACS CHEMICAL BIOLOGY

IF3.8

2022-04-21

OAAI

Guidotti, Nora; Eoerdogh, Adam; Mivelaz, Maxime; Rivera-Fuentes, Pablo; Fierz, Beat

Structure-Activity Relationship and In Silico Evaluation of cis- and trans-PCPA-Derived Inhibitors of LSD1 and LSD2

ACS MEDICINAL CHEMISTRY LETTERS

IF4

2022-08-18

OAAI

Niwa, Hideaki; Watanabe, Chiduru; Sato, Shin; Harada, Toshiyuki; Watanabe, Hisami; Tabusa, Ryo; Fukasawa, Shunsuke; Shiobara, Ayane; Hashimoto, Tomoko; Ohno, Osamu; Nakamura, Kana; Tsuganezawa, Keiko; Tanaka, Akiko; Shirouzu, Mikako; Honma, Teruki; Matsuno, Kenji; Umehara, Takashi

Laboratory investigation of indigenous consortia TERIJ-188 for incremental oil recovery.

IF0

PREAI

From Hit Seeking to Magic Bullets: The Successful Union of Epigenetic and Fragment Based Drug Discovery (EPIDD plus FBDD)

JOURNAL OF MEDICINAL CHEMISTRY

IF6.8

2021-09-30

PREAI

Vaidergorn, Miguel M.; Emery, Flavio da Silva; Ganesan, A.

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