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SaveRetinal degeneration protein 3 mutants are associated with cell-cycle arrest and apoptosis
Chen, Yaoyu; Hausmann, Jens; Zimmermann, Benjamin; Helgers, Simeon Oscar Arnulfo; Doemer, Patrick; Woitzik, Johannes; Raap, Ulrike; Gray, Natalie; Buettner, Andreas; Koch, Karl-Wilhelm; Braeuer, Anja U.
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SaveCDK2 inhibition demonstrates synthetic lethality in SCLC through apoptotic induction
Schomer, Nathan; Chen, Jinhong; Pang, Wei; Zhou, Tingru; Liu, Xipan; Liang, Wenhen; Guo, Yali; Cheng, Dai; Li, Fang; Liang, Jiaqi; Chen, Yaoyu; Sheng, Qing
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SaveThe anti-tumor activity of CDK2 inhibition alone or in combination with other anti-cancer agents in human cancers
Chen, Yaoyu; Chen, Jinhong; Guo, Yali; Pang, Wei; Zhou, Tingru; Liu, Xipan; Schomer, Nathan; Li, Fang; Liang, Jiaqi; Sheng, Qing
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SaveDiscovery of Novel Pyrazolopyrimidines as Potent, Selective, and Orally Bioavailable Inhibitors of ALK2
Nguyen, Minh H.; Atasoylu, Onur; Wu, Liangxing; Kapilashrami, Kanishk; Pusey, Michelle; Gallagher, Karen; Lai, Cheng-Tsung; Zhao, Peng; Barbosa, Joseph; Liu, Kai; He, Chunhong; Zhang, Colin; Styduhar, Evan D.; Witten, Michael R.; Chen, Yaoyu; Lin, Luping; Yang, Yan-ou; Covington, Maryanne; Diamond, Sharon; Yeleswaram, Swamy; Yao, Wenqing
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SaveCharacterization of ARTS-011, a potent and selective TYK2 inhibitor for the treatment of inflammatory disease
Liang, Jiaqi; Liu, Yiting; Zhang, Xiaobin; Zhang, Tao; Liu, Xipan; Fu, Jia; Cheng, Dai; Xiong, Wen; Ding, Peter; Zhu, Cong; Li, Fang; Chen, Yaoyu
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SaveThe role of HPK1 in the regulation of T cell function and anti-tumor immune activity
Chen, Yaoyu; Rios-Doria, Jonathan; Pusey, Michelle; Lasky, Kerri; Ye, Min; Thekkat, Pramod; Gallagher, Karen; Stump, Kristine; Conlen, Patricia; Gardiner, Christine; Wang, Hui; Sokolsky, Alexander; Rupar, Mark; Lin, Luping; Behshad, Elham; Covington, Maryanne; Koblish, Holly; Vechorkin, Oleg; Yao, Wenqing; Kim, Sunkyu; Chen, Yingnan
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SaveIdentification of pAKT as a pharmacodynamic marker for MER kinase in human melanoma G361 cells
Chen, Yaoyu; Favata, Margaret; Pusey, Michelle; Li, Jun; Lo, Yvonne; Ye, Min; Wynn, Richard; Wang, Xiaozhao; Yao, Wenqing; Chen, Yingnan
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