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Vedagopuram Sreekanth

Broad Institute of MIT and Harvard

17H-index
45Paper Count
931Citation Count
Published Papers 18
Publication Date
Ultrasmall Chemogenetic Tags with Group-Transfer Ligands
err2025-09-27
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errOAAI
errVedagopuram Sreekanth; Shaimaa H. Sindi; Santosh K. Chaudhary; Rajaiah Pergu; Prashant Singh; Endri Karaj; Surached Siriwongsup; Jeffrey E. Fung; Arghya Deb; Stephan J. DeCarlo; Jaron A. M. Mercer; Kei Yamada; Diego Rodriguez; David R. Liu; Amit Choudhary
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Phosphorylation-Inducing Molecules for Regulating Dynamic Cellular Processes
err2025-07-14
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errOAAI
errRajaiah Pergu; Vedagopuram Sreekanth; Praveen Kokkonda; Sophia Lai; Praveen K. Tiwari; Sameek Singh; Junya Kawai; Santanu Singha; Wenzhi Tian; Vikram Thimaradka; Surached Siriwongsup; Kien Tran; Amit Choudhary
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Small molecules that disrupt RAD54-BLM interaction hamper tumor proliferation in colon cancer chemoresistance models
err2024-02-29
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errOAAI
errKaur, Ekjot; Agrawal, Ritu; Arun, Rimpy; Madhavan, Vinoth; Srivastava, Vivek; Kumar, Dilip; Rath, Pragyan Parimita; Kumar, Nitin; Vedagopuram, Sreekanth; Pandey, Nishant; Priya, Swati; Legembre, Patrick; Gourinath, Samudrala; Bajaj, Avinash; Sengupta, Sagar
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FALCON systematically interrogates free fatty acid biology and identifies a novel mediator of lipotoxicity
err2023-05-01
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errOAAI
errWieder, Nicolas; Fried, Juliana Coraor; Kim, Choah; Sidhom, Eriene-Heidi; Brown, Matthew R.; Marshall, Jamie L.; Arevalo, Carlos; Dvela-Levitt, Moran; Kost-Alimova, Maria; Sieber, Jonas; Gabriel, Katlyn R.; Pacheco, Julian; Clish, Clary; Abbasi, Hamdah Shafqat; Singh, Shantanu; Rutter, Justine C.; Therrien, Martine; Yoon, Haejin; Lai, Zon Weng; Baublis, Aaron; Subramanian, Renuka; Devkota, Ranjan; Small, Jonnell; Sreekanth, Vedagopuram; Han, Myeonghoon; Lim, Donghyun; Carpenter, Anne E.; Flannick, Jason; Finucane, Hilary; Haigis, Marcia C.; Claussnitzer, Melina; Sheu, Eric; Stevens, Beth; Wagner, Bridget K.; Choudhary, Amit; Shaw, Jillian L.; Pablo, Juan Lorenzo; Greka, Anna
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A general approach to identify cell-permeable and synthetic anti-CRISPR small molecules
err2022-11-17
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errOAAI
errLim, Donghyun; Zhou, Qingxuan; Cox, Kurt J.; Law, Benjamin K.; Lee, Miseon; Kokkonda, Praveen; Sreekanth, Vedagopuram; Pergu, Rajaiah; Chaudhary, Santosh K.; Gangopadhyay, Soumyashree A.; Maji, Basudeb; Lai, Sophia; Amako, Yuka; Thompson, David B.; Subramanian, Hari K. K.; Mesleh, Michael F.; Dandik, Vlado; Clemons, Paul A.; Wagner, Bridget K.; Woo, Christina M.; Church, George M.; Choudhary, Amit
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CRISPR-based therapeutics: current challenges and future applications
err2022-02-01
err41
errOAAI
errModell, Ashley E.; Lim, Donghyun; Nguyen, Tuan M.; Sreekanth, Vedagopuram; Choudhary, Amit
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Bile Acid Tethered Docetaxel-Based Nanomicelles Mitigate Tumor Progression through Epigenetic Changes
err2021-01-19
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PREAI
errSreekanth, Vedagopuram; Kar, Animesh; Kumar, Sandeep; Pal, Sanjay; Yadav, Poonam; Sharma, Yamini; Komalla, Varsha; Sharma, Harsh; Shyam, Radhey; Sharma, Ravi Datta; Mukhopadhyay, Arnab; Sengupta, Sagar; Dasgupta, Ujjaini; Bajaj, Avinash
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Self-assembled supramolecular nanomicelles from a bile acid-docetaxel conjugate are highly tolerable with improved therapeutic efficacy
err2021-01-01
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PREAI
errSreekanth, Vedagopuram; Pal, Sanjay; Kumar, Sandeep; Komalla, Varsha; Yadav, Poonam; Shyam, Radhey; Sengupta, Sagar; Bajaj, Avinash
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A 3D culture platform enables development of zinc-binding prodrugs for targeted proliferation of β cells
err2020-11-20
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errOAAI
errYang, Kisuk; Lee, Miseon; Jones, Peter Anthony; Liu, Sophie S.; Zhou, Angela; Xu, Jun; Sreekanth, Vedagopuram; Wu, Jamie L. Y.; Vo, Lillian; Lee, Eunjee A.; Pop, Ramona; Lee, Yuhan; Wagner, Bridget K.; Melton, Douglas A.; Choudhary, Amit; Karp, Jeffrey M.
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Chemogenetic System Demonstrates That Cas9 Longevity Impacts Genome Editing Outcomes
err2020-11-18
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errSreekanth, Vedagopuram; Zhou, Qingxuan; Kokkonda, Praveen; Bermudez-Cabrera, Heysol C.; Lim, Donghyun; Law, Benjamin K.; Holmes, Benjamin R.; Chaudhary, Santosh K.; Pergu, Rajaiah; Leger, Brittany S.; Walker, James A.; Gifford, David K.; Sherwood, Richard, I; Choudhary, Amit
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Engineering designer beta cells with a CRISPR-Cas9 conjugation platform
err2020-08-13
err35
errOAAI
errLim, Donghyun; Sreekanth, Vedagopuram; Cox, Kurt J.; Law, Benjamin K.; Wagner, Bridget K.; Karp, Jeffrey M.; Choudhary, Amit
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Tethering of Chemotherapeutic Drug/Imaging Agent to Bile Acid-Phospholipid Increases the Efficacy and Bioavailability with Reduced Hepatotoxicity
err2017-11-09
err17
PREAI
errSreekanth, Vedagopuram; Medatwal, Nihal; Kumar, Sandeep; Pal, Sanjay; Vamshikrishna, Malyla; Kar, Animesh; Bhargava, Priyanshu; Naaz, Aaliya; Kumar, Nitin; Sengupta, Sagar; Bajaj, Avinash
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Transcription regulation of CDKN1A (p21/CIP1/WAF1) by TRF2 is epigenetically controlled through the REST repressor complex
err2017-09-14
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errOAAI
errHussain, Tabish; Saha, Dhurjhoti; Purohit, Gunjan; Kar, Anirban; Mukherjee, Anand Kishore; Sharma, Shalu; Sengupta, Suman; Dhapola, Parashar; Maji, Basudeb; Vedagopuram, Sreekanth; Horikoshi, Nobuko T.; Horikoshi, Nobuo; Pandita, Raj K.; Bhattacharya, Santanu; Bajaj, Avinash; Riou, Jean-Francois; Pandita, Tej K.; Chowdhury, Shantanu
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Design, regioselective synthesis and cytotoxic evaluation of 2-aminoimidazole-quinoline hybrids against cancer and primary endothelial cells
err2014-11-01
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PREAI
errSingh, Kuldeep; Verma, Vikas; Yadav, Kavita; Sreekanth, Vedagopuram; Kumar, Devinder; Bajaj, Avinash; Kumar, Vinod
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Injectable small molecule hydrogel as a potential nanocarrier for localized and sustained in vivo delivery of doxorubicin
err2014-01-01
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PREAI
errSingh, Manish; Kundu, Somanath; Reddy, Amarendar M.; Sreekanth, Vedagopuram; Motiani, Rajender K.; Sengupta, Sagar; Srivastava, Aasheesh; Bajaj, Avinash
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Design, Synthesis, and Mechanistic Investigations of Bile Acid-Tamoxifen Conjugates for Breast Cancer Therapy
err2013-08-21
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PREAI
errSreekanth, Vedagopuram; Bansal, Sandhya; Motiani, Rajender K.; Kundu, Somanath; Muppu, Sravan Kumar; Majumdar, Tapodhara Datta; Panjamurthy, Kuppusamy; Sengupta, Sagar; Bajaj, Avinash
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