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Thomas J. Abbruscato

Texas Tech University

36H-index
113Paper Count
3.6KCitation Count
Published Papers 54
Publication Date
Discovery of a pyridine-piperazine-based small molecule that enhances the activity of peptidase neurolysin
err2026-02-03
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PREAI
errHeba ElSayed ElZorkany; Haya Kandil; Srinidhi Jayaraman; Asmaa Aly; Shiva Hadi Esfahani; Dhavalkumar Patel; Dennis Dannecker; Monika Maciag; Alyssa Paul; Kaitlin Lowran; Shikha Kumari; Samik Bose; David A. Ostrov; Colin G. Wu; Alex Dickson; Thomas J. Abbruscato; Paul C. Trippier; Benjamin J. Orlando; Vardan T. Karamyan
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Metformin's Permeability Across the Ischemic Brain and an Assessment of Blood-Brain Barrier
err2025-03-01
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PREAI
errAkter, Khondker Ayesha; Sharma, Sejal; Jadhav, Sejal Rajesh; Zhang, Yong; Abbruscato, Thomas J.
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Evaluation of systemic and brain pharmacokinetic parameters for repurposing metformin using intravenous bolus administration
err2025-01-01
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errOAAI
errSharma, Sejal; Zhang, Yong; Patel, Dhavalkumar; Akter, Khondker Ayesha; Bagchi, Sounak; Sifat, Ali Ehsan; Nozohouri, Ehsan; Ahn, Yeseul; Karamyan, Vardan T.; Bickel, Ulrich; Abbruscato, Thomas J.
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The Acute Impact of Propofol on Blood-Brain Barrier Integrity in Mice
err2024-07-24
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PREAI
errNozohouri, Ehsan; Ahn, Yeseul; Zoubi, Sumaih; Patel, Dhavalkumar; Archie, Sabrina Rahman; Akter, Khondker Ayesha; Siddique, Muhammad Bilal; Huang, Juyang; Abbruscato, Thomas J.; Bickel, Ulrich
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Imidazole Bioisostere Activators of Endopeptidase Neurolysin with Enhanced Potency and Metabolic Stability
err2024-03-29
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PREAI
errRahman, Md. Shafikur; Esfahani, Shiva Hadi; Zhang, Yong; Queen, Aarfa; Aljarrah, Manar; Kandil, Haya; Baez, Andrew; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C.
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Discovery of the Next Generation of Non-peptidomimetic Neurolysin Activators with High Blood-Brain Barrier Permeability: a Pharmacokinetics Study in Healthy and Stroke Animals
err2023-10-13
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PREAI
errZhang, Yong; Sharma, Sejal; Jonnalagadda, Shirisha; Kumari, Shikha; Queen, Aarfa; Esfahani, Shiva Hadi; Archie, Sabrina Rahman; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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Studies on diketopiperazine and dipeptide analogs as opioid receptor ligands
err2023-06-01
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errOAAI
errNia, Siavash Shahbazi; Hossain, Mohammad Anwar; Ji, Guangchen; Jonnalagadda, Sravan K.; Obeng, Samuel; Rahman, Md Ashrafur; Sifat, Ali Ehsan; Nozohouri, Saeideh; Blackwell, Collin; Patel, Dhavalkumar; Thompson, Jon; Runyon, Scott; Hiranita, Takato; McCurdy, Christopher R.; McMahon, Lance; Abbruscato, Thomas J.; Trippier, Paul C.; Neugebauer, Volker; German, Nadezhda A.
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High brain-blood barrier permeability highlights a new class of neurolysin activators as promising candidates for stroke treatment: a pilot pharmacokinetic study in mice
err2023-06-01
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errOAAI
errZhang, Yong; Sharma, Sejal; Esfahani, Shiva H.; Jonnalagadda, Shirisha; Queen, Aarfa; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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Permeability of Metformin across an In Vitro Blood-Brain Barrier Model during Normoxia and Oxygen-Glucose Deprivation Conditions: Role of Organic Cation Transporters (Octs)
err2023-04-28
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errOAAI
errSharma, Sejal; Zhang, Yong; Akter, Khondker Ayesha; Nozohouri, Saeideh; Archie, Sabrina Rahman; Patel, Dhavalkumar; Villalba, Heidi; Abbruscato, Thomas
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Endothelial-Specific Targeting of RhoA Signaling via CD31 Antibody-Conjugated Nanoparticles
err2023-04-01
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PREAI
errLahooti, Behnaz; Akwii, Racheal G.; Patel, Dhavalkumar; ShahbaziNia, Siavash; Lamprou, Margarita; Madadi, Mahboubeh; Abbruscato, Thomas J.; Astrinidis, Aristotelis; Bickel, Ulrich; Al-Ahmad, Abraham; German, Nadezhda A.; Mattheolabakis, George; Mikelis, Constantinos M.
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Maternal e-cigarette use can disrupt postnatal blood-brain barrier (BBB) integrity and deteriorates motor, learning and memory function: influence of sex and age
err2023-03-10
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errOAAI
errArchie, Sabrina Rahman; Sifat, Ali Ehsan; Zhang, Yong; Villalba, Heidi; Sharma, Sejal; Nozohouri, Saeideh; Abbruscato, Thomas J.
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Potential role of astrocyte angiotensin converting enzyme 2 in the neural transmission of COVID-19 and a neuroinflammatory state induced by smoking and vaping (vol 19, 46, 2022)
err2022-11-17
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errOAAI
errZhang, Yong; Archie, Sabrina Rahman; Ghanwatkar, Yashwardhan; Sharma, Sejal; Nozohouri, Saeideh; Burks, Elizabeth; Mdzinarishvili, Alexander; Liu, Zijuan; Abbruscato, Thomas J.
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Dental Pulp-Derived Stem Cells Preserve Astrocyte Health During Induced Gliosis by Modulating Mitochondrial Activity and Functions
err2022-10-06
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PREAI
errBarthels, Derek; Prateeksha, Prateeksha; Nozohouri, Saeideh; Villalba, Heidi; Zhang, Yong; Sharma, Sejal; Anderson, Sarah; Howlader, Md Sariful Islam; Nambiar, Adarsh; Abbruscato, Thomas J.; Das, Hiranmoy
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Short-term exposure to JUUL electronic cigarettes can worsen ischemic stroke outcome
err2022-09-09
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errOAAI
errSifat, Ali Ehsan; Archie, Sabrina Rahman; Nozohouri, Saeideh; Villalba, Heidi; Zhang, Yong; Sharma, Sejal; Ghanwatkar, Yashwardhan; Vaidya, Bhuvaneshwar; Mara, David; Cucullo, Luca; Abbruscato, Thomas J.
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Potential role of astrocyte angiotensin converting enzyme 2 in the neural transmission of COVID-19 and a neuroinflammatory state induced by smoking and vaping
err2022-06-07
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errOAAI
errZhang, Yong; Archie, Sabrina Rahman; Ghanwatkar, Yashwardhan; Sharma, Sejal; Nozohouri, Saeideh; Burks, Elizabeth; Mdzinarishvili, Alexander; Liu, Zijuan; Abbruscato, Thomas J.
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Prenatal E-Cigarette Use Disrupts Blood-Brain Barrier (BBB) Integrity and Induces Pro-Inflammatory Cytokines in Postnatal Brain
err2022-05-13
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PREAI
errArchie, Sabrina Rahman; Sifat, Ali Ehsan; Villalba, Heidi; Sharma, Sejal; Nozohouri, Saeideh; Zhang, Yong; Abbruscato, Thomas
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In-Vivo and Ex-Vivo Brain Uptake Studies of Peptidomimetic Neurolysin Activators in Healthy and Stroke Animals
err2022-03-03
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errOAAI
errNozohouri, Saeideh; Esfahani, Shiva Hadi; Noorani, Behnam; Patel, Dhaval; Villalba, Heidi; Ghanwatkar, Yashwardhan; Rahman, Md Shafikur; Zhang, Yong; Bickel, Ulrich; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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