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SaveOptimization of Selective and CNS Penetrant Alkyne-Based TREK Inhibitors: The Discovery and Characterization of ONO-9517601 (VU6022856) and ONO-7927846 (VU6024391)
Tanaka, Motoyuki; Sekioka, Yoko; Hashimoto, Gakuji; Mori, Takahiro; Shono, Tomoyuki; Isaji, Yuuki; Hisaichi, Katsuya; Childress, Elizabeth S.; Bollinger, Sean; Schmitt, Joza A.; Chopko, Trevor C.; Garrison, Aaron T.; Perry, Charles K.; Chronister, Keagan; Kramer, Meghan; Chang, Sichen; Watson, Katherine J.; Dickerson, Jonathan W.; Bubser, Michael; Rook, Jerri M.; Jones, Carrie K.; Boutaud, Olivier; Bridges, Thomas M.; Denton, Jerod S.; Engers, Darren W.; Kurata, Haruto; Lindsley, Craig W.
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SaveDiscovery of ONO-TR-772 (VU6018042): A Highly Selective and CNS Penetrant TREK Inhibitor in Vivo Tool Compound
Tanaka, M; Mori, T; Hashimoto, G; Mitsui, K; Kishi, A; Childress, ES; Bollinger, SR; Chopko, TC; Bridges, TM; Stafford, DG; Huang, ZP; Wolf, MA; Engers, DW; Denton, JS; Kurata, H; Lindsley, CW
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SaveDiscovery of ONO-2920632 (VU6011887): A Highly Selective and CNS Penetrant TREK-2 (TWIK-Related K+ Channel 2) Preferring Activator In Vivo Tool Compound
Yashiro, K; Iwaki, Y; Urata, H; Kokubo, M; Mori, T; Sekioka, Y; Isami, K; Kato, J; Wieting, J; Mcgowan, KM; Bridges, TM; Boutaud, O; Engers, DW; Denton, JS; Kurata, H; Lindsley, CW
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SaveMolecular basis for the diversification of lincosamide biosynthesis by pyridoxal phosphate-dependent enzymes
Mori, Takahiro; Moriwaki, Yoshitaka; Sakurada, Kosuke; Lyu, Shuang; Kadlcik, Stanislav; Janata, Jiri; Mazumdar, Aninda; Koberska, Marketa; Terada, Tohru; Kamenik, Zdenek; Abe, Ikuro
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SaveMechanistic Analysis of Stereodivergent Nitroalkane Cyclopropanation Catalyzed by Nonheme Iron Enzymes
Ushimaru, Richiro; Cha, Lide; Shimo, Shotaro; Li, Xiaojun; Paris, Jared C.; Mori, Takahiro; Miyamoto, Kazunori; Coffer, Lindsay; Uchiyama, Masanobu; Guo, Yisong; Chang, Wei-chen; Abe, Ikuro
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SaveCordycicadins A-D, Antifeedant Polyketides from the Entomopathogenic Fungus Cordyceps cicadae JXCH1
Li, Xinyang; Chen, He-Ping; Zhou, Lin; Fan, Jing; Awakawa, Takayoshi; Mori, Takahiro; Ushimaru, Richiro; Abe, Ikuro; Liu, Ji-Kai
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SaveIdentification of a diarylpentanoid-producing polyketide synthase revealing an unusual biosynthetic pathway of 2-(2-phenylethyl)chromones in agarwood
Wang, Xiao-Hui; Gao, Bo-Wen; Nakashima, Yu; Mori, Takahiro; Zhang, Zhong-Xiu; Kodama, Takeshi; Lee, Yuan-E; Zhang, Ze-Kun; Wong, Chin-Piow; Liu, Qian-Qian; Qi, Bo-Wen; Wang, Juan; Li, Jun; Liu, Xiao; Abe, Ikuro; Morita, Hiroyuki; Tu, Peng-Fei; Shi, She-Po
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