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Paul S. Rennie

University of British Columbia

64H-index
521Paper Count
1.4WCitation Count
Published Papers 127
Publication Date
Endoplasmic reticulum stress-driven nucleotide catabolism fuels prostate cancer
err2025-07-03
err0
errOAAI
errKe Deng; Nora Pällmann; Marte Livgård; Wanja Kildal; Manohar Pradhan; Ladan Fazli; Paul S. Rennie; Yang Jin; Fahri Saatcioglu; Omer F. Kuzu
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IRE1α-XBP1s pathway promotes prostate cancer by activating c-MYC signaling (vol10, 323, 2019)
err2024-07-23
err1
errOAAI
errSheng, Xia; Nenseth, Hatice Zeynep; Qu, Su; Kuzu, Omer F.; Frahnow, Turid; Simon, Lukas; Greene, Stephanie; Zeng, Qingping; Fazli, Ladan; Rennie, Paul S.; Mills, Ian G.; Danielsen, Havard; Theis, Fabian; Patterson, John B.; Jin, Yang; Saatcioglu, Fahri
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Clinically-observed FOXA1 mutations upregulate SEMA3C through transcriptional derepression in prostate cancer
err2024-03-25
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errOAAI
errTam, Kevin J.; Liu, Liangliang; Hsing, Michael; Dalal, Kush; Thaper, Daksh; McConeghy, Brian; Yenki, Parvin; Bhasin, Satyam; Peacock, James W.; Wang, Yuzhuo; Cherkasov, Artem; Rennie, Paul S.; Gleave, Martin E.; Ong, Christopher J.
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Dynamic phase separation of the androgen receptor and its coactivators key to regulate gene expression
err2022-12-20
err30
errOAAI
errZhang, Fan; Biswas, Maitree; Massah, Shabnam; Lee, Joseph; Lingadahalli, Shreyas; Wong, Samantha; Wells, Christopher; Foo, Jane; Khan, Nabeel; Morin, Helene; Saxena, Neetu; Kung, Sonia H. Y.; Sun, Bei; Nunez, Ana Karla Parra; Sanchez, Christophe; Chan, Novia; Ung, Lauren; Altintas, Umut Berkay; Bui, Jennifer M.; Wang, Yuzhuo; Fazli, Ladan; Oo, Htoo Zarni; Rennie, Paul S.; Lack, Nathan A.; Cherkasov, Artem; Gleave, Martin E.; Gsponer, Jorg; Lallous, Nada
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Structure-Based Study to Overcome Cross-Reactivity of Novel Androgen Receptor Inhibitors
errCELLS
IF5.2
err2022-09-07
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errOAAI
errRadaeva, Mariia; Li, Huifang; LeBlanc, Eric; Dalal, Kush; Ban, Fuqiang; Ciesielski, Fabrice; Chow, Bonny; Morin, Helene; Awrey, Shannon; Singh, Kriti; Rennie, Paul S.; Lallous, Nada; Cherkasov, Artem
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Development of 2-(5,6,7-Trifluoro-1H-Indol-3-yl)-quinoline-5-carboxamide as a Potent, Selective, and Orally Available Inhibitor of Human Androgen Receptor Targeting Its Binding Function-3 for the Treatment of Castration-Resistant Prostate Cancer
err2021-10-18
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PREAI
errLeblanc, Eric; Ban, Fuqiang; Cavga, Ayse Derya; Lawn, Sam; Huang, Chia-Chi Flora; Mohan, Sankar; Chang, Matthew E. K.; Flory, Mark R.; Ghaidi, Fariba; Lingadahalli, Shreyas; Chen, Gang; Yu, Ivan Pak Lok; Morin, Helene; Lallous, Nada; Gleave, Martin E.; Mohammed, Hisham; Young, Robert N.; Rennie, Paul S.; Lack, Nathan A.; Cherkasov, Artem
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Stress-Mediated Reprogramming of Prostate Cancer One-Carbon Cycle Drives Disease Progression
err2021-06-28
err14
errOAAI
errPallmann, Nora; Deng, Ke; Livgard, Marte; Tesikova, Martina; Jin, Yixin; Frengen, Nicolai Sebastian; Kahraman, Nermin; Mokhlis, Hamada M.; Ozpolat, Bulent; Kildal, Wanja; Danielsen, Havard Emil; Fazli, Ladan; Rennie, Paul S.; Banerjee, Partha P.; Uren, Aykut; Jin, Yang; Kuzu, Omer F.; Saatcioglu, Fahri
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Androgen receptor plasticity and its implications for prostate cancer therapy
err2019-12-01
err43
PREAI
errSnow, Oliver; Lallous, Nada; Singh, Kriti; Lack, Nathan; Rennie, Paul; Cherkasov, Artem
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Regulation of the unfolded protein response through ATF4 and FAM129A in prostate cancer Nora
err2019-07-16
err45
PREAI
errPallmann, Nora; Livgard, Marte; Tesikova, Martina; Nenseth, Hatice Zeynep; Akkus, Erman; Sikkeland, Jorgen; Jin, Yixin; Koc, Dogukan; Kuzu, Omer Faruk; Pradhan, Manohar; Danielsen, Havard E.; Kahraman, Nermin; Mokhlis, Hamada M.; Ozpolat, Bulent; Banerjee, Partha P.; Uren, Aykut; Fazli, Ladan; Rennie, Paul S.; Jin, Yang; Saatcioglu, Fahri
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UV Light-inactivated HSV-1 Stimulates Natural Killer Cell-induced Killing of Prostate Cancer Cells
err2019-06-01
err7
PREAI
errSamudio, Ismael; Hofs, Elyse; Cho, Brandon; Li, Michael; Bolduc, Kayla; Bu, Luke; Liu, Guoyu; Lam, Vivian; Rennie, Paul; Jia, William; Elisia, Ingrid; Krystal, Gerald
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ETS transcription factors as emerging drug targets in cancer
err2019-03-29
err54
PREAI
errHsing, Michael; Wang, Yuzhuo; Rennie, Paul S.; Cox, Michael E.; Cherkasov, Artem
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Computer-Aided Discovery of Small Molecules Targeting the RNA Splicing Activity of hnRNP A1 in Castration-Resistant Prostate Cancer
err2019-02-20
err30
errOAAI
errCarabet, Lavinia A.; Leblanc, Eric; Lallous, Nada; Morin, Helene; Ghaidi, Fariba; Lee, Joseph; Rennie, Paul S.; Cherkasov, Artem
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IRE1α-XBP1s pathway promotes prostate cancer by activating c-MYC signaling
err2019-01-24
err201
errOAAI
errSheng, Xia; Nenseth, Hatice Zeynep; Qu, Su; Kuzu, Omer F.; Frahnow, Turid; Simon, Lukas; Greene, Stephanie; Zeng, Qingping; Fazli, Ladan; Rennie, Paul S.; Mills, Ian G.; Danielsen, Havard; Theis, Fabian; Patterson, John B.; Jin, Yang; Saatcioglu, Fahri
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EComputer-aided drug discovery of Myc-Max inhibitors as potential therapeutics for prostate cancer
err2018-12-01
err40
errOAAI
errCarabet, Lavinia A.; Lallous, Nada; Leblanc, Eric; Ban, Fuqiang; Morin, Helene; Lawn, Sam; Ghaidi, Fariba; Lee, Joseph; Mills, Ian G.; Gleave, Martin E.; Rennie, Paul S.; Cherkasov, Artem
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Computer-Aided Discovery of Small Molecule Inhibitors of Transcriptional Activity of TLX (NR2E1) Nuclear Receptor
err2018-11-14
err10
errOAAI
errDueva, Evgenia; Singh, Kriti; Kalyta, Anastasia; LeBlanc, Eric; Rennie, Paul S.; Cherkasov, Artem
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Selectively targeting the dimerization interface of human androgen receptor with small-molecules to treat castration-resistant prostate cancer
err2018-11-01
err49
PREAI
errDalal, Kush; Ban, Fuqiang; Li, Huifang; Morin, Helene; Roshan-Moniri, Mani; Tam, Kevin J.; Shepherd, Ashley; Sharma, Aishwariya; Peacock, James; Carlson, Michael L.; LeBlanc, Eric; Perez, Carl; Duong, Franck; Ong, Christopher J.; Rennie, Paul S.; Cherkasov, Artem
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Small molecule-induced degradation of the full length and V7 truncated variant forms of human androgen receptor
err2018-09-01
err16
PREAI
errDalal, Kush; Morin, Helene; Ban, Fuqiang; Shepherd, Ashley; Fernandez, Michael; Tam, Kevin J.; Li, Huifang; LeBlanc, Eric; Lack, Nathan; Prinz, Helge; Rennie, Paul S.; Cherkasov, Artem
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AR is ablated: Now what? Targeting the double-negative phenotype.
err2018-08-14
err0
PREAI
errMorrissey, Colm; Bluemn, Eric G.; Coleman, Ilsa M.; Lucas, Jared M.; Coleman, Roger T.; Tharakan, Robin; Bianchi-Frias, Daniella; Dumpit, Ruth F.; Kaipainen, Arja; Corella, Alexandra N.; Yang, Yu Chi; Nyquist, Michael D.; Mostaghel, Elahe; Zhang, Xiaotun; Corey, Eva; Brown, Lisha G.; Nguyen, Holly M.; Schweizer, Michael; True, Lawrence D.; Rennie, Paul S.; Vessella, Robert L.; Nelson, Peter S.
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Toxic Colors: The Use of Deep Learning for Predicting Toxicity of Compounds Merely from Their Graphic Images
err2018-07-31
err94
PREAI
errFernandez, Michael; Ban, Fuqiang; Woo, Godwin; Hsing, Michael; Yamazaki, Takeshi; LeBlanc, Eric; Rennie, Paul S.; Welch, William J.; Cherkasov, Artem
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Oncolytic Virotherapy Blockade by Microglia and Macrophages Requires STAT1/3
err2018-01-31
err39
errOAAI
errDelwar, Zahid M.; Kuo, Yvonne; Wen, Yan H.; Rennie, Paul S.; Jia, William
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