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Dimitri E. Grigoriadis

Feinberg School of Medicine

57H-index
198Paper Count
9.8KCitation Count
Published Papers 32
Publication Date
Corticotropin-Releasing Factor Receptor 1 Antagonism Is Ineffective for Women With Posttraumatic Stress Disorder
err2017-12-01
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errDunlop, Boadie W.; Binder, Elisabeth B.; Iosifescu, Dan; Mathew, Sanjay J.; Neylan, Thomas C.; Pape, Julius C.; Carrillo-Roa, Tania; Green, Charles; Kinkead, Becky; Grigoriadis, Dimitri; Rothbaum, Barbara O.; Nemeroff, Charles B.; Mayberg, Helen S.
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Pharmacologic Characterization of Valbenazine (NBI-98854) and Its Metabolites
err2017-06-01
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errOAAI
errGrigoriadis, Dimitri E.; Smith, Evan; Hoare, Sam R. J.; Madan, Ajay; Bozigian, Haig
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Valbenazine (NBI-98854) and Its Major Metabolites Specifically Modulate Neuronal Monoaminergic Function
err2017-05-01
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PREAI
errKudwa, Andrea; Meltzer, Herbert; Huang, Mei; Grigoriadis, Dimitri
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The CRFI Antagonist Verucerfont in Anxious Alcohol-Dependent Women: Translation of Neuroendocrine, But not of Anti-Craving Effects
err2016-04-25
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errSchwandt, Melanie L.; Cortes, Carlos R.; Kwako, Laura E.; George, David T.; Momenan, Reza; Sinha, Rajita; Grigoriadis, Dimitri E.; Pich, Emilio Merlo; Leggio, Lorenzo; Heilig, Markus
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Single-Dose Study of a Corticotropin-Releasing Factor Receptor-1 Antagonist in Women With 21-Hydroxylase Deficiency
err2016-03-01
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errTurcu, Adina F.; Spencer-Segal, Joanna L.; Farber, Robert H.; Luo, Rosa; Grigoriadis, Dimitri E.; Ramm, Carole A.; Madrigal, David; Muth, Tim; O'Brien, Christopher F.; Auchus, Richard J.
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Hypocretin Receptor 2 Antagonism Dose-Dependently Reduces Escalated Heroin Self-Administration in Rats
err2014-11-04
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errSchmeichel, Brooke E.; Barbier, Estelle; Misra, Kaushik K.; Contet, Candice; Schlosburg, Joel E.; Grigoriadis, Dimitri; Williams, John P.; Karlsson, Camilla; Pitcairn, Caleb; Heilig, Markus; Koob, George F.; Vendruscolo, Leandro F.
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Binding Kinetics Redefine the Antagonist Pharmacology of the Corticotropin-Releasing Factor Type 1 Receptor
err2012-05-01
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PREAI
errFleck, Beth A.; Hoare, Sam R. J.; Pick, Rebecca R.; Bradbury, Margaret J.; Grigoriadis, Dimitri E.
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Depressive and cardiovascular disease comorbidity in a rat model of social stress: a putative role for corticotropin-releasing factor
err2012-02-10
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errWood, Susan K.; McFadden, Kile V.; Grigoriadis, Dimitri; Bhatnagar, Seema; Valentino, Rita J.
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CRF system recruitment mediates dark side of compulsive eating
err2009-11-24
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errCottone, Pietro; Sabino, Valentina; Roberto, Marisa; Bajo, Michal; Pockros, Lara; Frihauf, Jennifer B.; Fekete, Eva M.; Steardo, Luca; Rice, Kenner C.; Grigoriadis, Dimitri E.; Conti, Bruno; Koob, George F.; Zorrilla, Eric P.
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Drugability of Extracellular Targets: Discovery of Small Molecule Drugs Targeting Allosteric, Functional, and Subunit-Selective Sites on GPCRs and Ion Channels
err2008-09-17
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errGrigoriadis, Dimitri E.; Hoare, Samuel R. J.; Lechner, Sandra M.; Slee, Deborah H.; Williams, John A.
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Allosteric ligands for the corticotropin releasing factor type 1 receptor modulate conformational states involved in receptor activation
err2008-05-01
err32
PREAI
errHoare, Sam R. J.; Fleck, Beth A.; Gross, Raymond S.; Crowe, Paul D.; Williams, John P.; Grigoriadis, Dimitri E.
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High-affinity CRF1 receptor antagonist NBI-34041:: Preclinical and clinical data suggest safety and efficacy in attenuating elevated stress response
err2007-02-07
err126
errOAAI
errIsing, Marcus; Zimmermann, Ulrich S.; Kuenzel, Heike E.; Uhr, Manfred; Foster, Alan C.; Learned-Coughlin, Susan M.; Holsboer, Florian; Grigoriadis, Dimitri E.
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Corticotropin-releasing hormone receptor 2-deficient mice have reduced intestinal inflammatory responses
err2006-09-01
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errKokkotou, Efi; Torres, Daniel; Moss, Alan C.; O'Brien, Michael; Grigoriadis, Dimitri E.; Karalis, Katia; Pothoulakis, Charalabos
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Single amino acid residue determinants of non-peptide antagonist binding to the corticotropin-releasing factor1 (CRF1) receptor
err2006-07-01
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PREAI
errHoare, Sam R. J.; Brown, Brock T.; Santos, Mark A.; Malany, Siobhan; Betz, Stephen F.; Grigoriadis, Dimitri E.
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Design and synthesis of tricyclic corticotropin-releasing factor-1 antagonists
err2005-08-10
err56
PREAI
errGross, RS; Guo, ZQ; Dyck, B; Coon, T; Huang, CQ; Lowe, RF; Marinkovic, D; Moorjani, M; Nelson, J; Zamani-Kord, S; Grigoriadis, DE; Hoare, SRJ; Crowe, PD; Bu, JH; Haddach, M; McCarthy, J; Saunders, J; Sullivan, R; Chen, TK; Williams, JP
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Design and synthesis of tricyclic imidazo[4,5-b]pyridin-2-ones as corticotropin-releasing factor-1 antagonists
err2005-07-09
err25
PREAI
errGuo, ZQ; Tellew, JE; Gross, RS; Dyck, B; Grey, J; Haddach, M; Kiankarimi, M; Lanier, M; Li, BF; Luo, ZY; McCarthy, JR; Moorjani, M; Saunders, J; Sullivan, R; Zhang, XH; Zamani-Kord, S; Grigoriadis, DE; Crowe, PD; Chen, TK; Williams, JP
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Potent, orally active corticotropin-releasing factor receptor-1 antagonists containing a tricyclic pyrrolopyridine or pyrazolopyridine core
err2005-05-06
err31
PREAI
errDyck, B; Grigoriadis, DE; Gross, RS; Guo, ZQ; Haddach, M; Marinkovic, D; McCarthy, JR; Moorjani, M; Regan, CF; Saunders, J; Schwaebe, MK; Szabo, T; Williams, JP; Zhang, XH; Bozigian, H; Chen, TK
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