Not logged inProdrugs of a 1-hydroxy-2-oxopiperidin-3-yl phosphonate enolase inhibitor for the treatment of ENO1-deleted cancers
Yan, Victoria C.; Pham, Cong-Dat; Ballato, Elliot S.; Yang, Kristine L.; Khadka, Sunada; Barektain, Yasaman; Shrestha, Prakriti; Tran, Theresa; Poral, Anton H.; Washington, Mykia; Raghavan, Sudhir; Czako, Barbara; Pisaneschi, Federica; Lin, Yu-Hsi; Satani, Nikunj; Hammoudi, Naima; Ackroyd, Jeffrey J.; Georgiou, Dimitra K.; Millward, Steven W.; Muller, Florian L.
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SaveProdrugs of a 1-Hydroxy-2-oxopiperidin-3-yl Phosphonate Enolase Inhibitor for the Treatment of ENO1-Deleted Cancers
Yan, Victoria C.; Pham, Cong-Dat; Ballato, Elliot S.; Yang, Kristine L.; Arthur, Kenisha; Khadka, Sunada; Barekatain, Yasaman; Shrestha, Prakriti; Tran, Theresa; Poral, Anton H.; Washington, Mykia; Raghavan, Sudhir; Czako, Barbara; Pisaneschi, Federica; Lin, Yu-Hsi; Satani, Nikunj; Hammoudi, Naima; Ackroyd, Jeffrey J.; Georgiou, Dimitra K.; Millward, Steven W.; Muller, Florian L.
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SaveQuantification of Phosphonate Drugs by 1H-31P HSQC Shows That Rats Are Better Models of Primate Drug Exposure than Mice
Barekatain, Yasaman; Khadka, Sunada; Harris, Kristen; Delacerda, Jorge; Yan, Victoria C.; Chen, Ko-Chien; Pham, Cong-Dat; Uddin, Md. Nasir; Avritcher, Rony; Eisenberg, Eugene J.; Kalluri, Raghu; Millward, Steven W.; Muller, Florian L.
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SaveHomozygous MTAP deletion in primary human glioblastoma is not associated with elevation of methylthioadenosine
Barekatain, Yasaman; Ackroyd, Jeffrey J.; Yan, Victoria C.; Khadka, Sunada; Wang, Lin; Chen, Ko-Chien; Poral, Anton H.; Tran, Theresa; Georgiou, Dimitra K.; Arthur, Kenisha; Lin, Yu-Hsi; Satani, Nikunj; Ballato, Elliot S.; Behr, Eliot, I; deCarvalho, Ana C.; Verhaak, Roel G. W.; de Groot, John; Huse, Jason T.; Asara, John M.; Kalluri, Raghu; Muller, Florian L.
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SaveImpaired anaplerosis is a major contributor to glycolysis inhibitor toxicity in glioma
Khadka, Sunada; Arthur, Kenisha; Barekatain, Yasaman; Behr, Eliot; Washington, Mykia; Ackroyd, Jeffrey; Crowley, Kaitlyn; Suriyamongkol, Pornpa; Lin, Yu-Hsi; Pham, Cong-Dat; Zielinski, Rafal; Trujillo, Marissa; Galligan, James; Georgiou, Dimitra K.; Asara, John; Muller, Florian
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SaveAn enolase inhibitor for the targeted treatment of ENO1-deleted cancers (vol 2, pg 1413, 2020)
Lin, Yu-Hsi; Satani, Nikunj; Hammoudi, Naima; Yan, Victoria C.; Barekatain, Yasaman; Khadka, Sunada; Ackroyd, Jeffrey J.; Georgiou, Dimitra K.; Pham, Cong-Dat; Arthur, Kenisha; Maxwell, David; Peng, Zhenghong; Leonard, Paul G.; Czako, Barbara; Pisaneschi, Federica; Mandal, Pijus; Sun, Yuting; Zielinski, Rafal; Pando, Susana Castro; Wang, Xiaobo; Tran, Theresa; Xu, Quanyu; Wu, Qi; Jiang, Yongying; Kang, Zhijun; Asara, John M.; Priebe, Waldemar; Bornmann, William; Marszalek, Joseph R.; DePinho, Ronald A.; Muller, Florian L.
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SaveAn enolase inhibitor for the targeted treatment of ENO1-deleted cancers
Lin, Yu-Hsi; Satani, Nikunj; Hammoudi, Naima; Yan, Victoria C.; Barekatain, Yasaman; Khadka, Sunada; Ackroyd, Jeffrey J.; Georgiou, Dimitra K.; Pham, Cong-Dat; Arthur, Kenisha; Maxwell, David; Peng, Zhenghong; Leonard, Paul G.; Czako, Barbara; Pisaneschi, Federica; Mandal, Pijus; Sun, Yuting; Zielinski, Rafal; Pando, Susana Castro; Wang, Xiaobo; Tran, Theresa; Xu, Quanyu; Wu, Qi; Jiang, Yongying; Kang, Zhijun; Asara, John M.; Priebe, Waldemar; Bornmann, William; Marszalek, Joseph R.; DePinho, Ronald A.; Muller, Florian L.
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SaveBioreducible Phosphonoamidate Pro-drug Inhibitor of Enolase: Proof of Concept Study
Yan, Victoria C.; Yang, Kristine L.; Ballato, Elliot S.; Khadka, Sunada; Shrestha, Prakriti; Arthur, Kenisha; Georgiou, Dimitra K.; Washington, Mykia; Tran, Theresa; Poral, Anton H.; Cong-Dat Pham; Yan, Matthew J.; Muller, Florian L.
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SaveAn In Vivo Screen Identifies PYGO2 as a Driver for Metastatic Prostate Cancer
Lu, Xin; Pan, Xiaolu; Wu, Chang-Jiun; Zhao, Di; Feng, Shan; Zang, Yong; Lee, Rumi; Khadka, Sunada; Amin, Samirkumar B.; Jin, Eun-Jung; Shang, Xiaoying; Deng, Pingna; Luo, Yanting; Morgenlander, William R.; Weinrich, Jacqueline; Lu, Xuemin; Jiang, Shan; Chang, Qing; Navone, Nora M.; Troncoso, Patricia; DePinho, Ronald A.; Wang, Y. Alan
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SaveCollateral lethality: A new target for personalized oncology
Lin, Yu-Hsi; Hammoudi, Naima; Satani, Nikunj; Ackroyd, Jeffrey; Khadka, Sunada; Georgiou, Dimitra; Marszalek, Joe; Sun, Yuting; Protopopova, Marina; Di Francesco, Maria E.; Czako, Barbara; Wang, Alan Y.; DePinho, Ronald A.; Muller, Florian L.
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SaveTargeting YAP-Dependent MDSC Infiltration Impairs Tumor Progression
Wang, Guocan; Lu, Xin; Dey, Prasenjit; Deng, Pingna; Wu, Chia Chin; Jiang, Shan; Fang, Zhuangna; Zhao, Kuo; Konaparthi, Ramakrishna; Hua, Sujun; Zhang, Jianhua; Li-Ning-Tapia, Elsa M.; Kapoor, Avnish; Wu, Chang-Jiun; Patel, Neelay Bhaskar; Guo, Zhenglin; Ramamoorthy, Vandhana; Tieu, Trang N.; Heffernan, Tim; Zhao, Di; Shang, Xiaoying; Khadka, Sunada; Hou, Pingping; Hu, Baoli; Jin, Eun-Jung; Yao, Wantong; Pan, Xiaolu; Ding, Zhihu; Shi, Yanxia; Li, Liren; Chang, Qing; Troncoso, Patricia; Logethetis, Christopher J.; McArthur, Mark J.; Chin, Lynda; Wang, Y. Alan; DePinho, Ronaldo A.
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