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SaveDocking 14 Million Virtual Isoquinuclidines against the μ and κ Opioid Receptors Reveals Dual Antagonists-Inverse Agonists with Reduced Withdrawal Effects
Vigneron, SF; Ohno, S; Braz, J; Kim, JY; Kweon, OS; Webb, C; Billesbolle, CB; Srinivasan, K; Bhardwaj, K; Irwin, JJ; Manglik, A; Basbaum, AI; Ellman, JA; Shoichet, BK
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SaveDefining the structure-activity relationship for a novel class of allosteric MKP5 inhibitors
Gannam, Zira T. K.; Jamali, Haya; Kweon, Oh Sang; Herrington, James; Shillingford, Shanelle R.; Papini, Christina; Gentzel, Erik; Lolis, Elias; Bennett, Anton M.; Ellman, Jonathan A.; Anderson, Karen S.
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