arrow
Back
G

Gabriele Cruciani

University of Perugia

61H-index
353Paper Count
1.4WCitation Count
Published Papers 161
Publication Date
Lipid signature in X-ALD: a comparison between phenotypes
err2026-09-19
err0
errOAAI
errAD Alessandra Di Veroli; SP Sara Petrillo; CT Caterina Torda; FL Federica Loia; TR Teresa Rizza; RC Rosalba Carrozzo; GC Gabriele Cruciani; EB Enrico Bertini; FN Francesco Nicita; FP Fiorella Piemonte; MC Marco Cappa
errShare
errSave
A Polypharmacology-Driven Approach to Alzheimer’s Disease and Tauopathies: Rational Design; Synthesis and Characterization of Amino-Pyrazole-Based Multikinase (GSK-3β/FYN-α/DYRK1A) Inhibitors
err2026-04-29
err0
errOAAI
errStefania Demuro; Debora Russo; Ilaria Penna; Siranuysh Grabska; Hovakim Grabski; Andrea Dalle Vedove; Aurora Valeri; Conall Sauvey; Giuliana Ottonello; Maria Summa; Sine Mandrup Bertozzi; Jose Ortega; Rosalia Bertorelli; Paola Storici; Stefania Girotto; Gabriele Cruciani; Rita M. C. Di Martino; Ruben Abagyan; Andrea Cavalli
errShare
errSave
Discovery of a tetrahydrobenzothiophen-2-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamide-based PROTAC as degrader of SARS-CoV-2 Main Protease
err2026-02-24
err0
errOAAI
errMichela Eleuteri; Alessandro Bazzacco; Beatrice Mercorelli; Jenny Desantis; Alessia Zago; Gabriele Cruciani; Arianna Loregian; Laura Goracci
errShare
errSave
Advancing spatial-omics through Pyxis, vendor-neutral software for ion mobility mass spectrometry imaging data analysis
err2025-12-20
err0
errOAAI
errSara Tortorella; Sebastian Bessler; Giuseppe Arturi; Giulia Sorbi; Jens Soltwisch; Gabriele Cruciani
errShare
errSave
Selection of short Gadd45β-binding peptides through a synergistic computational and biophysical approach
err2025-11-18
err0
errOAAI
errDi Cristofano, Samuele; Iaccarino, Emanuela; Caporale, Andrea; Verzella, Daniela; Falcigno, Lucia; D'Auria, Gabriella; Russo, Rosita; Rega, Camilla; Chambery, Angela; Oliver, Angela; Barisciano, Giovannina; Cross, Simon; Cruciani, Gabriele; Capece, Daria; Zazzeroni, Francesca; Ruvo, Menotti; Sandomenico, Annamaria; Raimondo, Domenico
errShare
errSave
errShare
errSave
Rational optimization of D3R/GSK-3β dual target-directed ligands as potential treatment for bipolar disorder: Design, synthesis, X-ray crystallography, molecular dynamics simulations, in vitro ADME, and in vivo pharmacokinetic studies
err2025-06-25
err0
PREAI
errR.M.C. Di Martino; D. Russo; I. Penna; S. Demuro; A. Dalle Vedove; R. Spagnuolo; G. Ottonello; S.M. Bertozzi; M. Summa; J. Desantis; A. Valeri; L. Pruccoli; S.K. Tripathi; A. Tarozzi; P. Storici; S. Girotto; R. Bertorelli; A. Armirotti; G. Cruciani; T. Bandiera; A. Cavalli; G. Bottegoni
errShare
errSave
Between Theory and Practice: Computational/Experimental Integrated Approaches to Understand the Solubility and Lipophilicity of PROTACs
err2024-09-13
err0
PREAI
errVenturi, Andrea; Di Bona, Stefano; Desantis, Jenny; Eleuteri, Michela; Bartalucci, Matteo; Baroni, Massimo; Benedetti, Paolo; Goracci, Laura; Cruciani, Gabriele
errShare
errSave
Amniotic fluid stem cell-derived extracellular vesicles educate type 2 conventional dendritic cells to rescue autoimmune disorders in a multiple sclerosis mouse model
err2024-06-06
err0
errOAAI
errManni, Giorgia; Gargaro, Marco; Ricciuti, Doriana; Fontana, Simona; Padiglioni, Eleonora; Cipolloni, Marco; Mazza, Tommaso; Rosati, Jessica; di Veroli, Alessandra; Mencarelli, Giulia; Pieroni, Benedetta; Barcelos, Estevao Carlos Silva; Scalisi, Giulia; Sarnari, Francesco; di Michele, Alessandro; Pascucci, Luisa; de Franco, Francesca; Zelante, Teresa; Antognelli, Cinzia; Cruciani, Gabriele; Talesa, Vincenzo Nicola; Romani, Rita; Fallarino, Francesca
errShare
errSave
Identification of small molecules affecting the interaction between human hemoglobin and Staphylococcus aureus IsdB hemophore
err2024-04-09
err0
errOAAI
errCozzi, Monica; Failla, Mariacristina; Gianquinto, Eleonora; Kovachka, Sandra; Comani, Valeria Buoli; Compari, Carlotta; De Bei, Omar; Giaccari, Roberta; Marchesani, Francesco; Marchetti, Marialaura; Ronda, Luca; Rolando, Barbara; Baroni, Massimo; Cruciani, Gabriele; Campanini, Barbara; Bettati, Stefano; Faggiano, Serena; Lazzarato, Loretta; Spyrakis, Francesca
errShare
errSave
Discovery and Structure-Activity Relationships of Novel ssDAF-12 Receptor Modulators
err2024-02-28
err0
PREAI
errCeccarelli, Giada; Goracci, Laura; Carotti, Andrea; Paccoia, Federico; Passeri, Daniela; Cipolloni, Marco; Di Bona, Stefano; Cruciani, Gabriele; Pellicciari, Roberto; Gioiello, Antimo
errShare
errSave
MARS: A Multipurpose Software for Untargeted LC-MS-Based Metabolomics and Exposomics
err2024-01-18
err2
errOAAI
errGoracci, Laura; Tiberi, Paolo; Di Bona, Stefano; Bonciarelli, Stefano; Passeri, Giovanna Ilaria; Piroddi, Marta; Moretti, Simone; Volpi, Claudia; Zamora, Ismael; Cruciani, Gabriele
errShare
errSave
Structure-Based Optimization of 1,2,4-Triazole-3-Thione Derivatives: Improving Inhibition of NDM-/VIM-Type Metallo-β-Lactamases and Synergistic Activity on Resistant Bacteria
err2023-12-02
err2
errOAAI
errBersani, Matteo; Failla, Mariacristina; Vascon, Filippo; Gianquinto, Eleonora; Bertarini, Laura; Baroni, Massimo; Cruciani, Gabriele; Verdirosa, Federica; Sannio, Filomena; Docquier, Jean-Denis; Cendron, Laura; Spyrakis, Francesca; Lazzarato, Loretta; Tondi, Donatella; Lopes, Bruno Silvester; Hanafiah, Alfizah
errShare
errSave
VHL-Modified PROteolysis TArgeting Chimeras (PROTACs) as a Strategy to Evade Metabolic Degradation in In Vitro Applications
err2023-09-12
err3
PREAI
errCastellani, Beatrice; Eleuteri, Michela; Di Bona, Stefano; Cruciani, Gabriele; Desantis, Jenny; Goracci, Laura
errShare
errSave
errShare
errSave
Targeting protein-protein interactions with low molecular weight and short peptide modulators: insights on disease pathways and starting points for drug discovery
err2023-05-29
err8
PREAI
errTrisciuzzi, Daniela; Villoutreix, Bruno O.; Siragusa, Lydia; Baroni, Massimo; Cruciani, Gabriele; Nicolotti, Orazio
errShare
errSave
Growth hormone secretagogues modulate inflammation and fibrosis in mdx mouse model of Duchenne muscular dystrophy
err2023-04-12
err8
errOAAI
errBoccanegra, Brigida; Cappellari, Ornella; Mantuano, Paola; Trisciuzzi, Daniela; Mele, Antonietta; Tulimiero, Lisamaura; De Bellis, Michela; Cirmi, Santa; Sanarica, Francesca; Cerchiara, Alessandro Giovanni; Conte, Elena; Meanti, Ramona; Rizzi, Laura; Bresciani, Elena; Denoyelle, Severine; Fehrentz, Jean-Alain; Cruciani, Gabriele; Nicolotti, Orazio; Liantonio, Antonella; Torsello, Antonio; De Luca, Annamaria
errShare
errSave
Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
err2022-12-07
err6
errOAAI
errCostantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo-Ahen, Outi M. H.; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela; Giovannetti, Elisa; Peters, Godefridus J.; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M.; Wade, Rebecca C.; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola
errShare
errSave
An Integrated Machine Learning Model To Spot Peptide Binding Pockets in 3D Protein Screening
err2022-11-02
err14
PREAI
errTrisciuzzi, Daniela; Siragusa, Lydia; Baroni, Massimo; Cruciani, Gabriele; Nicolotti, Orazio
errShare
errSave
Analytical and computational workflow for in-depth analysis of oxidized complex lipids in blood plasma
err2022-11-01
err25
errOAAI
errCriscuolo, Angela; Nepachalovich, Palina; Garcia-del Rio, Diego Fernando; Lange, Mike; Ni, Zhixu; Baroni, Massimo; Cruciani, Gabriele; Goracci, Laura; Blueher, Matthias; Fedorova, Maria
errShare
errSave