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Christian Gege

innovative molecules gmbh

26H-index
76Paper Count
1.9KCitation Count
Published Papers 32
Publication Date
Carboxylic Acid Bioisosteres Boost Nurr1 Agonist Selectivity
err2025-07-17
err0
errOAAI
errTanja Stiller; Christian Gege; Wael Saeb; Jan Vietor; Úrsula López-García; Romy Busch; Hella Kohlhof; Daniel Vitt; Daniel Merk
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Identification of JNJ-61803534, a RORγt Inverse Agonist for the Treatment of Psoriasis
err2025-04-16
err0
PREAI
errKinzel, Olaf; Goldberg, Steven D.; Cummings, Maxwell D.; Gege, Christian; Steeneck, Christoph; Xue, Xiaohua; Albers, Michael; Schluter, Thomas; Kleymann, Gerald; Scott, Brian; Sepassi, Kia; Schoetens, Freddy; Venkatesan, Hariharan; Tanis, Virginia M.; Coe, Kevin; Sales, Zachary S.; Spurlino, John; Milligan, Cynthia; Fourie, Anne M.; Edwards, James P.; Hoffmann, Thomas
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New developments in celiac disease treatments
err2024-09-01
err4
errOAAI
errBurianek, Franziska; Gege, Christian; Marinkovic, Petar
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Synthesis and Characterization of DHODH Inhibitors Based on the Vidofludimus Scaffold with Pronounced Anti-SARS-CoV-2 Activity
err2024-08-06
err4
errOAAI
errGege, Christian; Hahn, Friedrich; Wangen, Christina; Haege, Sigrun; Herrmann, Alexandra; Uhlig, Nadja; Eberlein, Valentina; Issmail, Leila; Klopfleisch, Robert; Grunwald, Thomas; Marschall, Manfred; Kohlhof, Hella; Vitt, Daniel
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Development of a Potent Nurr1 Agonist Tool for In Vivo Applications
err2023-04-26
err18
errOAAI
errVietor, Jan; Gege, Christian; Stiller, Tanja; Busch, Romy; Schallmayer, Espen; Kohlhof, Hella; Hoefner, Georg; Pabel, Joerg; Marschner, Julian A.; Merk, Daniel
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Interplay of Trans- and Cis-Interactions of Glycolipids in Membrane Adhesion
err2021-11-19
err4
errOAAI
errKav, Batuhan; Deme, Bruno; Gege, Christian; Tanaka, Motomu; Schneck, Emanuel; Weikl, Thomas R.
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A helicase-primase drug candidate with sufficient target tissue exposure affects latent neural herpes simplex virus infections
err2021-06-16
err28
PREAI
errGege, Christian; Bravo, Fernando J.; Uhlig, Nadja; Hagmaier, Timo; Schmachtenberg, Rosanne; Elis, Julia; Burger-Kentischer, Anke; Finkelmeier, Doris; Hamprecht, Klaus; Grunwald, Thomas; Bernstein, David, I; Kleymann, Gerald
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Identification of a potent, orally bioavailable and selective MCT4 Inhibitor for the treatment of solid Warburg tumors
err2019-07-01
err2
PREAI
errHambruch, Nina; Herkert, Barbara; Gege, Christian; Mallinger, Aurelie; Fabian, Johannes; Kinzel, Olaf; Wang, Yansong; Fink, Gero; Albers, Michael; Funk, Anette; Bittman-Waetzig, Annika; Fleckenstein, Tilly; Braun, Floriane; Kremoser, Claus
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How to develop a differentiated FXR agonist: GS-9674 shows a reduced side effect profile in mice, monkeys amd human phase I studies compared to its predecessor Px-102
err2019-04-01
err1
PREAI
errHambruch, Eva; Hollenback, David; Liles, John; Kinzel, Olaf; Birkel, Manfred; Fink, Gero; French, Dorothy; Gege, Christian; Hornberger, Martin; Watkins, William; Kremoser, Claus
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LXR inverse agonists reduce steatosis and fibrosis in the STAM mouse model but also improve insulin sensitivity in a high fat diet mouse clamp study
err2019-04-01
err0
PREAI
errHambruch, Eva; Gege, Christian; Kinzel, Olaf; Hauser, Katharina; Birkel, Manfred; Deuschle, Ulrich; Kremoser, Claus
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LXR inverse agonists inhibit de novo lipogenesis and reduce intestinal lipid and cholesterol absorption in a NAFLD mouse model
err2018-04-01
err0
PREAI
errKremoser, C.; Deuschle, U.; Gege, C.; Kinzel, O.; Krol, H. D.; Albers, M.; Birkel, M.; Hambruch, E.
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