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SaveAnakinra restores immunological misfiring that drives influenza-associated pulmonary aspergillosis
Seldeslachts, Laura; Kraisin, Sirima; Dewi, Intan M. W.; Feys, Simon; Staels, Frederik; Gkountzinopoulou, Marina; Jacobs, Cato; Tielemans, Birger; Vanhoffelen, Eliane; Resendiz-Sharpe, Agustin; De Herdt, Lander; Kwan, Oswin; Vandamme, Niels; Roels, Jana; Neumann, Julika; Prezzemolo, Teresa; Malengier-Devlies, Bert; Stroobants, Mathias; Carvalho, Agostinho; Matthys, Patrick; Naesens, Lieve; Lagrou, Katrien; Khan, Mona; Mombaerts, Peter; Verbeken, Erik; Martinod, Kimberly; Wauters, Joost; van de Veerdonk, Frank L.; Vande Velde, Greetje; Humblet-Baron, Stephanie
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SaveTrypstatin as a Novel TMPRSS2 Inhibitor with Broad-Spectrum Efficacy against Corona and Influenza Viruses
Lawrenz, J; Wettstein, L; Alfonso, AR; Nchioua, R; von Maltitz, P; Albers, DPJ; Zech, F; Vandeput, J; Naesens, L; Fois, G; Neubauer, V; Preising, N; Schmierer, E; Almeida-Hernandez, Y; Petersen, M; Staendker, L; Wiese, S; Braubach, P; Frick, M; Barth, E; Sauter, D; Kirchhoff, F; Sanchez-Garcia, E; Stevaert, A; Muench, J
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SaveA guanidine-based coronavirus replication inhibitor which targets the nsp15 endoribonuclease and selects for interferon-susceptible mutant viruses
Van Loy, Benjamin; Pujol, Eugenia; Kamata, Kenichi; Lee, Xiao Yin; Bakirtzoglou, Nikolai; Van Berwaer, Ria; Vandeput, Julie; Mestdagh, Cato; Persoons, Leentje; De Wijngaert, Brent; Goovaerts, Quinten; Noppen, Sam; Jacquemyn, Maarten; Ahmadzadeh, Kourosh; Bernaerts, Eline; Martin-Lopez, Juan; Escriche, Celia; Vanmechelen, Bert; Krasniqi, Besir; Singh, Abhimanyu K.; Daelemans, Dirk; Maes, Piet; Matthys, Patrick; Dehaen, Wim; Rozenski, Jef; Das, Kalyan; Voet, Arnout; Vazquez, Santiago; Naesens, Lieve; Stevaert, Annelies
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SaveExploration of isatin-based inhibitors of SARS-CoV-2 Nsp15 endoribonuclease
Rampias, Theodoros; Antoniou, Thomas; Stevaert, Annelies; Kravaritid, Lara; Van Loy, Benjamin; Vandeput, Julie; Sgrignani, Jacopo; Filippidou, Natalia; Locatelli, Patrizia; Samiotaki, Martina; Tzakos, Eleftherios Paraskevas; Cavalli, Andrea; Naesens, Lieve; Sideris, Diamantis C.; Tzakos, Andreas G.
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SaveDamping excessive viral-induced IFN-γ rescues the impaired anti-Aspergillus host immune response in influenza-associated pulmonary aspergillosis
Seldeslachts, Laura; Staels, Frederik; Gkountzinopoulou, Marina; Jacobs, Cato; Tielemans, Birger; Vanhoffelen, Eliane; Resendiz-Sharpe, Agustin; De Herdt, Lander; Haughton, Jeason; Prezzemolo, Teresa; Burton, Oliver; Feys, Simon; van de Veerdonk, Frank L.; Carvalho, Agostinho; Naesens, Lieve; Matthys, Patrick; Lagrou, Katrien; Verbeken, Erik; Chamilos, Georgios; Wauters, Joost; Humblet-Baron, Stephanie; Vande Velde, Greetje
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SaveNovel pentafluorosulfanyl-containing triclocarban analogs selectively kill Gram-positive bacteria
Pormohammad, Ali; Moradi, Melika; Hommes, Josefien W.; Pujol, Eugenia; Naesens, Lieve; Vazquez, Santiago; Surewaard, Bas G. J.; Zarei, Mohammad; Vazquez-Carrera, Manuel; Turner, Raymond J.
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SaveSemisynthetic teicoplanin derivatives with dual antimicrobial activity against SARS-CoV-2 and multiresistant bacteria
Bereczki, Ilona; Vimberg, Vladimir; Lorincz, Eszter; Papp, Henrietta; Nagy, Lajos; Keki, Sandor; Batta, Gyula; Mitrovic, Ana; Kos, Janko; Zsigmond, Aron; Hajdu, Istvan; Lorincz, Zsolt; Bajusz, David; Petri, Laszlo; Hodek, Jan; Jakab, Ferenc; Keseru, Gyorgy M.; Weber, Jan; Naesens, Lieve; Herczegh, Pal; Borbas, Aniko
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SaveA Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In Vitro
De Castro, Sonia; Stevaert, Annelies; Maldonado, Miguel; Delpal, Adrien; Vandeput, Julie; Van Loy, Benjamin; Eydoux, Cecilia; Guillemot, Jean-Claude; Decroly, Etienne; Gago, Federico; Canard, Bruno; Camarasa, Maria-Jose; Velazquez, Sonsoles; Naesens, Lieve
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SaveFunctional Analysis of Human and Feline Coronavirus Cross-Reactive Antibodies Directed Against the SARS-CoV-2 Fusion Peptide
Vanderheijden, Nathalie; Stevaert, Annelies; Xie, Jiexiong; Ren, Xiaolei; Barbezange, Cyril; Noppen, Sam; Desombere, Isabelle; Verhasselt, Bruno; Geldhof, Peter; Vereecke, Nick; Stroobants, Veerle; Oh, Dayoung; Vanhee, Merijn; Naesens, Lieve M. J.; Nauwynck, Hans J.
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