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Dipeptidic Phosphonates: Potent Inhibitors of Pseudomonas aeruginosa Elastase B Showing Efficacy in a Murine Keratitis Model Kiefer, AF; Schütz, C; Englisch, CN; Kolling, D; Speicher, S; Kany, AM; Shafiei, R; Wadood, NA; Aljohmani, A; Wirschem, N; Jumde, RP; Klein, A; Sikandar, A; Park, YM; Krasteva-Christ, G; Yildiz, D; Abdelsamie, AS; Rox, K; Köhnke, J; Müller, R; Bischoff, M; Haupenthal, J; Hirsch, AKH Share Save
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Development of Fragment-Based Inhibitors of the Bacterial Deacetylase LpxC with Low Nanomolar Activity Mielniczuk, Sebastian; Hoff, Katharina; Baselious, Fady; Li, Yunqi; Haupenthal, Joerg; Kany, Andreas M.; Riedner, Maria; Rohde, Holger; Rox, Katharina; Hirsch, Anna K. H.; Krimm, Isabelle; Sippl, Wolfgang; Holl, Ralph Share Save
Target-Directed Dynamic Combinatorial Chemistry Affords Binders of Mycobacterium tuberculosis IspE Braun-Cornejo, Maria; Ornago, Camilla; Sonawane, Vidhisha; Haupenthal, Joerg; Kany, Andreas M.; Diamanti, Eleonora; Jezequel, Gwenaelle; Reiling, Norbert; Blankenfeldt, Wulf; Maas, Peter; Hirsch, Anna K. H. Share Save
Dual inhibitors of Pseudomonas aeruginosa virulence factors LecA and LasB Metelkina, Olga; Konstantinovic, Jelena; Klein, Andreas; Shafiei, Roya; Fares, Mario; Alhayek, Alaa; Yahiaoui, Samir; Elgaher, Walid A. M.; Haupenthal, Joerg; Titz, Alexander; Hirsch, Anna K. H. Share Save
Clean Synthetic Strategies to Biologically Active Molecules from Lignin: A Green Path to Drug Discovery Afanasenko, Anastasiia M.; Wu, Xianyuan; De Santi, Alessandra; Elgaher, Walid A. M.; Kany, Andreas M.; Shafiei, Roya; Schulze, Marie-Sophie; Schulz, Thomas F.; Haupenthal, Joerg; Hirsch, Anna K. H.; Barta, Katalin Share Save
Inhibitors of the Elastase LasB for the Treatment of Pseudomonas aeruginosa Lung Infections Konstantinovic, Jelena; Kany, Andreas M.; Alhayek, Alaa; Abdelsamie, Ahmed S.; Sikandar, Asfandyar; Voos, Katrin; Yao, Yiwen; Andreas, Anastasia; Shafiei, Roya; Loretz, Brigitta; Schoenauer, Esther; Bals, Robert; Brandstetter, Hans; Hartmann, Rolf W.; Ducho, Christian; Lehr, Claus-Michael; Beisswenger, Christoph; Mueller, Rolf; Rox, Katharina; Haupenthal, Joerg; Hirsch, Anna K. H. Share Save
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors Ropponen, Henni-Karoliina; Diamanti, Eleonora; Johannsen, Sandra; Illarionov, Boris; Hamid, Rawia; Jaki, Miriam; Sass, Peter; Fischer, Markus; Haupenthal, Joerg; Hirsch, Anna K. H. Share Save
Not Every Hit-Identification Technique Works on 1-Deoxy-d-Xylulose 5-Phosphate Synthase (DXPS): Making the Most of a Virtual Screening Campaign Johannsen, Sandra; Gierse, Robin M.; Olshanova, Aleksandra; Smerznak, Ellie; Laggner, Christian; Eschweiler, Lea; Adeli, Zahra; Hamid, Rawia; Alhayek, Alaa; Reiling, Norbert; Haupenthal, Joerg; Hirsch, Anna K. H. Share Save
Discovery and Characterization of Synthesized and FDA-Approved Inhibitors of Clostridial and Bacillary Collagenases Alhayek, Alaa; Abdelsamie, Ahmed S.; Schoenauer, Esther; Camberlein, Virgyl; Hutterer, Evelyn; Posselt, Gernot; Serwanja, Jamil; Bloechl, Constantin; Huber, Christian G.; Haupenthal, Jorg; Brandstetter, Hans; Wessler, Silja; Hirsch, Anna K. H. Share Save
Discovery of the First Selective Nanomolar Inhibitors of ERAP2 by Kinetic Target-Guided Synthesis Camberlein, Virgyl; Fleau, Charlotte; Sierocki, Pierre; Li, Lenong; Gealageas, Ronan; Bosc, Damien; Guillaume, Valentin; Warenghem, Sandrine; Leroux, Florence; Rosell, Melissa; Cheng, Keguang; Medve, Laura; Prigent, Mathilde; Decanter, Myriam; Piveteau, Catherine; Biela, Alexandre; Eveque, Maxime; Dumont, Julie; Mpakali, Anastasia; Giastas, Petros; Herledan, Adrien; Couturier, Cyril; Haupenthal, Joerg; Lesire, Laetitia; Hirsch, Anna K. H.; Deprez, Benoit; Stratikos, Efstratios; Bouvier, Marlene; Deprez-Poulain, Rebecca Share Save
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Structure-Based Design of α-Substituted Mercaptoacetamides as Inhibitors of the Virulence Factor LasB from Pseudomonas aeruginosa Kaya, Cansu; Walter, Isabell; Alhayek, Alaa; Shafiei, Roya; Jezequel, Gwenaelle; Andreas, Anastasia; Konstantinovic, Jelena; Schoenauer, Esther; Sikandar, Asfandyar; Haupenthal, Joerg; Mueller, Rolf; Brandstetter, Hans; Hartmann, Rolf W.; Hirsch, Anna K. H. Share Save
N-Aryl Mercaptopropionamides as Broad-Spectrum Inhibitors of Metallo-β-Lactamases Kaya, Cansu; Konstantinovic, Jelena; Kany, Andreas M.; Andreas, Anastasia; Kramer, Jan S.; Brunst, Steffen; Weizel, Lilia; Rotter, Marco J.; Frank, Denia; Yahiaoui, Samir; Mueller, Rolf; Hartmann, Rolf W.; Haupenthal, Joerg; Proschak, Ewgenij; Wichelhaus, Thomas A.; Hirsch, Anna K. H. Share Save
Inhibition of Collagenase Q1 of Bacillus cereus as a Novel Antivirulence Strategy for the Treatment of Skin-Wound Infections Alhayek, Alaa; Khan, Essak S.; Schoenauer, Esther; Daeinghaus, Tobias; Shafiei, Roya; Voos, Katrin; Han, Mitchell K. L.; Ducho, Christian; Posselt, Gernot; Wessler, Silja; Brandstetter, Hans; Haupenthal, Joerg; del Campo, Aranzazu; Hirsch, Anna K. H. Share Save
Discovery of novel drug-like antitubercular hits targeting the MEP pathway enzyme DXPS by strategic application of ligand-based virtual screening Zhu, Di; Johannsen, Sandra; Masini, Tiziana; Simonin, Celine; Haupenthal, Jorg; Illarionov, Boris; Andreas, Anastasia; Awale, Mahendra; Gierse, Robin M.; van der Laan, Tridia; van der Vlag, Ramon; Nasti, Rita; Poizat, Mael; Buhler, Eric; Reiling, Norbert; Mueller, Rolf; Fischer, Markus; Reymond, Jean-Louis; Hirsch, Anna K. H. Share Save
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