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Kaoru Kobayashi

Meiji Pharmaceutical University

93H-index
717Paper Count
3.2WCitation Count
Published Papers 153
Publication Date
CYP3A5 polymorphism affects the disposition of tacrolimus and its metabolite in systemic circulation and peripheral tissues of mice introduced with the CYP3A5 gene
err2026-05-08
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errOAAI
errGenki Minegishi; Yuna Hiramatsu; Manami Sugahara; Satoshi Abe; Kanako Kazuki; Atsushi Miyajima; Yasuhiro Kazuki; Kaoru Kobayashi
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Characterization of fatty acid amide hydrolase 2 as a drug-metabolizing enzyme: Contribution to the hydrolysis of DS-8500a and its analogues
err2026-02-09
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PREAI
errChie Makino; Takuma Chiashi; Mayumi Hayashi; Yuji Ogura; Hidenori Namiki; Tomoyo Honda; Akiko Watanabe; Hideyuki Shiozawa; Hideo Takakusa; Daisuke Nakai; Kaoru Kobayashi
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Double-humanized Rats for CYP3A and PXR as an Improved Model for Analyzing Drug-drug Interactions Mediated by CYP3A4
err2025-07-28
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PREAI
errKaoru Kobayashi; Genki Minegishi; Kanako Kazuki; Satoshi Abe; Miyuki Sato; Atsushi Miyajima; Masumi Hirabayashi; Tetsushi Sakuma; Takashi Yamamoto; Yasuhiro Kazuki
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Contribution of Japanese scientists to drug metabolism and disposition
err2025-05-01
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PREAI
errNakajima, Miki; Yamazaki, Hiroshi; Yoshinari, Kouichi; Kobayashi, Kaoru; Ishii, Yuji; Nakai, Daisuke; Kamimura, Hidetaka; Kume, Toshiyuki; Saito, Yoshiro; Maeda, Kazuya; Kusuhara, Hiroyuki; Tamai, Ikumi
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Hepatic arterial infusion of autologous CD34+cells for hepatitis C virus-related decompensated cirrhosis: A multicenter, open-label, exploratory randomized controlled trial
err2024-12-01
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errOAAI
errNakamura, Toru; Masuda, Atsutaka; Kako, Makoto; Enomoto, Hirayuki; Kaibori, Masaki; Fujita, Yasuyuki; Tanizawa, Kyoko; Ioji, Tetsuya; Fujimori, Yoshihiro; Fukami, Kei; Hazama, Takuma; Iwamoto, Hideki; Kako, Yasukazu; Kobayashi, Kaoru; Koga, Hironori; Nagafuji, Koji; Ohtake, Takayasu; Suzuki, Hiroyuki; Takashima, Tomoyuki; Tsukiyama, Toshitaka; Uojima, Haruki; Yamahara, Kenichi; Yamakado, Koichiro; Yamamoto, Hidekazu; Yoh, Kazunori; Yoshihara, Satoshi; Kawamoto, Atsuhiko; Nishiguchi, Shuhei; Kobayashi, Shuzo; Torimura, Takuji; Kawaguchi, Takumi
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A small molecule iCDM-34 identified by in silico screening suppresses HBV DNA through activation of aryl hydrocarbon receptor
err2023-12-22
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errOAAI
errFurutani, Yutaka; Hirano, Yoshinori; Toguchi, Mariko; Higuchi, Shoko; Qin, Xian-Yang; Yanaka, Kaori; Sato-Shiozaki, Yumi; Takahashi, Nobuaki; Sakai, Marina; Kongpracha, Pornparn; Suzuki, Takehiro; Dohmae, Naoshi; Kukimoto-Niino, Mutsuko; Shirouzu, Mikako; Nagamori, Shushi; Suzuki, Harukazu; Kobayashi, Kaoru; Masaki, Takahiro; Koyama, Hiroo; Sekiba, Kazuma; Otsuka, Motoyuki; Koike, Kazuhiko; Kohara, Michinori; Kojima, Soichi; Kakeya, Hideaki; Matsuura, Tomokazu
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ncBAF enhances PXR-mediated transcriptional activation in the human and mouse liver
err2023-09-01
err2
errOAAI
errKurosawa, Kiamu; Nakano, Masataka; Yokoseki, Itsuki; Nagaoka, Mai; Takemoto, Seiya; Sakai, Yoshiyuki; Kobayashi, Kaoru; Kazuki, Yasuhiro; Fukami, Tatsuki; Nakajima, Miki
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Quantitative prediction of P-glycoprotein-mediated drug-drug interactions and intestinal absorption using humanized mice
err2021-09-06
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errOAAI
errMiyake, Taiji; Tsutsui, Haruka; Haraya, Kenta; Tachibana, Tatsuhiko; Morimoto, Kayoko; Takehara, Shoko; Ayabe, Miho; Kobayashi, Kaoru; Kazuki, Yasuhiro
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Nuclear receptor phosphorylation in xenobiotic signal transduction
err2020-11-01
err40
errOAAI
errNegishi, Masahiko; Kobayashi, Kaoru; Sakuma, Tsutomu; Sueyoshi, Tatsuya
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Development of Caco-2 cells expressing four CYPs via a mammalian artificial chromosome
err2020-08-20
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errOAAI
errOhta, Yumi; Kazuki, Kanako; Abe, Satoshi; Oshimura, Mitsuo; Kobayashi, Kaoru; Kazuki, Yasuhiro
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CYP3A4 Induction in the Liver and Intestine of Pregnane X Receptor/CYP3A-Humanized Mice: Approaches by Mass Spectrometry Imaging and Portal Blood Analysis
err2019-11-01
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errOAAI
errKobayashi, Kaoru; Kuze, Jiro; Abe, Satoshi; Takehara, Shoko; Minegishi, Genki; Igarashi, Katsuhide; Kitajima, Satoshi; Kanno, Jun; Yamamoto, Takushi; Oshimura, Mitsuo; Kazuki, Yasuhiro
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Indirect activation of constitutive androstane receptor in three-dimensionally cultured HepG2 cells
err2019-10-01
err8
PREAI
errYokobori, Kosuke; Azuma, Ikuko; Chiba, Kan; Akita, Hidetaka; Furihata, Tomomi; Kobayashi, Kaoru
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Humanized UGT2 and CYP3A transchromosomic rats for improved prediction of human drug metabolism
err2019-02-04
err27
errOAAI
errKazuki, Yasuhiro; Kobayashi, Kaoru; Hirabayashi, Masumi; Abe, Satoshi; Kajitani, Naoyo; Kazuki, Kanako; Takehara, Shoko; Takiguchi, Masato; Satoh, Daisuke; Kuze, Jiro; Sakuma, Tetsushi; Kaneko, Takehito; Mashimo, Tomoji; Osamura, Minori; Hashimoto, Mari; Wakatsuki, Riko; Hirashima, Rika; Fujiwara, Ryoichi; Deguchi, Tsuneo; Kurihara, Atsushi; Tsukazaki, Yasuko; Senda, Naoto; Yamamoto, Takashi; Scheer, Nico; Oshimura, Mitsuo
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Dynamic Kinetic Resolution of N-Protected Amino Acid Esters via Phase-Transfer Catalytic Base Hydrolysis
err2018-05-21
err18
PREAI
errYamamoto, Eiji; Wakafuji, Kodai; Furutachi, Yuho; Kobayashi, Kaoru; Kamachi, Takashi; Tokunaga, Makoto
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Modification of single-nucleotide polymorphism in a fully humanized CYP3A mouse by genome editing technology
err2017-11-09
err27
errOAAI
errAbe, Satoshi; Kobayashi, Kaoru; Oji, Asami; Sakuma, Tetsushi; Kazuki, Kanako; Takehara, Shoko; Nakamura, Kazuomi; Okada, Azusa; Tsukazaki, Yasuko; Senda, Naoto; Honma, Kazuhisa; Yamamoto, Takashi; Ikawa, Masahito; Chiba, Kan; Oshimura, Mitsuo; Kazuki, Yasuhiro
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Balloon-occluded retrograde transvenous obliteration of varices: focusing on the portal hemodynamics and the recent techniques
err2017-09-05
err13
PREAI
errHirota, Shozo; Kobayashi, Kaoru; Kako, Yasukazu; Takaki, Haruyuki; Yamakado, Koichiro
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Biochemical Markers Reflecting Thyroid Function in Athyreotic Patients on Levothyroxine Monotherapy
errTHYROID
IF6.7
err2017-04-01
err65
errOAAI
errIto, Mitsuru; Miyauchi, Akira; Hisakado, Mako; Yoshioka, Waka; Ide, Akane; Kudo, Takumi; Nishihara, Eijun; Kihara, Minoru; Ito, Yasuhiro; Kobayashi, Kaoru; Miya, Akihiro; Fukata, Shuji; Nishikawa, Mitsushige; Nakamura, Hirotoshi; Amino, Nobuyuki
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