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SavePresynaptic and Postsynaptic Mesolimbic Dopamine D3 Receptors Play Distinct Roles in Cocaine Versus Opioid Reward in Mice
Xi, Zheng-Xiong; Bocarsly, Miriam E.; Galaj, Ewa; Hempel, Briana; Teresi, Catherine; Shaw, Marlisa; Bi, Guo-Hua; Jordan, Chloe; Linz, Emily; Alton, Hannah; Tanda, Gianluigi; Freyberg, Zachary; Alvarez, Veronica A.; Newman, Amy Hauck
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SaveAM6527, a neutral CB1 receptor antagonist, suppresses opioid taking and seeking, as well as cocaine seeking in rodents without aversive effects
Soler-Cedeno, Omar; Alton, Hannah; Bi, Guo-Hua; Linz, Emily; Ji, Lipin; Makriyannis, Alexandros; Xi, Zheng-Xiong
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SaveModifications to 1-(4-(2-Bis(4-fluorophenyl)methyl)sulfinyl)alkyl Alicyclic Amines That Improve Metabolic Stability and Retain an Atypical DAT Inhibitor Profile
Okorom, Amarachi V.; Camacho-Hernandez, Gisela Andrea; Salomon, Kristine; Lee, Kuo Hao; Ku, Therese C.; Cao, Jianjing; Won, Sung Joon; Friedman, Jacob; Lam, Jenny; Paule, James; Rais, Rana; Klein, Benjamin; Xi, Zheng-Xiong; Shi, Lei; Loland, Claus J.; Newman, Amy Hauck
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SaveDopamine D3/D2 Receptor Ligands Based on Cariprazine for the Treatment of Psychostimulant Use Disorders That May Be Dual Diagnosed with Affective Disorders
Gogarnoiu, Emma S.; Vogt, Caleb D.; Sanchez, Julie; Bonifazi, Alessandro; Saab, Elizabeth; Shaik, Anver Basha; Soler-Cedeno, Omar; Bi, Guo-Hua; Klein, Benjamin; Xi, Zheng-Xiong; Lane, J. Robert; Newman, Amy Hauck
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SavePharmacological targeting of G protein-coupled receptor heteromers
Moreno, Estefania; Casajuana-Martin, Nil; Coyle, Michael; Campos, Baruc Campos; Galaj, Ewa; del Torrent, Claudia Llinas; Seyedian, Arta; Rea, William; Cai, Ning-Sheng; Bonifazi, Alessandro; Floran, Benjamin; Xi, Zheng-Xiong; Guitart, Xavier; Casado, Vicent; Newman, Amy H.; Bishop, Christopher; Pardo, Leonardo; Ferre, Sergi
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SaveA red nucleus-VTA glutamate pathway underlies exercise reward and the therapeutic effect of exercise on cocaine use
He, Yi; Madeo, Graziella; Liang, Ying; Zhang, Cindy; Hempel, Briana; Liu, Xiaojie; Mu, Lianwei; Liu, Shui; Bi, Guo-Hua; Galaj, Ewa; Zhang, Hai-Ying; Shen, Hui; McDevitt, Ross A.; Gardner, Eliot L.; Liu, Qing-Song; Xi, Zheng-Xiong
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SaveA highly D3R-selective and efficacious partial agonist (S)-ABS01-113 compared to its D3R-selective antagonist enantiomer (R)-ABS01-113 as potential treatments for opioid use disorder
Galaj, Ewa; Bi, Guo-Hua; Klein, Benjamin; Hempel, Briana; Shaik, Anver Basha; Gogarnoiu, Emma S.; Friedman, Jacob; Lam, Jenny; Rais, Rana; Reed, John F.; Bloom, Shelley H.; Swanson, Tracy L.; Schmachtenberg, Jennifer L.; Eshleman, Amy J.; Janowsky, Aaron; Xi, Zheng-Xiong; Newman, Amy Hauck
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SaveTherapeutic potential of PIMSR, a novel CB1 receptor neutral antagonist, for cocaine use disorder: evidence from preclinical research
Galaj, Ewa; Hempel, Briana; Moore, Allamar; Klein, Benjamin; Bi, Guo-Hua; Gardner, Eliot L.; Seltzman, Herbert H.; Xi, Zheng-Xiong
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SaveInvolvement of the ghrelin system in the maintenance of oxycodone self-administration: converging evidence from endocrine, pharmacologic and transgenic approaches
You, Zhi-Bing; Gardner, Eliot L.; Galaj, Ewa; Moore, Allamar R.; Buck, Tristram; Jordan, Chloe J.; Humburg, Bree A.; Bi, Guo-Hua; Xi, Zheng-Xiong; Leggio, Lorenzo
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SaveInvolvement of the ghrelin system in the maintenance and reinstatement of cocaine-motivated behaviors: a role of adrenergic action at peripheral β1 receptors
You, Zhi-Bing; Galaj, Ewa; Alen, Francisco; Wang, Bin; Bi, Guo-Hua; Moore, Allamar R.; Buck, Tristram; Crissman, Madeline; Pari, Sruti; Xi, Zheng-Xiong; Leggio, Lorenzo; Wise, Roy A.; Gardner, Eliot L.
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