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SaveIntegrative Multi-Omics Approaches Reveal Selectivity Profiles and Molecular Mechanisms of FIIN-2, a Covalent FGFR Inhibitor
Fu, Y; Zhu, DD; Chen, XJ; Qu, LZ; Guo, M; Zhang, SH; Xu, GY; Chen, ZC; Li, MY; Chen, YH
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Savepaper Design, synthesis and biological evaluation of 5-amino-1 H-pyrazole-4-carboxamide derivatives as pan-FGFR covalent inhibitors
Deng, Wuqing; Chen, Xiaojuan; Liang, Hong; Song, Xiaojuan; Xiang, Shuang; Guo, Jing; Tu, Zhengchao; Zhou, Yang; Chen, Yongheng; Lu, Xiaoyun
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SaveTGF-β1 mediates hypoxia-preconditioned olfactory mucosa mesenchymal stem cells improved neural functional recovery in Parkinson's disease models and patients
Zhuo, Yi; Li, Wen-Shui; Lu, Wen; Li, Xuan; Ge, Li-Te; Huang, Yan; Gao, Qing-Tao; Deng, Yu-Jia; Jiang, Xin-Chen; Lan, Zi-Wei; Deng, Que; Chen, Yong-Heng; Xiao, Yi; Lu, Shuo; Jiang, Feng; Liu, Zuo; Hu, Li; Liu, Yu; Ding, Yu; He, Zheng-Wen; Tan, De-An; Duan, Da; Lu, Ming
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SaveCurcumin-primed olfactory mucosa-derived mesenchymal stem cells mitigate cerebral ischemia/reperfusion injury-induced neuronal PANoptosis by modulating microglial polarization
Lan, Ziwei; Tan, Fengbo; He, Jialin; Liu, Jianyang; Lu, Ming; Hu, Zhiping; Zhuo, Yi; Liu, JunJiang; Tang, Xiangqi; Jiang, Zheng; Lian, Aojie; Chen, Yongheng; Huang, Yan
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SaveMafG/MYH9-LCN2 axis promotes liver fibrosis through inhibiting ferroptosis of hepatic stellate cells
Deng, Yalan; Lu, Liqing; Zhu, Dandan; Zhang, Huajun; Fu, Ying; Tan, Yuying; Tan, Xuemei; Guo, Ming; Zhang, Ye; Yang, Heping; Yang, Bing; Liu, Ting; Chen, Yongheng
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SaveDesign, synthesis, and biological evaluation of selective covalent inhibitors of FGFR4
Chen, Xiaojuan; Li, Huiliang; Lin, Qianmeng; Dai, Shuyan; Qu, Lingzhi; Guo, Ming; Zhang, Lin; Liao, Jiaxuan; Wei, Hudie; Xu, Guangyu; Jiang, Longying; Chen, Yongheng
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SaveDiscovery of 6-Formylpyridyl Urea Derivatives as Potent Reversible-Covalent Fibroblast Growth Factor Receptor 4 Inhibitors with Improved Anti-Hepatocellular Carcinoma Activity
Yang, Fang; Lin, Qianmeng; Song, Xiaojuan; Huang, Huisi; Chen, Xiaojuan; Tan, Jianwen; Li, Yun; Zhou, Yang; Tu, Zhengchao; Du, Hongli; Zhang, Zhi-min; Ortega, Raquel; Lin, Xiaojing; Patterson, Adam V.; Smaill, Jeff B.; Chen, Yongheng; Lu, Xiaoyun
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SaveStructural insights into the HDAC4-MEF2A-DNA complex and its implication in long-range transcriptional regulation
Dai, Shuyan; Guo, Liang; Dey, Raja; Guo, Ming; Zhang, Xiangqian; Bates, Darren; Cayford, Justin; Jiang, Longying; Wei, Hudie; Chen, Zhuchu; Zhang, Ye; Chen, Lin; Chen, Yongheng
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