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SaveNatural and synthetic 2-oxoglutarate derivatives are substrates for oncogenic variants of human isocitrate dehydrogenase 1 and 2
Liu, Xiao; Reinbold, Raphael; Liu, Shuang; Herold, Ryan A.; Rabe, Patrick; Duclos, Stephanie; Yadav, Rahul B.; Abboud, Martine I.; Thieffine, Sandrine; Armstrong, Fraser A.; Brewitz, Lennart; Schofield, Christopher J.
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SaveResistance to the isocitrate dehydrogenase 1 mutant inhibitor ivosidenib can be overcome by alternative dimer-interface binding inhibitors
Reinbold, Raphael; Hvinden, Ingvild C.; Rabe, Patrick; Herold, Ryan A.; Finch, Alina; Wood, James; Morgan, Melissa; Staudt, Maximillian; Clifton, Ian J.; Armstrong, Fraser A.; McCullagh, James S. O.; Redmond, Jo; Bardella, Chiara; Abboud, Martine, I; Schofield, Christopher J.
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