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Luc Brunsveld

Eindhoven University of Technology

63H-index
330Paper Count
1.8WCitation Count
Published Papers 155
Publication Date
Induced ubiquitination of the partially disordered estrogen receptor alpha via a 14-3-3 directed molecular glue-PROTAC
err2026-07-15
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errCarlo J. A. Verhoef; Charlotte Crowe; Mark A. Nakasone; Aitana DeLaCuadra-Basté; Tessa Harzing; Naomi A. S. Span; Gajanan Sathe; Laura C. Demmers; Kentaro Iso; Christian Ottmann; Luc Brunsveld; Alessio Ciulli; Peter J. Cossar
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Modulation of the 14-3-3σ/C-RAF “Auto”inhibited Complex by Molecular Glues
err2026-01-30
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errMarkella Konstantinidou; Holly R. Vickery; Marloes A. M. Pennings; Johanna M. Virta; Shu Yue Luo; Emira J. Visser; Sean D. Bannier; Mrudula Srikanth; Sabine Z. Cismoski; Lucy C. Young; Maxime C. M. van den Oetelaar; Frank McCormick; Christian Ottmann; Luc Brunsveld; Michelle R. Arkin
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Macrocyclic Molecular Glues for the 14-3-3/ChREBP Interaction: Affinity and Cooperativity in an Inverse Relationship
err2025-12-01
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errPennings, Marloes A. M.; van den Bosch, Merel A. W.; Oberheide, Ansgar; Verhoef, Carlo J. A.; Ottmann, Christian; Markvoort, Albert J.; Miley, Galen P.; Brunsveld, Luc
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Automated navigation of condensate phase behavior with active machine learning
err2025-10-30
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errYannick H. A. Leurs; Willem van den Hout; Andrea Gardin; Joost L. J. van Dongen; Andoni Rodriguez-Abetxuko; Nadia A. Erkamp; Jan C. M. van Hest; Francesca Grisoni; Luc Brunsveld
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Identifying 14-3-3 interactome binding sites with deep learning
err2025-08-08
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errLaura D van Weesep; Riza Ozcelik; Marloes Pennings; Emanuele Criscuolo; Christian Ottmann; Luc Brunsveld; Francesca Grisoni
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Stoichiometric 14-3-3ζ binding promotes phospho-Tau microtubule dissociation and reduces aggregation and condensation
err2025-07-31
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errJanine Hochmair; Maxime C. M. van den Oetelaar; Leandre Ravatt; Lisa Diez; Lenne J. M. Lemmens; Renata Ponce-Lina; Rithika Sankar; Maximilian Franck; Gesa Nolte; Ekaterina Semenova; Satabdee Mohapatra; Christian Ottmann; Luc Brunsveld; Susanne Wegmann
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Scaffold-hopping for molecular glues targeting the 14-3-3/ERα complex
err2025-07-14
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errMarkella Konstantinidou; Marios Zingiridis; Marloes A. M. Pennings; Michael Fragkiadakis; Johanna M. Virta; Jezrael L. Revalde; Emira J. Visser; Christian Ottmann; Luc Brunsveld; Constantinos G. Neochoritis; Michelle R. Arkin
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The three body solution: Structural insights into molecular glues
err2025-04-01
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errTomlinson, Aidan C. A.; Knox, John E.; Brunsveld, Luc; Ottmann, Christian; Yano, Jason K.
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Site-specific molecular glues for the 14-3-3/Tau pS214 protein-protein interaction via reversible covalent imine tethering
err2025-01-01
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errOberheide, Ansgar; van den Oetelaar, Maxime C. M.; Scheele, Jakob J. A.; Borggraefe, Jan; Engelen, Semmy F. H.; Sattler, Michael; Ottmann, Christian; Cossar, Peter J.; Brunsveld, Luc
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Immunoaffinity Intact Top-Down Mass Spectrometry for Quantification of Neuron-Specific Enolase Gamma, a Low-Abundance Protein Biomarker
err2024-12-23
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errvan den Wildenberg, Sebastian A. H.; Genet, Sylvia A. A. M.; Broeren, Maarten A. C.; van Dongen, Joost L. J.; van den Oetelaar, Maxime C. M.; Brunsveld, Luc; Scharnhorst, Volkher; van de Kerkhof, Daan
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Partial protein binding of uracil and thymine affects accurate dihydropyrimidine dehydrogenase (DPD) phenotyping
err2024-10-01
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errvan den Wildenberg, Sebastian A. H.; Genet, Sylvia A. A. M.; Streng, Alexander S.; Broeren, Maarten A. C.; Deenen, Maarten J.; van Dongen, Joost L. J.; Brunsveld, Luc; Scharnhorst, Volkher; van de Kerkhof, Daan
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Spatiotemporal Control Over Protein Release from Artificial Cells via a Light-Activatable Protease
err2024-09-27
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errNikroo, Arjan Hazegh; Altenburg, Wiggert J.; van Veldhuisen, Thijs W.; Brunsveld, Luc; van Hest, Jan C. M.
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Immunoaffinity Intact-Mass Spectrometry for the Detection of Endogenous Concentrations of the Acetylated Protein Tumor Biomarker Neuron Specific Enolase
err2024-07-16
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errvan den Wildenberg, Sebastian A. H.; Genet, Sylvia A. A. M.; Broeren, Maarten A. C.; van Dongen, Joost L. J.; Brunsveld, Luc; Scharnhorst, Volkher; van de Kerkhof, Daan
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Competitive protein recruitment in artificial cells
err2024-06-28
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errvan Veldhuisen, Thijs W.; Verwiel, Madelief A. M.; Novosedlik, Sebastian; Brunsveld, Luc; van Hest, Jan C. M.
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Crosstalk interactions between transcription factors ERR a and PPAR a assist PPAR a-mediated gene expression
err2024-06-01
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errDesmet, Sofie J.; Thommis, Jonathan; Vanderhaeghen, Tineke; Vandenboorn, Edmee M. F.; Clarisse, Dorien; Li, Yunkun; Timmermans, Steven; Fijalkowska, Daria; Ratman, Dariusz; Van Hamme, Evelien; De Cauwer, Lode; Staels, Bart; Brunsveld, Luc; Peelman, Frank; Libert, Claude; Tavernier, Jan; De Bosscher, Karolien
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14-3-3τ as a Modulator of Early α-Synuclein Multimerization and Amyloid Formation
err2024-04-18
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errHeesink, Gobert; van den Oetelaar, Maxime C. M.; Semerdzhiev, Slav A.; Ottmann, Christian; Brunsveld, Luc; Blum, Christian; Claessens, Mireille M. A. E.
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Functional Classification and Interaction Selectivity Landscape of the Human SH3 Domain Superfamily
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IF5.2
err2024-01-20
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errKazemein Jasemi, Neda S.; Mehrabipour, Mehrnaz; Magdalena Estirado, Eva; Brunsveld, Luc; Dvorsky, Radovan; Ahmadian, Mohammad R.
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Quantification of the lung cancer tumor marker CYFRA 21-1 using protein precipitation, immunoaffinity bottom-up LC-MS/MS
err2023-10-30
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errGenet, Sylvia A. A. M.; van den Wildenberg, Sebastian A. H.; Broeren, Maarten A. C.; van Dongen, Joost L. J.; Brunsveld, Luc; Scharnhorst, Volkher; van de Kerkhof, Daan
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Structure-Based Optimization of Covalent, Small-Molecule Stabilizers of the 14-3-3s/ERa Protein-Protein Interaction from Nonselective Fragments
err2023-09-07
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errKonstantinidou, Markella; Visser, Emira J.; Vandenboorn, Edmee; Chen, Sheng; Jaishankar, Priyadarshini; Overmans, Maurits; Dutta, Shubhankar; Neitz, R. Jeffrey; Renslo, Adam R.; Ottmann, Christian; Brunsveld, Luc; Arkin, Michelle R.
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From Tethered to Freestanding Stabilizers of 14-3-3 Protein-Protein Interactions through Fragment Linking
err2023-08-01
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errVisser, Emira J.; Jaishankar, Priyadarshini; Sijbesma, Eline; Pennings, Marloes A. M.; Vandenboorn, Edmee M. F.; Guillory, Xavier; Neitz, R. Jeffrey; Morrow, John; Dutta, Shubhankar; Renslo, Adam R.; Brunsveld, Luc; Arkin, Michelle R.; Ottmann, Christian
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