arrow
Back
A

Andrew B. Waight

discovery biologics, merck & co., inc., 213 east grand ave., south san francisco, ca 94080, usa

17H-index
73Paper Count
1.5KCitation Count
Published Papers 20
Publication Date
Structural Characterization of Linker Shielding in ADC Site-Specific Conjugates
err2025-12-05
err0
errOAAI
errMaru Jaime-Garza; Andrew Waight; Manish Hudlikar; Michael J. Eddins; Elnaz S. Rasti; Jan Paulo T. Zaragoza; Laurence Fayadat-Dilman; Jill E. Chrencik; Sandra B. Gabelli; Yun-Ting Chen; Cameron L. Noland
errShare
errSave
Biologics developability data analysis using hierarchical clustering accelerates candidate lead selection, optimization, and preformulation screening
errmAbs
IF7.3
err2025-05-10
err0
errOAAI
errKevin James Metcalf; Galen Wo; Jan Paulo Zaragoza; Fahimeh Raoufi; Jeanne Baker; Daoyang Chen; Mehabaw Derebe; Jason Hogan; Amy Hsu; Esther Kofman; David Leigh; Mandy Li; Dan Malashock; Cate Mann; Soha Motlagh; Jihea Park; Karthik Sathiyamoorthy; Madhura Shidhore; Yinyan Tang; Kevin Teng; Katharine Williams; Andrew Waight; Sultan Yilmaz; Fan Zhang; Huimin Zhong; Laurence Fayadat-Dilman; Marc Bailly
errShare
errSave
A machine learning strategy for the identification of key in silico descriptors and prediction models for IgG monoclonal antibody developability properties
errMABS
IF7.3
err2023-08-23
err9
errOAAI
errWaight, Andrew B.; Prihoda, David; Shrestha, Rojan; Metcalf, Kevin; Bailly, Marc; Ancona, Marco; Widatalla, Talal; Rollins, Zachary; Cheng, Alan C.; Bitton, Danny A.; Fayadat-Dilman, Laurence
errShare
errSave
BioPhi: A platform for antibody design, humanization, and humanness evaluation based on natural antibody repertoires and deep learning
errMABS
IF7.3
err2022-02-08
err71
errOAAI
errPrihoda, David; Maamary, Jad; Waight, Andrew; Juan, Veronica; Fayadat-Dilman, Laurence; Svozil, Daniel; Bitton, Danny A.
errShare
errSave
Engineering an Enhanced EGFR Engager: Humanization of Cetuximab for Improved Developability
err2022-01-13
err9
errOAAI
errGoulet, Dennis R.; Chatterjee, Soumili; Lee, Wai-Ping; Waight, Andrew B.; Zhu, Yi; Mak, Amanda Nga-Sze
errShare
errSave
Improving Antibody-Tubulysin Conjugates through Linker Chemistry and Site-Specific Conjugation
err2021-02-12
err9
errOAAI
errHamilton, Joseph Z.; Pires, Thomas A.; Mitchell, Jamie A.; Cochran, Julia H.; Emmerton, Kim K.; Zaval, Margo; Stone, Ivan J.; Anderson, Martha E.; Jin, Steven; Waight, Andrew B.; Lyon, Robert P.; Senter, Peter D.; Jeffrey, Scott C.; Burke, Patrick J.
errShare
errSave
Novel Auristatins with High Bystander and Cytotoxic Activities in Drug Efflux-positive Tumor Models
err2021-02-05
err18
errOAAI
errMoquist, Philip N.; Bovee, Tim D.; Waight, Andrew B.; Mitchell, Jamie A.; Miyamoto, Jamie B.; Mason, Marsha L.; Emmerton, Kim K.; Stevens, Nicole; Balasubramanian, Cindy; Simmons, Jessica K.; Lyon, Robert P.; Senter, Peter D.; Doronina, Svetlana O.
errShare
errSave
Antibody-drug conjugates of NAMPT inhibitors: Discovery, optimization, and preclinical characterization
err2019-07-01
err0
PREAI
errNeumann, Chris; Olivas, Kathleen C.; Wang, Kung Pern; Waight, Andrew B.; Meyer, David W.; Loftus, Luke V.; Zaval, Margo C.; Anderson, Martha E.; Jin, Steven; Cochran, Julia H.; Simmons, Jessica K.; Pittman, Paul G.; Li, Fu; Ulrich, Michelle L.; Wong, Abbie; Zeng, Weiping; Lyon, Robert P.; Senter, Peter D.
errShare
errSave
Targeted Delivery of Cytotoxic NAMPT Inhibitors Using Antibody-Drug Conjugates
err2018-12-03
err35
errOAAI
errNeumann, Christopher S.; Olivas, Kathleen C.; Anderson, Martha E.; Cochran, Julia H.; Jin, Steven; Li, Fu; Loftus, Luke, V; Meyer, David W.; Neale, Jason; Nix, Jay C.; Pittman, Paul G.; Simmons, Jessica K.; Ulrich, Michelle L.; Waight, Andrew B.; Wong, Abbie; Zaval, Margo C.; Zeng, Weiping; Lyon, Robert P.; Senter, Peter D.
errShare
errSave
Glucuronide-Linked Antibody-Tubulysin Conjugates Display Activity in MDR+ thorn and Heterogeneous Tumor Models
err2018-07-31
err17
errOAAI
errBurke, Patrick J.; Hamilton, Joseph Z.; Pires, Thomas A.; Lai, Holden W. H.; Leiske, Christopher I.; Emmerton, Kim K.; Waight, Andrew B.; Senter, Peter D.; Lyon, Robert P.; Jeffrey, Scott C.
errShare
errSave
Novel auristatins with high activity on efflux-positive models and demonstrable bystander activity
err2018-07-01
err0
PREAI
errMoquist, Philip N.; Bovee, Tim D.; Waight, Andrew B.; Owen, Sarah; Mitchell, Jamie A.; Zaval, Margo; Quick, Marsha; Sandall, Sharsti; Emmerton, Kim K.; Blesie, Nicole; Lyon, Robert P.; Senter, Peter; Doronina, Svetlana
errShare
errSave
Impact of linker and conjugation site on tubulysin M ADC stability and in vivo activity
err2018-07-01
err0
PREAI
errBurke, Patrick J.; Hamilton, Joseph Z.; Pires, Thomas A.; Leiske, Christopher I.; Cochran, Julia H.; Setter, Jocelyn R.; Emmerton, Kim K.; Waight, Andrew B.; Senter, Peter D.; Lyon, Robert P.; Jeffrey, Scott C.
errShare
errSave
Targeted delivery of cytotoxic NAMPT inhibitors using antibody-drug conjugates
err2018-07-01
err0
PREAI
errNeumann, Christopher S.; Olivas, Kathleen C.; Waight, Andrew B.; Meyer, David; Loftus, Luke V.; Zaval, Margo; Anderson, Martha E.; Jin, Steven; Cochran, Julia H.; Simmons, Jessica K.; Pittman, Paul G.; Lyon, Robert P.; Senter, Peter D.
errShare
errSave
Cysteine mutant location affects chemotype lability in site-specific antibody drug conjugates
err2017-07-01
err0
PREAI
errWaight, Andrew; Leiske, Chris; Biechele, Travis; Burke, Patrick; Rohm, Rory; Senter, Peter; Benjamin, Dennis; Sussman, Django
errShare
errSave
Development of Novel Quaternary Ammonium Linkers for Antibody-Drug Conjugates
err2016-05-05
err66
errOAAI
errBurke, Patrick J.; Hamilton, Joseph Z.; Pires, Thomas A.; Setter, Jocelyn R.; Hunter, Joshua H.; Cochran, Julia H.; Waight, Andrew B.; Gordon, Kristine A.; Toki, Brian E.; Emmerton, Kim K.; Zeng, Weiping; Stone, Ivan J.; Senter, Peter D.; Lyon, Robert P.; Jeffrey, Scott C.
errShare
errSave
Mechanism of inhibition of human glucose transporter GLUT1 is conserved between cytochalasin B and phenylalanine amides
err2016-04-12
err168
errOAAI
errKapoor, Khyati; Finer-Moore, Janet S.; Pedersen, Bjorn P.; Caboni, Laura; Waight, Andrew; Hillig, Roman C.; Bringmann, Peter; Heisler, Iring; Mueller, Thomas; Siebeneicher, Holger; Stroud, Robert M.
errShare
errSave
errShare
errSave
Ion selectivity and gating mechanisms of FNT channels
err2013-08-01
err19
errOAAI
errWaight, Andrew B.; Czyzewski, Bryan K.; Wang, Da-Neng
errShare
errSave
Structure and mechanism of a pentameric formate channel
err2009-12-13
err87
errOAAI
errWaight, Andrew B.; Love, James; Wang, Da-Neng
errShare
errSave
Discovery of a new phosphotyrosine mimetic for PTP1B using breakaway tethering
err2003-04-18
err56
PREAI
errErlanson, DA; McDowell, RS; He, MM; Randal, M; Simmons, RL; Kung, J; Waight, A; Hansen, SK
errShare
errSave