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Raymond F. Schinazi

 emory university

87H-index
876Paper Count
3.4WCitation Count
Published Papers 293
Publication Date
Phospholipid-driven conformational switching of HCV NS5A links protein folding to replication membrane remodeling
err2026-04-03
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errOAAI
errAnna V. Bulankina; Rebecca M. Richter; James H. Nettles; Daisuke Yamane; Christian Grimm; Yasaman Karami; Richard A. Stanton; Bianca Introini; Jonas Hermann; Hanaa Charif; Mia S. König; Claudia Stroß; Cristina Ortiz; Nico Kraus; Daniel Wood; Facundo Galceran; Rupert Abele; Bernard Maigret; Raymond F. Schinazi; Stefan Zeuzem; Ricardo M. Biondi; MinKyung Yi; Robert Tampé; Mikhail Kudryashev; Christoph Welsch
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The 2′-α-Fluoro,2′-β-Bromo uridine phosphoramidate prodrug (2-BFU) reduces dengue virus replication and attenuates infection-induced thrombocytopenia In Vivo
err2026-03-02
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errOAAI
errAngélica Samer Lallo Dias; Felipe Rocha da Silva Santos; Jenniffer Ramos Martins; Viviane Lima Batista; Talita Cristina Martins da Fonseca; Leticia Pereira Soldati; Celso Martins Queiroz-Junior; Franck Amblard; Raymond F. Schinazi; Mauro Martins Teixeira; Vivian Vasconcelos Costa
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Novel Dimeric Capsid Assembly Modulators as a Unique Class of Highly Potent Anti-HBV Agents
err2025-11-01
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PREAI
errAmblard, Franck; Chen, Zhe; Kra, Kalouna; Patel, Dharmeshkumar; Bassit, Leda; Gargowitsch, Laetitia; Degrouard, Jeril; Rat, Virgile; Arteni, Ana-Andreea; Matthews, Lauren; Ravichandran, Shreya M.; Jiang, Alfred; Athanasiadis, Antonis; Dangas, Georgios; Abate, Maedot; Tresset, Guillaume; Pronost, Julien; Salman, Mohammad; Verma, Kiran; Kirby, Karen A.; Michailidis, Eleftherios; de Rocquigny, Hugues; Durantel, David; Bressanelli, Stephane; Sarafianos, Stefan G.; Schinazi, Raymond F.
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The structural and mechanistic bases for the viral resistance to allosteric HIV-1 integrase inhibitor pirmitegravir (vol 15, pg e00465, 2024)
errMBIO
IF4.7
err2025-11-01
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PREAI
errDinh, Tung; Tber, Zahira; Rey, Juan S.; Mengshetti, Seema; Annamalai, Arun S.; Haney, Reed; Briganti, Lorenzo; Amblard, Franck; Fuchs, James R.; Cherepanov, Peter; Kim, Kyungjin; Schinazi, Raymond F.; Perilla, Juan R.; Kim, Baek; Kvaratskhelia, Mamuka
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1′-Cyanocytidine-5′-isobutyryl is a potent SARS-CoV-2 inhibitor in culture and infected Syrian hamsters
err2025-10-03
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PREAI
errFranck Amblard; Mahesh Kasthuri; Julia C. LeCher; Sijia Tao; Ramyani De; Rana Abdelnabi; Ingrid Marko; Longhu Zhou; Chengwei Li; Junxing Shi; Shu Ling Goh; Jessica Downs-Bowen; Leda Bassit; Selwyn Hurwitz; Keivan Zandi; Tamara McBrayer; Birgit Weynand; Kenneth A. Johnson; Johan Neyts; Raymond F. Schinazi
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Addition of hydroxyurea (hydroxycarbamide) enhances the efficacy of fludarabine/cytarabine-based salvage regimens against acute myeloid leukaemia
err2025-09-27
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errOAAI
errIngrid Lilienthal; Sijia Tao; Christer Nilsson; Elory Leonard; Runqing Zhang; Agnes L. Sorteberg; Louisa Fredrikson; Ioanna Xagoraris; Shahrzad Shirazi Fard; Nikolaos Tsesmetzis; Vasilios Zachariadis; Huan Cai; Lakshmi Sandhow; Anette Langebäck; Anna Bohlin; Katja Pokrovskaja Tamm; Sofia Bengtzén; Raymond F. Schinazi; Sören Lehmann; Baek Kim; Georgios Z. Rassidakis; Hong Qian; Martin Jädersten; Nikolas Herold
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Discovery of broad-spectrum antivirals targeting viral proteases using in silico structural modeling and cellular analysis
err2025-07-29
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PREAI
errDharmeshkumar Patel; Ramyani De; Niloufar Azadi; Sujin Lee; Savannah Shooter; Sarah Amichai; Shaoman Zhou; Danielle Monroe; Cameron Mahanke; Tamara R. McBrayer; Michael Muczynski; Abdullah Al-Homoudi; Joseph Engel; Yury A. Bochkov; James E. Gern; Ladislau C. Kovari; Franck Amblard; Raymond F. Schinazi
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Combating yellow fever virus with 7-deaza-7-fluoro-2′-C-methyladenosine
err2025-04-01
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errOAAI
errLecher, Julia C.; Costa, Vivian Vasconcelos; Rust, Lauren N.; Bassit, Leda C.; Patel, Dharmeshkumar; Rezaei, Sahar; Moua, Justin; Santos, Felipe Rocha da Silva; Goncalves, Matheus Rodrigues; Queroz Jr, Celso Martins; Marim, Fernanda Martins; Zhou, Longhu; Lee, Sujin; Mcbrayer, Tamara; De, Ramyani; Azadi, Niloufar; Salman, Mohammad; Zandi, Keivan; Amblard, Franck; Burwitz, Benjamin; Teixeira, Mauro M.; Schinazi, Raymond F.
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Safety, pharmacokinetics, and biological activity of CD4-mimetic BNM-III-170 in SHIV-infected rhesus macaques
err2025-04-01
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errOAAI
errViox, Elise G.; Richard, Jonathan; Grandea, Andres G., III; Nguyen, Kevin; Harper, Justin; Auger, James; Ding, Shilei; Gasser, Romain; Prevost, Jeremie; Marchitto, Lorie; Medjahed, Halima; Bourassa, Catherine; Gaudette, Fleur; Pagliuzza, Amelie; Trifone, Cesar Ariel; Gavegnano, Christina; Hurwitz, Selwyn J.; Park, Jun; Clark, Natasha M.; Hammad, Iman; Capuano III, Saverio; Martin, Malcolm A.; Schinazi, Raymond F.; Silvestri, Guido; Kulpa, Deanna A.; Kumar, Priti; Chomont, Nicolas; Pazgier, Marzena; Smith III, Amos B.; Sodroski, Joseph; Evans, David T.; Finzi, Andres; Paiardini, Mirko
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Reader comment on: Comprehensive genotoxicity and carcinogenicity assessment of molnupiravir
err2024-12-18
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PREAI
errFrederick, Clay B.; Schinazi, Raymond F.; Swanstrom, Ronald
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The Discovery and Preclinical Profile of ALG-000184, a Prodrug of the Potent Hepatitis B Virus Capsid Assembly Modulator ALG-001075
err2024-11-22
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PREAI
errVendeville, Sandrine; Amblard, Franck; Bassit, Leda; Beigelman, Leonid N.; Blatt, Lawrence M.; Chen, Xiaoyuan; Chou, Lang; Kum, Dieudonne Buh; Chanda, Sushmita; Deval, Jerome; Geng, Xiu; Gupta, Kusum; Jekle, Andreas; Hu, Haiyang; Hu, Xiaojuan; Kang, Hyunsoon; Liu, Cheng; Liu, Jyanwei; Mcgowan, David C.; Misner, Dinah L.; Raboisson, Pierre; Sanchez, Abel Acosta; Serebryany, Vladimir; Stoycheva, Antitsa D.; Symons, Julian A.; Tan, Hua; Vanrusselt, Hannah; Williams, Caroline; Welch, Michael; Zhang, Liangliang; Zhang, Qingling; Zhang, Yafeng; Schinazi, Raymond F.; Smith, David B.; Debing, Yannick
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The structural and mechanistic bases for the viral resistance to allosteric HIV-1 integrase inhibitor pirmitegravir
errMBIO
IF4.7
err2024-11-13
err0
errOAAI
errDinh, Tung; Tber, Zahira; Rey, Juan S.; Mengshetti, Seema; Annamalai, Arun S.; Haney, Reed; Briganti, Lorenzo; Amblard, Franck; Fuchs, James R.; Cherepanov, Peter; Kim, Kyungjin; Schinazi, Raymond F.; Perilla, Juan R.; Kim, Baek; Kvaratskhelia, Mamuka
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Cannabinoid-Inspired Inhibitors of the SARS-CoV-2 Coronavirus 2′-O-Methyltransferase (2′-O-MTase) Non-Structural Protein (Nsp10-16)
err2024-10-28
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errBenjamin, Menny M.; Hanna, George S.; Dickinson, Cody F.; Choo, Yeun-Mun; Wang, Xiaojuan; Downs-Bowen, Jessica A.; De, Ramyani; Mcbrayer, Tamara R.; Schinazi, Raymond F.; Nielson, Sarah E.; Hevel, Joan M.; Pandey, Pankaj; Doerksen, Robert J.; Townsend, Danyelle M.; Zhang, Jie; Ye, Zhiwei; Wyer, Scott; Bialousow, Lucas; Hamann, Mark T.
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Why Certain Repurposed Drugs Are Unlikely to Be Effective Antivirals to Treat SARS-CoV-2 Infections
err2024-04-22
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errOAAI
errHurwitz, Selwyn J.; De, Ramyani; Lecher, Julia C.; Downs-Bowen, Jessica A.; Goh, Shu Ling; Zandi, Keivan; Mcbrayer, Tamara; Amblard, Franck; Patel, Dharmeshkumar; Kohler, James J.; Bhasin, Manoj; Dobosh, Brian S.; Sukhatme, Vikas; Tirouvanziam, Rabindra M.; Schinazi, Raymond F.
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Biophysics-Guided Lead Discovery of HBV Capsid Assembly Modifiers
err2024-04-02
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errOAAI
errFan, Zixing; Pavlova, Anna; Jenkins, Matthew C.; Bassit, Leda; Salman, Mohammad; Lynch, Diane L.; Patel, Dharmeshkumar; Korablyov, Maksym; Finn, M. G.; Schinazi, Raymond F.; Gumbart, James C.
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Synthesis and biological evaluation of novel peptidomimetic inhibitors of the coronavirus 3C-like protease
err2024-03-01
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PREAI
errAmblard, Franck; Lecher, Julia C.; De, Ramyani; Zhou, Shaoman; Liu, Peng; Goh, Shu Ling; Tao, Sijia; Patel, Dharmeshkumar; Downs-Bowen, Jessica; Zandi, Keivan; Zhang, Huanchun; Chaudhry, Gitika; McBrayer, Tamara; Muczynski, Michael; Al-Homoudi, Abdullah; Engel, Joseph; Lan, Shuiyun; Sarafianos, Stefan G.; Kovari, Ladislau C.; Schinazi, Raymond F.
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Biochemical and structural characterization of second-generation inhibitors targeting the SARS-CoV-2 3CL protease
err2024-03-01
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PREAI
errMuczynski, Michael; Engel, Joseph; Amblard, Franck; Patel, Dharmeshkumar; Schinazi, Raymond; Kovari, Ladislau
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Direct Synthesis of Aryloxy Phosphonamidate Nucleotide Prodrugs Using the Cross Metathesis Assisted by Ultrasonic Irradiation
err2024-02-21
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PREAI
errChoi, Se Myeong; Nam, Ye Eun; An, Yeon Jin; Choi, Eun Rang; Park, Hyejin; Schinazi, Raymond F.; Cho, Jong Hyun
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