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Robert A. Everley

2nd floor

29H-index
59Paper Count
3.3KCitation Count
Published Papers 34
Publication Date
A practical method for determining the rate of covalent modification of fragments and leads
err2025-12-18
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errOAAI
errJanice Jeon; Svetlana A. Kholodar; Brian H. Tran; Kimberly E. Mallinger; Daniel A. Erlanson; Robert A. Everley
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Structural basis for DCAF2 as a novel E3 ligase for PROTAC-mediated targeted protein degradation
err2025-10-03
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PREAI
errEvan J. McMahon; Alexander G. Cioffi; Patrick R. Visperas; Yueqing Lin; Michael Shaghafi; Courtney M. Daczkowski; Johannes C. Hermann; Robert A. Everley; Richard M. Neve; Daniel A. Erlanson; Kevin R. Webster; Vikram Narayan; Weiru Wang
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Corrigendum to “Comprehensive Proteomics Metadata and Integrative Web Portals Facilitate Sharing and Integration of LINCS Multiomics Data”
err2025-08-07
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PREAI
errDušica Vidović; Behrouz Shamsaei; Stephan C. Schürer; Phillip Kogan; Szymon Chojnacki; Michal Kouril; Mario Medvedovic; Wen Niu; Evren U. Azeloglu; Marc R. Birtwistle; Yibang Chen; Tong Chen; Jens Hansen; Bin Hu; Ravi Iyengar; Gomathi Jayaraman; Hong Li; Tong Liu; Eric A. Sobie; Yuguang Xiong; Matthew J. Berberich; Gary Bradshaw; Mirra Chung; Robert A. Everley; Ben Gaudio; Marc Hafner; Marian Kalocsay; Caitlin E. Mills; Maulik K. Nariya; Peter K. Sorger; Kartik Subramanian; Chiara Victor; Maria Banuelos; Victoria Dardov; Ronald Holewinski; Danica-Mae Manalo; Berhan Mandefro; Andrea D. Matlock; Loren Ornelas; Dhruv Sareen; Clive N. Svendsen; Vineet Vaibhav; Jennifer E. Van Eyk; Vidya Venkatraman; Steve Finkbiener; Ernest Fraenkel; Jeffrey Rothstein; Leslie Thompson; Jacob Asiedu; Steven A. Carr; Karen E. Christianson; Desiree Davison; Deborah O. Dele-Oni; Katherine C. DeRuff; Shawn B. Egri; Alvaro Sebastian Vaca Jacome; Jacob D. Jaffe; Daniel Lam; Lev Litichevskiy; Xiaodong Lu; James Mullahoo; Adam Officer; Malvina Papanastasiou; Ryan Peckner; Caidin Toder; Joel Blanchard; Michael Bula; Tak Ko; Li-Huei Tsai; Jennie Z. Young; Vagisha Sharma; Jarek Meller; Michael J. MacCoss
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Discovery of FMC-376 a novel orally bioavailable inhibitor of activated KRASG12C
err2023-04-04
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PREAI
errPatel, Snahel; Bhhatarai, Barun; Calses, Philamer; Erlanson, Daniel; Everley, Robert; Fong, Susan; Gerken, Phil; Hermann, Johannes C.; Le, Tiep; Liu, Li-kai; McMahon, Evan; Neve, Richard M.; Phan, Tony; Roberts, Allison; Shanafelt, Mikayla; Siemsgluess, Sophie; Staunton, Jocelyn; Wang, Yan; Wang, Weiru; Williams, Monika; Webster, Kevin R.
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Combining chemoproteomics with machine learning identifies functionally active covalent fragments for hard-to-drug cancer drivers
err2023-04-04
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PREAI
errHermann, Johannes C.; Everley, Robert; Marholz, Laura; Berberich, Matthew; Yang, Tzu-Yi; Chao, Yu-Hsin; Awol, Abduselam K.; Shaghafi, Michael; Yoon, Han; Varma, Rohan; Stein, Reed; Krug, Karsten; Lachtara, Emily; Erlanson, Daniel; Varma, Chris; Webster, Kevin R.
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Tandem mass tag-based quantitative proteomic profiling identifies candidate serum biomarkers of drug-induced liver injury in humans
err2023-03-03
err15
errOAAI
errRavindra, Kodihalli C.; Vaidya, Vishal S.; Wang, Zhenyu; Federspiel, Joel D.; Virgen-Slane, Richard; Everley, Robert A.; Grove, Jane I.; Stephens, Camilla; Ocana, Mireia F.; Robles-Diaz, Mercedes; Isabel Lucena, M.; Andrade, Raul J.; Atallah, Edmond; Gerbes, Alexander L.; Weber, Sabine; Cortez-Pinto, Helena; Fowell, Andrew J.; Hussaini, Hyder; Bjornsson, Einar S.; Patel, Janisha; Stirnimann, Guido; Verma, Sumita; Elsharkawy, Ahmed M.; Griffiths, William J. H.; Hyde, Craig; Dear, James W.; Aithal, Guruprasad P.; Ramaiah, Shashi K.
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A Comparison of Two Stability Proteomics Methods for Drug Target Identification in OnePot 2D Format
err2021-08-10
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PREAI
errXu, Yingrong; West, Graham M.; Abdelmessih, Mario; Troutman, Matthew D.; Everley, Robert A.
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Multiomics Profiling Establishes the Polypharmacology of FDA-Approved CDK4/6 Inhibitors and the Potential for Differential Clinical Activity
err2019-08-01
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errOAAI
errHafner, Marc; Mills, Caitlin E.; Subramanian, Kartik; Chen, Chen; Chung, Mirra; Boswell, Sarah A.; Everley, Robert A.; Liu, Changchang; Walmsley, Charlotte S.; Juric, Dejan; Sorger, Peter K.
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Multi-omics profiling establishes the polypharmacology of FDA Approved CDK4/6 inhibitors and its impact on drug response
err2019-07-01
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PREAI
errMills, Caitlin E.; Hafner, Marc A.; Subramanian, Kartik; Chen, Chen; Chung, Mirra; Boswell, Sarah A.; Everley, Robert A.; Liu, Changchang; Walmsley, Charlotte S.; Juric, Dejan; Sorger, Peter K.
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Leveraging Compound Promiscuity to Identify Targetable Cysteines within the Kinome
err2019-06-01
err42
errOAAI
errRao, Suman; Gurbani, Deepak; Du, Guangyan; Everley, Robert A.; Browne, Christopher M.; Chaikuad, Apirat; Tan, Li; Schroeder, Martin; Gondi, Sudershan; Ficarro, Scott B.; Sim, Taebo; Kim, Nam Doo; Berberich, Matthew J.; Knapp, Stefan; Marto, Jarrod A.; Westover, Kenneth D.; Sorger, Peter K.; Gray, Nathanael S.
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PF-06651600, a Dual JAK3/TEC Family Kinase Inhibitor
err2019-05-13
err115
PREAI
errXu, Hua; Jesson, Michael I.; Seneyiratne, Uthpala I.; Lin, Tsung H.; Shari, M. Nusrat; Xue, Liang; Nguyen, Chuong; Everley, Robert A.; Trujillo, John I.; Johnson, Douglas S.; Point, Gary R.; Thorarensen, Atli; Kilty, Lain; Telliez, Jean-Baptiste
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Adaptation of Human iPSC-Derived Cardiomyocytes to Tyrosine Kinase Inhibitors Reduces Acute Cardiotoxicity via Metabolic Reprogramming
err2019-05-01
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errOAAI
errWang, Huan; Sheehan, Robert P.; Palmer, Adam C.; Everley, Robert A.; Boswell, Sarah A.; Ron-Harel, Noga; Ringel, Alison E.; Holton, Kristina M.; Jacobson, Connor A.; Erickson, Alison R.; Maliszewski, Laura; Haigis, Marcia C.; Sorger, Peter K.
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The NAD+ Salvage Pathway Supports PHGDH-Driven Serine Biosynthesis
err2018-08-01
err54
errOAAI
errMurphy, J. Patrick; Giacomantonio, Michael A.; Paulo, Joao A.; Everley, Robert A.; Kennedy, Barry E.; Pathak, Gopal P.; Clements, Derek R.; Kim, Youra; Dai, Cathleen; Sharif, Tanveer; Gygi, Steven P.; Gujar, Shashi
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Role of Selenof as a Gatekeeper of Secreted Disulfide-Rich Glycoproteins
err2018-05-01
err52
errOAAI
errYim, Sun Hee; Everley, Robert A.; Schildberg, Frank A.; Lee, Sang-Goo; Orsi, Andrea; Barbati, Zachary R.; Karatepe, Kutay; Fomenko, Dmitry E.; Tsuji, Petra A.; Luo, Hongbo R.; Gygi, Steven P.; Sitia, Roberto; Sharpe, Arlene H.; Hatfield, Dolph L.; Gladyshev, Vadim N.
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Identification of translationally controlled tumor protein in promotion of DNA homologous recombination repair in cancer cells by affinity proteomics
err2017-08-28
err15
errOAAI
errLi, Y.; Sun, H.; Zhang, C.; Liu, J.; Zhang, H.; Fan, F.; Everley, R. A.; Ning, X.; Sun, Y.; Hu, J.; Liu, J.; Zhang, J.; Ye, W.; Qiu, X.; Dai, S.; Liu, B.; Xu, H.; Fu, S.; Gygi, S. P.; Zhou, C.
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Developing kinase inhibitors with polypharmacological profiles for the treatment of resistant cancers
err2017-07-01
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PREAI
errRao, Suman; Li, Tan; Everley, Robert; Du, Guangyan; Sorger, Peter; Gray, Nathanael
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Aminoglycoside-driven biosynthesis of selenium-deficient Selenoprotein P
err2017-06-29
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errOAAI
errRenko, Kostja; Martitz, Janine; Hybsier, Sandra; Heynisch, Bjoern; Voss, Linn; Everley, Robert A.; Gygi, Steven P.; Stoedter, Mette; Wisniewska, Monika; Koehrle, Josef; Gladyshev, Vadim N.; Schomburg, Lutz
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A Strategy to Combine Sample Multiplexing with Targeted Proteomics Assays for High-Throughput Protein Signature Characterization
err2017-01-01
err121
errOAAI
errErickson, Brian K.; Rose, Christopher M.; Braun, Craig R.; Erickson, Alison R.; Knott, Jeffrey; McAlister, Graeme C.; Wuhr, Martin; Paulo, Joao A.; Everley, Robert A.; Gygi, Steven P.
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Neutral Loss Is a Very Common Occurrence in Phosphotyrosine-Containing Peptides Labeled with Isobaric Tags
err2016-12-30
err23
errOAAI
errEverley, Robert A.; Huttlin, Edward L.; Erickson, Alison R.; Beausoleil, Sean A.; Gygi, Steven P.
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