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Nathanael S. Gray

stanford university

145H-index
1.5KPaper Count
8.5WCitation Count
Published Papers 443
Publication Date
A Type II CDK6 Degrader Enables Cellular Targeting beyond the Limits of Type II Inhibition
err2026-06-26
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errOAAI
errJi Hyeon Kim; Caitlin E. Mills; Zuzanna Kozicka; Daniel C. Scott; Cyrus Jin; Zixuan Jiang; Brendan G. Dwyer; Qixiang Geng; Sean T. Toenjes; Woong Sub Byun; Dina ElHarouni; Hongyu Li; Keith L. Ligon; Abby M. Thornhill; Hannah M. Jones; Bryan A. Romero; Stephen M. Hinshaw; Benjamin L. Ebert; Brenda A. Schulman; Katherine A. Donovan; Eric S. Fischer; Nathanael S. Gray
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Activating p53Y220C with a mutant-specific small molecule
err2026-05-02
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errOAAI
errXijun Zhu; Woong Sub Byun; Dominika Ewa Pieńkowska; Kha The Nguyen; Mengxiong Wang; Sabin A. Nettles; Sai Gourisankar; Nick A. Phillips; Jan Gerhartz; Qixiang Geng; Tian Qiu; Jianing Zhong; Zixuan Jiang; Roman C. Sarott; Stephen M. Hinshaw; Tinghu Zhang; Laura D. Attardi; Radosław P. Nowak; Nathanael S. Gray
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Correction: Discovery and optimization of tau targeted protein degraders enabled by patient induced pluripotent stem cells-derived neuronal models of tauopathy
err2026-04-07
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errOAAI
errMC M. Catarina Silva; GN Ghata Nandi; KA Katherine A. Donovan; QC Quan Cai; BC Bethany C. Berry; RP Radoslaw P. Nowak; ES Eric S. Fischer; NS Nathanael S. Gray †; FM Fleur M. Ferguson †; SJ Stephen J. Haggarty
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Charged molecular glue discovery enabled by targeted degron display
err2026-04-06
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errOAAI
errZhe Zhuang; Woong Sub Byun; Jakub Chrustowicz; Zuzanna Kozicka; Veronica L. Li; Dinah M. Abeja; Katherine A. Donovan; Sara Sepic; Inchul You; Mikołaj Słabicki; Eric S. Fischer; Stephen M. Hinshaw; Benjamin L. Ebert; Brenda A. Schulman; Nathanael S. Gray
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The protocol for a patient-driven online prospective European observational cohort aiming to determine risk factors for the development of psoriatic arthritis among people living with psoriasis: the HIPPOCRATES Prospective Observational Study
err2026-03-25
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PREAI
errTeresa Grohmann; Timeo Mtenga; David Kerr; Joe Barrett; Nathanael Gray; Heidi Bertheussen; Juan D. Cañete; Kurt de Vlam; Maarten de Wit; Theodoros Dimitroulas; Sam Groothuizen; Glenn Haugeberg; Mari Hoff; Rudolf Horváth; Jana Hurnakova; Michaela Koehm; Przemyslaw Kotyla; Jean-Guillaume Letarouilly; Rik Lories; Mari Løset; Christine Möser; Burkhard Möller; Maria Mytilinaiou; Mikkel Østergaard; Ana Rodrigues; Caitriona Ryan; Carlo Selmi; Liv Eidsmo; Axel Svedbom; Tiago Torres; Florentin Ananu Vreju; Marleen G. H. van de Sande; Lars Werner; Stephen R. Pennington; Oliver FitzGerald; Laura C. Coates
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A druggable redox switch on SHP1 controls macrophage inflammation
err2026-03-12
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PREAI
errMei Ying Ng; Meredith N. Nix; Guangyan Du; Ivan Davidek; Nils Burger; Sanghee Shin; Sean Toenjes; Haruna Takeda; Megan Cheah Xin Yan; Bingsen Zhang; Haopeng Xiao; Shelley M. Wei; Hyuk-Soo Seo; Sirano Dhe-Paganon; Thomas E. Wales; John R. Engen; Evanna L. Mills; Jianwei Che; Tinghu Zhang; Nathanael S. Gray; Edward T. Chouchani
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Degraders of the dengue virus capsid protein exhibit differentiated pharmacology relative to capsid inhibitors
err2026-02-10
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errOAAI
errAntara Chakravarty; Lu-Ning Wang; Ryan P. Golden; Zhengnian Li; Katherine A. Donovan; Oshri Afanzar; Yupeng Zhang; Eric S. Fischer; Nathanael S. Gray; Priscilla L. Yang
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Design and Development of DNA Damage Chemical Inducers of Proximity for Targeted Cancer Therapy
err2026-01-01
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PREAI
errQiu, Tian; Lee, Yeuan Ting; Dwyer, Brendan G.; Tan, Yi Jer; Chen, Ting; Romero, Bryan A.; Wang, Yanlan; Deng, Jiehui; Zhang, Tinghu; Crabtree, Gerald R.; Hinshaw, Stephen M.; Wong, Kwok-Kin; Gray, Nathanael S.
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Selective CDK6 Degradation via the KLHDC2 E3 Ubiquitin Ligase
err2025-12-01
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PREAI
errJeon, Eunhye; Kim, Younghoon; Ahn, Hyunwoo; Martinez, Michael J.; Hwang, Kyubin; Cho, Soyeong; Dwyer, Brendan G.; Romero, Bryan A.; Hinshaw, Stephen M.; Gray, Nathanael S.; Sim, Taebo
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Structural basis for the recruitment and selective phosphorylation of Akt by mTORC2
errScience
IF45.8
err2025-11-27
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PREAI
errMartin S. Taylor; Maggie Chen; Matthew Hancock; Maximilian Wranik; Bryant D. Miller; Timothy R. O’Meara; Brad A. Palanski; Scott B. Ficarro; Brian J. Groendyke; Yufei Xiang; Kazuma T. Kondo; Karen Y. Linde-Garelli; Michelle J. Lee; Dibyendu Mondal; Daniel Freund; Samantha Congreve; Kaay Matas; Maximiliaan Hennink; Kera Xibinaku; Max L. Valenstein; Trevor van Eeuwen; Jarrod A. Marto; Andrej Sali; Yi Shi; Nathanael S. Gray; David M. Sabatini; Nam Chu; Kacper B. Rogala; Philip A. Cole
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Rewiring the Fusion Oncoprotein EWSR1::FLI1 in Ewing Sarcoma with Bivalent Small Molecules
err2025-11-27
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PREAI
errMichael J. Bond; Ryan P. Golden; Giulia DiGiovanni; Briana Howard; Roman C. Sarott; Basel A. Karim; Sai Gourisankar; Gabriela Alexe; Kenneth Ross; Hannah M. Jones; Brendan G. Dwyer; Nathanael S. Gray; Kimberly Stegmaier
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Inhibitors supercharge kinase turnover through native proteolytic circuits
errNature
IF48.5
err2025-11-26
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errOAAI
errNatalie S. Scholes; Martino Bertoni; Arnau Comajuncosa-Creus; Katharina Kladnik; Xuefei Guo; Fabian Frommelt; Matthias Hinterndorfer; Hlib Razumkov; Polina Prokofeva; Martin P. Schwalm; Florian Born; Sandra Roehm; Hana Imrichova; Brianda L. Santini; Eleonora Barone; Caroline Schätz; Miquel Muñoz i Ordoño; Severin Lechner; Andrea Rukavina; Iciar Serrano; Miriam Abele; Anna Koren; Stefan Kubicek; Stefan Knapp; Nathanael S. Gray; Giulio Superti-Furga; Bernhard Kuster; Yigong Shi; Patrick Aloy; Georg E. Winter
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Development of FBXO22 Degraders and the Recruitment Ligand 2-Pyridinecarboxyaldehyde (2-PCA)
err2025-11-01
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PREAI
errQiu, Tian; Zhuang, Zhe; Byun, Woong Sub; Kozicka, Zuzanna; Baek, Kheewoong; Zhong, Jianing; Thornhill, Abby M.; Ryan, Julia K.; Donovan, Katherine A.; Fischer, Eric S.; Ebert, Benjamin L.; Gray, Nathanael S.
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Expanding the druggable zinc-finger proteome defines properties of drug-induced degradation
err2025-08-21
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errOAAI
errMikołaj Słabicki; Jiho Park; Radosław P. Nowak; Shourya S. Roy Burman; Jesse Pellman; Charles Zou; Hlib Razumkov; Jeannie Carreiro; Simran Rastogi; Anna Goldstein; Marek M. Nagiec; Katherine A. Donovan; Jianwei Che; Moritz Hunkeler; Qixiang Geng; Chi-Lin Hsu; Megha Lakshminarayan; Chelsea Shu; Rebecca L. Zon; Zuzanna Kozicka; Paul M.C. Park; Jonathan M. Tsai; Hojong Yoon; Lyn H. Jones; Adam S. Sperling; Nathanael S. Gray; Eric S. Fischer; Benjamin L. Ebert
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Unveiling the hidden interactome of CRBN molecular glues
err2025-07-24
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errOAAI
errKheewoong Baek; Rebecca J. Metivier; Shourya S. Roy Burman; Jonathan W. Bushman; Hojong Yoon; Ryan J. Lumpkin; Julia K. Ryan; Dinah M. Abeja; Megha Lakshminarayan; Hong Yue; Samuel Ojeda; Yuan Xiong; Jianwei Che; Alyssa L. Verano; Anna M. Schmoker; Nathanael S. Gray; Katherine A. Donovan; Eric S. Fischer
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Rational Design of CDK12/13 and BRD4 Molecular Glue Degraders
err2025-07-08
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PREAI
errDr. Zhe Zhuang; Dr. Woong Sub Byun; Dr. Zuzanna Kozicka; Dr. Katherine A. Donovan; Dr. Brendan G. Dwyer; Abby M. Thornhill; Hannah M. Jones; Zixuan Jiang; Xijun Zhu; Prof. Dr. Eric S. Fischer; Prof. Dr. Nicolas H. Thomä; Prof. Dr. Nathanael S. Gray
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Plasmodium falciparum protein kinase 6 and hemozoin formation are inhibited by a type II human kinase inhibitor exhibiting antimalarial activity
err2025-07-07
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PREAI
errFlore Nardella; Tiantian Jiang; Lushun Wang; Monica J. Bohmer; Subhoja Chakraborty; John Okombo; Jaeson Calla; Tatiane Macedo Silva; Samuel Pazicky; Jianwei Che; Jin Jeon; Evie Vincent; Nonlawat Boonyalai; Rachael Coyle; Mairi J. Buchanan; Samuel Schaefer; Daisy Chen; Amaan Khan; Emily Mayville; Mariana Laureano De Souza; Mayland Treat; Jordan Charlton; Patrick K. Tumwebaze; Seth Tjia; Lukas Montejo; Karen Cover; Philip J. Rosenthal; Roland A. Cooper; Zbynek Bozdech; Marcus C.S. Lee; Ratna Chakrabarti; Sanjay A. Desai; David A. Fidock; Jinhua Wang; Nathanael S. Gray; Elizabeth A. Winzeler; Debopam Chakrabarti
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Brain penetrant allosteric EGFR inhibitors for NSCLC David Scott;
err2024-12-09
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PREAI
errScott, David; Cullis, Courtney; Beyett, Tyler; Feru, Frederic; Gero, Thomas; Gipson, Krista; Gokhalle, Praful; Gray, Nathanael; Heppner, David; Huang, Sampson; Janne, Pasi; Pusalkar, Sandeepraj; Eck, Michael
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Exploration of the tunability of BRD4 degradation by DCAF16 trans-labelling covalent glues
err2024-12-01
err3
errOAAI
errHassan, Muhammad Murtaza; Li, Yen-Der; Ma, Michelle W.; Teng, Mingxing; Byun, Woong Sub; Puvar, Kedar; Lumpkin, Ryan; Sandoval, Brittany; Rutter, Justine C.; Jin, Cyrus Y.; Wang, Michelle Y.; Xu, Shawn; Schmoker, Anna M.; Cheong, Hakyung; Groendyke, Brian J.; Qi, Jun; Fischer, Eric S.; Ebert, Benjamin L.; Gray, Nathanael S.
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