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Rajshekhar Karpoormath

university of kwazulu-natal

35H-index
216Paper Count
3.8KCitation Count
Published Papers 77
Publication Date
Development of Isoniazid–Pyrazole Hybrids as Potential Antitubercular Agents
err2026-05-15
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errOAAI
errMukanda Gedeon Kadima; Vinayak Singh; Gobind Kumar; Sahil Mishra; Pule Seboletswe; Ankit; Afsana Kajee; Françoise Roquet-Banères; Laurent Kremer; Rajshekhar Karpoormath; Parvesh Singh
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An innovative electrochemical approach for forensic identification of saliva
err2026-03-17
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PREAI
errPriyanka Govender; John Alake; Afsana Kajee; Fernando Albericio; Beatriz G. de la Torre; Ashish Kumar; Darko Kwabena Adu; Meenu Ghai; Rajshekhar Karpoormath
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Iboga-Indole Alkaloids as Potential Plasmodial Inhibitors: Identification, Biosynthesis, and Molecular Docking Studies
err2025-10-01
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PREAI
errBabiaka, Smith B.; Lahngong, Methodius S.; Simoben, Conrad V.; Ongarora, Dennis S. B.; Chi, Godloves F.; Tshitenge, Dieudonne T.; Karpoormath, Rajshekhar; Rylands, Marwaan; Mbah, James A.; Abuga, Kennedy O.; Loveridge, E. Joel; Frederich, Michel
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New piperazine-sulfonamide-hydrazide and hydrazine hybrids: design, Synthesis, and antibacterial activity
err2025-09-24
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PREAI
errPankaj Sanjay Girase; Rina Soni; Jayashree V. Patil; Shubhangi S. Soman; Sithabile Mokoena; Rajshekhar Karpoormath; Ramandeep Singh
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Rational Design and Antimycobacterial Evaluation of Aryl Sulfonamide–Linked Isoniazid Hydrazones Against Mycobacterium Tuberculosis
err2025-09-17
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errOAAI
errMukanda Gedeon Kadima; Sahil Mishra; Gobind Kumar; Pule Seboletswe; Afsana Kajee; Ankit; Françoise Roquet-Banères; Maëlle Foubert; Laurent Kremer; Rajshekhar Karpoormath; Parvesh Singh
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Rationally Designed InhA Inhibitors: A Comparative Anti-Tubercular Activity Study of Sulfonate Esters of Isoniazid Hydrazones and Their Structurally Flexible Benzyl Analogues
err2025-09-10
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errOAAI
errMukanda Gedeon Kadima; Sahil Mishra; Gobind Kumar; Pule Seboletswe; Françoise Roquet-Banères; Maëlle Foubert; Laurent Kremer; Rajshekhar Karpoormath; Parvesh Singh
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Synthesis, Characterization, and Bioactivity of Quinoxaline Thiazolotriazoles
err2025-09-01
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errOAAI
errMhlongo, Silungile; Senzani, Sibusiso; Islam, Shahidul; Olofinsan, Kolawole; Singh, Moganavelli; Nundkumar, Nirasha; Mokoena, Sithabile; Karpoormath, Rajshekhar; Koorbanally, Neil A.
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The association between antibiotic use in hospitals and residual antibiotic concentrations in hospital effluents: a pilot study
err2025-05-12
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errOAAI
errDeedat, Fatima Zahra; Faya, Andile Mbuso; Gumbi, Bhekumuzi Prince; Johnston, Deanne Mary Graham; Karpoormath, Rajshekhar; Essack, Sabiha Yusuf
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Pyridazinone: A privileged scaffold for synthetic and biomedical applications
err2025-04-01
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PREAI
errKushwaha, Babita; Kushwaha, Narva Deshwar; Shaik, Baji Baba; Chandrasekaran, Balakumar; Obakachi, Vincent A.; Mokoena, Sithabile; Mohite, Sachin Balaso; Karpoormath, Rajshekhar
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Synthesis, Anticancer Screening, and In Silico Evaluations of Thieno[2,3-c]pyridine Derivatives as Hsp90 Inhibitors
err2025-01-24
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errOAAI
errChandrasekaran, Balakumar; Bayan, Mohammad F.; Hmedat, Ali; Al-Jaidi, Bilal A.; Al-Tawalbeh, Deniz M.; Abuarqoub, Duaa; Rasras, Anas J.; Jaradat, Da'san M. M.; Dakkah, Abdel Naser; Hourani, Wafa; Karpoormath, Rajshekhar
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Assessing the efficacy of iso-mukaadial acetate and betulinic acid against selected Plasmodium falciparum glycolytic pathway proteins: in silico and in vitro studies
err2025-01-18
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errOAAI
errZuma, Lindiwe Khumbuzile; Pooe, Ofentse Jacob; Mabaso, Nonduduzo Hlengiwe; Alake, John; Obakachi, Vincent A.; Yakobi, Sinethemba; Gasa, Nothando; Karpoormath, Rajshekhar; Simelane, Mthokozisi
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A promising class of antiprotozoal agents, design and synthesis of novel Pyrimidine-Cinnamoyl hybrids
err2025-01-01
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PREAI
errKayamba, Francis; Karpoormath, Rajshekhar; Obakachi, Vincent A.; Mahlalela, Mavela; Banda, Danny; van Zyl, Robyn L.; Lala, Sahil; Zininga, Tawanda; Shonhai, Addmore; Shaik, Baji Baba; Pooe, Ofentse J.
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Development of Water-Soluble Nanoformulations of Novel Pyrazolone Derivatives and the Evaluation of Their Antibacterial and Antioxidant Activities
err2024-12-26
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errOAAI
errIgbokwe, Nkeiruka N.; Ismail, Eman A.; Obakachi, Vincent A.; Ntsethe, Aviwe; Gamede, Mlindeli; Karpoormath, Rajshekhar; Faya, Mbuso A.
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Advances in Pyridine C-H Functionalizations: Beyond C2 Selectivity
err2024-12-10
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PREAI
errMohite, Sachin Balaso; Mirza, Yafia Kousin; Bera, Partha Sarathi; Nadigar, Siddaram; Yugendhar, Soorni; Karpoormath, Rajsekhar; Bera, Milan
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Computational, microscale thermophoresis and electrochemical study of a hepta-peptide for a simple, sensitive electrochemical biosensor for PSA
err2024-11-01
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PREAI
errAlake, John; Mahlalela, Mavela Cleopus; Mohite, Sachin; Partap, Sangh; Gafar, Mohammed A.; Adu, Darko Kwabena; Ike, Blessing Wisdom; Chauhan, Ruchika; Nate, Zondi; Karpoormath, Rajshekhar
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Computational simulation and fabrication of a simple, rapid and sensitive dopamine electrochemical sensor based on recycled biomass
err2024-11-01
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PREAI
errIke, Blessing Wisdom; Alake, John; Akintemi, Eric O.; Adu, Darko Kwabena; Nate, Zondi; Chauhan, Ruchika; Miya, Lungelo; Karpoormath, Rajshekhar; Faya, Mbuso
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One pot fabrication of diamino naphthalene -AuNPs decorated graphene nanoplatform for the MRSA detection in the biological sample
err2024-06-01
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PREAI
errChauhan, Ruchika; Nate, Zondi; Ike, Blessing; Adu, Darko Kwabena; Alake, John; Gill, Atal A. S.; Miya, Lungelo; Thapliyal, Neeta Bachheti; Karpoormath, Rajshekhar
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Rapid and label-free A2 peptide epitope decorated CoFe2O4-C60 nanocomposite-based electrochemical immunosensor for detecting Visceral Leishmaniasis
err2024-06-01
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PREAI
errAdu, Darko Kwabena; Nate, Zondi; Alake, John; Ike, Blessing Wisdom; Mahlalela, Mavela Cleopus; Mohite, Sachin Balaso; Mokoena, Sithabile; Chauhan, Ruchika; Karpoormath, Rajshekhar
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Novel 4,5-dibromo-N-phenyl-1H-pyrrole-2-carboxamide Hybrids as Promising DNA Gyrase Inhibitors: Design, synthesis and antimicrobial evaluation
err2024-04-01
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PREAI
errMerugu, Srinivas Reddy; Mokoena, Sithabile; Obakachi, Vincent A.; Shaik, Baji Baba; Kushawaha, Babita; Kushwaha, Narva Deshwar; Ike, Blessing Wisdom; Palkar, Mahesh B.; Bonde, Chandrakant G.; Ganai, Ab Majeed; Chauhan, Ruchika; Kajee, Afsana; Ghai, Meenu; Kidwai, Saqib; Singh, Ramandeep; Karpoormath, Rajshekhar
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Electrochemical immunosensing of tumor markers
err2024-04-01
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PREAI
errPalakollu, Venkata Narayana; Reddy, Y. Veera Manohara; Shekh, Mehdihasan I.; Vattikuti, S. V. Prabhakar; Shim, Jaesool; Karpoormath, Rajshekhar
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