Not logged inIdentification and biological evaluation of benzimidazole-based compounds as novel TGFβR1 inhibitors
Tseng, Hui-Ju; Wu, Yi-Wen; Chen, Yan-Ling; Lin, Tony Eight; Fang-Chin, Yu-Ting; Wu, Yueh-Lin; Sung, Tzu-Ying; Yen, Shih-Chung; Hsieh, Jui-Hua; Hsu, Kai-Cheng; Pan, Shiow-Lin
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SaveExploring diarylheptanoid derivatives to target LIMK1 as potential agents against colorectal cancer
Chen, Liang-Chieh; Chang, Tung-Cheng; Tseng, Hui-Ju; Chu, Jung-Chun; Huang, Yun-Yi; Peng, Hao-Yuan; Kuo, Yi-Chen; Wu, Yi-Wen; Lin, Tony Eight; Yen, Shih-Chung; Hsu, Kai-Cheng; Huang, Wei-Jan; Pan, Shiow-Lin
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SaveConsensus Pharmacological Interactions for PLK2 Inhibitor Identification in Colorectal Cancer Treatment
Wu, Yi-Wen; Yang, Chun-Lin; Lin, Tony Eight; Yeh, Yun-Hsuan; Fang-Chin, Yu-Ting; Sung, Tzu-Ying; Yen, Shih-Chung; Hsieh, Jui-Hua; Chung, Cheng-Chih; Pan, Shiow-Lin; Hsu, Kai-Cheng
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SaveIdentification of pyrazole scaffold inhibitors targeting cyclin-dependent kinase 8 for potential use in pulmonary fibrosis
Lin, Tony Eight; Hsu, Kai-Cheng; Chou, Ching-Hsuan; Tsai, En-Yun; Wu, Yi-Wen; Sung, Tzu-Ying; Hsu, Jui-Yi; Hsieh, Jui-Hua; Yen, Shih-Chung; Chang, Yu-Wei; Pan, Shiow-Lin; Huang, Wei-Jan; Yang, Chia-Ron
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SaveIdentification and Biological Evaluation of a Novel CLK4 Inhibitor Targeting Alternative Splicing in Pancreatic Cancer Using Structure-Based Virtual Screening
Yang, CL; Wu, YW; Tu, HJ; Yeh, YH; Lin, TE; Sung, TY; Li, MC; Yen, SC; Hsieh, JH; Yu, MC; Hsieh, SY; Hsieh, HP; Pan, SL; Hsu, KC
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SaveIdentification of a Potent CDK8 Inhibitor Using Structure-Based Virtual Screening
Lin, Tony Eight; Chou, Ching-Hsuan; Wu, Yi-Wen; Sung, Tzu-Ying; Hsu, Jui-Yi; Yen, Shih-Chung; Hsieh, Jui-Hua; Chang, Yu-Wei; Pan, Shiow-Lin; Huang, Wei-Jan; Hsu, Kai-Cheng; Yang, Chia-Ron
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SaveIdentification, biological evaluation, and crystallographic analysis of coumestrol as a novel dual-specificity tyrosine-phosphorylation-regulated kinase 1A inhibitor
Peng, Chao-Hsiang; Hwang, Tsong-Long; Hung, Shao-Chi; Tu, Huang-Ju; Tseng, Yen-Tzu; Lin, Tony Eight; Lee, Cheng-Chung; Tseng, Yi-Chi; Ko, Chiung-Yuan; Yen, Shih-Chung; Hsu, Kai-Cheng; Pan, Shiow-Lin; Huangfu, Wei-Chun
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SaveDiscovery of novel TANK-Binding Kinase 1 (TBK1) inhibitor against pancreatic ductal adenocarcinoma
Shih, Wan-Hsi; Huang, Han-Li; Huangfu, Wei-Chun; Lin, Tony Eight; Sung, Tzu-Ying; Li, Mu-Chun; Huang, Guan-Lin; Chang, Yu-Wei; Yen, Shih-Chung; Hsieh, Hsing-Pang; Hsu, Kai-Cheng; Pan, Shiow-Lin
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SaveDiscovering a novel dual specificity tyrosine-phosphorylation-regulated kinase 1A (DYRK1A) inhibitor and its impact on tau phosphorylation and amyloid-β formation
Tu, Huang-Ju; Chao, Min-Wu; Lee, Cheng-Chung; Peng, Chao-Shiang; Wu, Yi-Wen; Lin, Tony Eight; Chang, Yu-Wei; Yen, Shih-Chung; Hsu, Kai-Cheng; Pan, Shiow-Lin; Huangfu, Wei-Chun
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SaveHSP90/LSD1 dual inhibitors against prostate cancer as well as patient-derived colorectal organoids
Tang, Di-Wei; Chen, I. -Chung; Chou, Po-Yu; Lai, Mei-Jung; Liu, Zheng-Yang; Tsai, Kelvin K.; Cheng, Li-Hsin; Zhao, Jian-Xun; Cho, Er-Chieh; Chang, Hung-Hsuan; Lin, Tony Eight; Hsu, Kai-Cheng; Chen, Mei-Chuan; Liou, Jing-Ping
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SaveFrom Sea to Science: Coral Aquaculture for Sustainable Anticancer Drug Development
Lin, Hung-Yu; Tsai, Tsen-Ni; Hsu, Kai-Cheng; Hsu, Yu-Ming; Chiang, Lin-Chien; El-Shazly, Mohamed; Chang, Ken-Ming; Lin, Yu-Hsuan; Tu, Shang-Yi; Lin, Tony Eight; Du, Ying-Chi; Liu, Yi-Chang; Lu, Mei-Chin
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SaveA novel HDAC8 inhibitor H7E exerts retinoprotective effects against glaucomatous injury via ameliorating aberrant Müller glia activation and oxidative stress
Wu, Liang-Huan; Cheng, Yu-Wen; Lin, Fan-Li; Hsu, Kai-Cheng; Wang, Mong-Heng; Yen, Jing -Lun; Wang, Tsung-Jen; Lin, Tony Eight; Liu, Yi-Chien; Huang, Wei-Jan; Hsiao, George
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SaveIdentification of selective dual-specificity tyrosine phosphorylation-regulated kinase 1A (DYRK1A) inhibitors and their effects on tau and microtubule
Wu, Yi-Wen; Huangfu, Wei-Chun; Lin, Tony Eight; Peng, Chao-Hsiang; Tu, Huang-Ju; Sung, Ting-Yi; Sung, Tzu-Ying; Yen, Shih-Chung; Pan, Shiow-Lin; Hsu, Kai-Cheng
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SaveDesign, synthesis, and biological activity of dual monoamine oxidase A and heat shock protein 90 inhibitors, N-Methylpropargylamine-conjugated 4-isopropylresorcinol for glioblastoma
Tseng, Hui-Ju; Banerjee, Suddhasatwa; Qian, Bin; Lai, Mei-Jung; Wu, Tung-Yun; Hsu, Tsung-, I; Lin, Tony Eight; Hsu, Kai Cheng; Chuang, Kuo-Hsiang; Liou, Jing-Ping; Shih, Jean C.
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SaveSynthesis and biological evaluation of C-4 substituted phenoxazine-bearing hydroxamic acids with potent class II histone deacetylase inhibitory activities
Chu, Jung-Chun; Tseng, Hui-Ju; Lee, Sung-Bau; Hsu, Kai-Cheng; Hsin, Ling-Wei; Liang, Ru-Hao; Lin, Tony Eight; Gao, Nain-Chu; Chen, Liang-Chieh; Lu, Wan-Hsun; Wang, Andrew H. -J; Huang, Wei-Jan
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