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Vardan T. Karamyan

oakland university

25H-index
119Paper Count
2.3KCitation Count
Published Papers 53
Publication Date
Structural and functional dissection of human neurolysin through alanine-scanning mutagenesis
err2026-04-17
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PREAI
errHeba ElSayed ElZorkany; Asmaa Aly; Shiva Hadi Esfahani; Vardan T. Karamyan
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Discovery of a pyridine-piperazine-based small molecule that enhances the activity of peptidase neurolysin
err2026-02-03
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PREAI
errHeba ElSayed ElZorkany; Haya Kandil; Srinidhi Jayaraman; Asmaa Aly; Shiva Hadi Esfahani; Dhavalkumar Patel; Dennis Dannecker; Monika Maciag; Alyssa Paul; Kaitlin Lowran; Shikha Kumari; Samik Bose; David A. Ostrov; Colin G. Wu; Alex Dickson; Thomas J. Abbruscato; Paul C. Trippier; Benjamin J. Orlando; Vardan T. Karamyan
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Assessing the effects of antidepressant use on stroke recurrence and related outcomes in ischemic stroke patients: a propensity score matched analysis
err2025-03-12
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errOAAI
errAlamri, Faisal F.; Almarghalani, Daniyah A.; Alatawi, Yasser; Alraddadi, Eman A.; Babateen, Omar; Alayyafi, Ahmed; Almalki, Ziyad; Alsalhi, Khaled; Alzahrani, Khaled; Alghamdi, Ahmed; Aldera, Hussain; Karamyan, Vardan T.
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Evaluation of systemic and brain pharmacokinetic parameters for repurposing metformin using intravenous bolus administration
err2025-01-01
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errOAAI
errSharma, Sejal; Zhang, Yong; Patel, Dhavalkumar; Akter, Khondker Ayesha; Bagchi, Sounak; Sifat, Ali Ehsan; Nozohouri, Ehsan; Ahn, Yeseul; Karamyan, Vardan T.; Bickel, Ulrich; Abbruscato, Thomas J.
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Structural basis of divergent substrate recognition and inhibition of human neurolysin
err2024-08-08
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errOAAI
errShi, Ke; Bagchi, Sounak; Bickel, Jordis; Esfahani, Shiva H.; Yin, Lulu; Cheng, Tiffany; Karamyan, Vardan T.; Aihara, Hideki
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Imidazole Bioisostere Activators of Endopeptidase Neurolysin with Enhanced Potency and Metabolic Stability
err2024-03-29
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PREAI
errRahman, Md. Shafikur; Esfahani, Shiva Hadi; Zhang, Yong; Queen, Aarfa; Aljarrah, Manar; Kandil, Haya; Baez, Andrew; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C.
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Systemic and Brain Pharmacokinetics of Milnacipran in Mice: Comparison of Intraperitoneal and Intravenous Administration
err2023-12-29
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errOAAI
errBagchi, Sounak; Nozohouri, Ehsan; Ahn, Yeseul; Patel, Dhavalkumar; Bickel, Ulrich; Karamyan, Vardan T.
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Discovery of the Next Generation of Non-peptidomimetic Neurolysin Activators with High Blood-Brain Barrier Permeability: a Pharmacokinetics Study in Healthy and Stroke Animals
err2023-10-13
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PREAI
errZhang, Yong; Sharma, Sejal; Jonnalagadda, Shirisha; Kumari, Shikha; Queen, Aarfa; Esfahani, Shiva Hadi; Archie, Sabrina Rahman; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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High brain-blood barrier permeability highlights a new class of neurolysin activators as promising candidates for stroke treatment: a pilot pharmacokinetic study in mice
err2023-06-01
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errOAAI
errZhang, Yong; Sharma, Sejal; Esfahani, Shiva H.; Jonnalagadda, Shirisha; Queen, Aarfa; Nozohouri, Saeideh; Patel, Dhavalkumar; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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Translating Animal Models of Ischemic Stroke to the Human Condition
err2022-09-20
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PREAI
errMatur, Abhijith, V; Candelario-Jalil, Eduardo; Paul, Surojit; Karamyan, Vardan T.; Lee, Jessica D.; Pennypacker, Keith; Fraser, Justin F.
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Vitamin D serum level predicts stroke clinical severity, functional independence, and disability-A retrospective cohort study
err2022-07-27
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errOAAI
errAlharbi, Abdullah R.; Alali, Amer S.; Samman, Yahya; Alghamdi, Nouf A.; Albaradie, Omar; Almaghrabi, Maan; Makkawi, Seraj; Alghamdi, Saeed; Alzahrani, Mohammad S.; Alsalmi, Mohammed; Karamyan, Vardan T.; Al Sulaiman, Khalid; Aljuhani, Ohoud; Alamri, Faisal F.
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Estrogen Metabolite 2-Methoxyestradiol Attenuates Blood Pressure in Hypertensive Rats by Downregulating Angiotensin Type 1 Receptor
err2022-05-02
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errOAAI
errZhang, Yong; Ogola, Benard O.; Iyer, Laxmi; Karamyan, Vardan T.; Thekkumkara, Thomas
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Integrative epigenomic and transcriptomic analyses reveal metabolic switching by intermittent fasting in brain
err2022-03-31
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errOAAI
errNg, Gavin Yong-Quan; Sheng, Dominic Paul Lee Kok; Bae, Han-Gyu; Kang, Sung Wook; Fann, David Yang-Wei; Park, Jinsu; Kim, Joonki; Alli-Shaik, Asfa; Lee, Jeongmi; Kim, Eunae; Park, Sunyoung; Han, Jeung-Whan; Karamyan, Vardan; Okun, Eitan; Dheen, Thameem; Hande, Manoor Prakash; Vemuganti, Raghu; Mallilankaraman, Karthik; Lim, Lina H. K.; Kennedy, Brian K.; Drummond, Grant R.; Sobey, Christopher G.; Gunaratne, Jayantha; Mattson, Mark P.; Foo, Roger Sik-Yin; Jo, Dong-Gyu; Arumugam, Thiruma V.
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In-Vivo and Ex-Vivo Brain Uptake Studies of Peptidomimetic Neurolysin Activators in Healthy and Stroke Animals
err2022-03-03
err9
errOAAI
errNozohouri, Saeideh; Esfahani, Shiva Hadi; Noorani, Behnam; Patel, Dhaval; Villalba, Heidi; Ghanwatkar, Yashwardhan; Rahman, Md Shafikur; Zhang, Yong; Bickel, Ulrich; Trippier, Paul C.; Karamyan, Vardan T.; Abbruscato, Thomas J.
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Discovery of First-in-Class Peptidomimetic Neurolysin Activators Possessing Enhanced Brain Penetration and Stability (vol 64, pg 12705, 2021)
err2021-12-22
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errOAAI
errRahman, Md. Shafikur; Kumari, Shikha; Esfahani, Shiva Hadi; Nozohouri, Saeideh; Jayaraman, Srinidhi; Kinarivala, Nihar; Kocot, Joanna; Baez, Andrew; Farris, Delaney; Abbruscato, Thomas J.; Karamyan, Vardan T.; Trippier, Paul C.
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